中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [10]
采集方式
OAI收割 [10]
内容类型
期刊论文 [10]
发表日期
2019 [1]
2018 [2]
2016 [3]
2015 [3]
2014 [1]
学科主题
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Recyclable and Stable alpha-Methylproline-Derived Chiral Ligands for the Chemical Dynamic Kinetic Resolution of free C,N-Unprotected alpha-Amino Acids
期刊论文
OAI收割
MOLECULES, 2019, 卷号: 24, 期号: 12, 页码: 19
作者:
Shu, Shuangjie
;
Zhao, Liang
;
Zhou, Shengbin
;
Wu, Chenglin
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2020/07/01
quaternary carbon
dynamic kinetic resolution
unprotected alpha-amino acids
Schiff base intermediates
ligands
Discovery of thiophene-containing biaryl amide derivatives as novel glucagon receptor antagonists
期刊论文
OAI收割
CHEMICAL BIOLOGY & DRUG DESIGN, 2018, 卷号: 92, 期号: 1, 页码: 1241-1254
作者:
Li, Jia
;
Feng, Yang
;
Li, Huihui
;
Shu, Shuangjie
;
Dai, Antao
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2019/01/08
biaryl amide
glucagon receptor antagonist
molecular simulation
A novel series of 4-methyl substituted pyrazole derivatives as potent glucagon receptor antagonists: Design, synthesis and evaluation of biological activities
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1896-1908
作者:
Shu, Shuangjie
;
Dai, Antao
;
Wang, Jiang
;
Wang, Bin
;
Feng, Yang
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
Pyrazole derivatives
Glucagon receptor antagonist
Docking study
Binding pocket
Design, synthesis, structure-activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 12, 页码: 2852-2863
作者:
Shu, Shuangjie
;
Cai, Xiaoqing
;
Li, Jia
;
Feng, Yang
;
Dai, Antao
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2019/01/08
Glucagon receptor
Antagonist
Molecular docking
Pyrazole
Type 2 diabetes mellitus
Advanced asymmetric synthesis of (1R,2S)-1-amino-2-vinylcyclopropanecarboxylic acid by alkylation/cyclization of newly designed axially chiral Ni(II) complex of glycine Schiff base
期刊论文
OAI收割
AMINO ACIDS, 2016, 卷号: 48, 期号: 4, 页码: 973-986
作者:
Kawashima, Aki
;
Shu, Shuangjie
;
Takeda, Ryosuke
;
Kawamura, Akie
;
Sato, Tatsunori
  |  
收藏
  |  
浏览/下载:164/0
  |  
提交时间:2019/01/08
Anti-viral (HCV) activity
Asymmetric synthesis
Amino acids
Chirality
Schiff bases
Application of Sulfonyl in Drug Design
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 36, 期号: 3, 页码: 490-501
作者:
Zhao Fei
;
Wang Jiang
;
Ding Xiao
;
Shu Shuangjie
;
Liu Hong
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
sulfonyl
drug design
lead optimization
gamma-Carbon Activation through N-Heterocyclic Carbene/Bronsted Acids Cooperative Catalysis: A Highly Enantioselective Route to delta-Lactams
期刊论文
OAI收割
ORGANIC LETTERS, 2015, 卷号: 17, 期号: 15, 页码: 3850-3853
作者:
Xiao, Yonglong
;
Wang, Jinxin
;
Xia, Wenjing
;
Shu, Shuangjie
;
Jiao, Shenchao
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Palladium-Catalyzed C2-Acylation of Indoles with alpha-Diketones Assisted by the Removable N-(2-Pyrimidyl) Group
期刊论文
OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2015, 期号: 17, 页码: 3743-3750
作者:
Li, Chunpu
;
Zhu, Wei
;
Shu, Shuangjie
;
Wu, Xiaoming
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
Synthetic methods
Acylation
C-H activation
Palladium
Nitrogen heterocycles
Palladium-catalyzed intramolecular addition of C-N bond to alkynes: a novel approach to 3-diketoindoles
期刊论文
OAI收割
RSC Advances, 2015, 卷号: 5, 期号: 110, 页码: 90396-90399
作者:
Wu, Chenglin
;
Zhao, Fei
;
Shu, Shuangjie
;
Wang, Jiang
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
A simple copper-catalyzed two-step one-pot synthesis of indolo[1,2-a]quinazoline
期刊论文
OAI收割
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY, 2014, 卷号: 10, 页码: 2441-2447
作者:
Li, Chunpu
;
Zhang, Lei
;
Shu, Shuangjie
;
Liu, Hong
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
copper
one pot
synthetic methods