中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
地质与地球物理研究... [13]
上海药物研究所 [9]
西北高原生物研究所 [9]
上海光学精密机械研究... [5]
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武汉病毒研究所 [2]
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期刊论文 [41]
会议论文 [1]
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2024 [3]
2023 [2]
2020 [1]
2019 [2]
2017 [9]
2016 [2]
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Discovery of CZL-046 with an (
S
)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:
Chen, Zonglong
;
Yang, Hong
;
Zhang, Yan
;
Lyu, Xiaodong
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/05
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads
期刊论文
OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:
Dong, Sanfeng
;
Huang, Hui
;
Li, Jintian
;
Li, Xiaomei
;
Bunu, Samuel Jacob
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/10/21
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/02/19
Multiple myeloma
TRIP13 inhibitor
Cantharidin
DCZ5418
DCZ0415
Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:
Wang, Yujie
;
Xu, Keshi
;
Liu, Hongchun
;
Zhang, Wei
;
Hu, Chun
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/12/19
Auristatin E
beta-Glucuronidase
Antiproliferation
Tumor microenvironment
Geology, geochronology, and geochemistry of the Gaojiabang tungsten-molybdenum deposit, Anhui Province, Southeast China
期刊论文
OAI收割
ORE GEOLOGY REVIEWS, 2023, 卷号: 157, 页码: 28
作者:
Zheng, Fangshun
;
Qin, Kezhang
;
Cook, Nigel J.
;
Li, Guangming
;
Ciobanu, Cristiana L.
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/12/29
Gaojiabang
Alteration stages
Porphyry-skarn type deposit
W-Mo mineralization
Ductile deformations
Qingyang-Jiuhua Complex
Investigation of the remote acyl group participation in glycosylation from conformational perspectives by using trichloroacetimidate as the acetyl surrogate
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2020, 卷号: 7, 期号: 13, 页码: 1606-1615
作者:
Xu, Ke
;
Man, Qingmin
;
Zhang, Yang
;
Guo, Jia
;
Liu, Yichu
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/12/24
Structural optimization and neurotrophic activity evaluation of neurotrophic gentiside derivatives
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 22, 页码: 6
作者:
Wang, Zhenkang
;
Ma, Chunhua
;
Wang, Yujie
;
Xiao, Qiang
;
Xu, Chenghui
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2020/07/01
Gentisides
Neurotrophic activity
Isosteric replacement
Conformational restriction
PC 12 cells
Scheelite geochemistry in porphyry-skarn W-Mo systems: A case study from the Gaojiabang Deposit, East China
期刊论文
OAI收割
ORE GEOLOGY REVIEWS, 2019, 卷号: 113, 页码: 17
作者:
Song, Guoxue
;
Cook, Nigel J.
;
Li, Guangming
;
Qin, Kezhang
;
Ciobanu, Cristiana L.
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/05/18
Scheelite
Substitution mechanism
Redox state
Sr-isotopes
Porphyry-skarn system
Gaojiabang deposit
CASCIRE surveillance network and work on avian influenza viruses
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2017
Bi, Yuhai
;
Shi, Weifeng
;
Chen, Jianjun
;
Chen, Quanjiao
;
Ma, Zhenghai
;
Wong, Gary
;
Tian, Wenxia
;
Yin, Renfu
;
Fu, Guanghua
;
Yang, Yongchun
;
Liu, William J.
;
Quan, Chuansong
;
Wang, Qianli
;
He, Shenghu
;
Li, Xiangdong
;
Xia, Qianfeng
;
Wang, Lixin
;
Pan, Zhaohui
;
Li, Laixing
;
Li, Hong
;
Xu, Wen
;
Luo, Ying
;
Zeng, Hui
;
Dai, Lianpan
;
Xiao, Haixia
;
Sharshov, Kirill
;
Shestopalov, Alexander
;
Shi, Yi
;
Yan, Jinghua
;
Li, Xuebing
;
Liu, Yingxia
;
Lei, Fumin
;
Liu, Wenjun
;
Gao, George F.
  |  
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2019/06/14
CASCIRE surveillance network and work on avian influenza viruses
期刊论文
OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2017
Bi, Yuhai
;
Shi, Weifeng
;
Chen, Jianjun
;
Chen, Quanjiao
;
Ma, Zhenghai
;
Wong, Gary
;
Tian, Wenxia
;
Yin, Renfu
;
Fu, Guanghua
;
Yang, Yongchun
;
Liu, William J.
;
Quan, Chuansong
;
Wang, Qianli
;
He, Shenghu
;
Li, Xiangdong
;
Xia, Qianfeng
;
Wang, Lixin
;
Pan, Zhaohui
;
Li, Laixing
;
Li, Hong
;
Xu, Wen
;
Luo, Ying
;
Zeng, Hui
;
Dai, Lianpan
;
Xiao, Haixia
;
Sharshov, Kirill
;
Shestopalov, Alexander
;
Shi, Yi
;
Yan, Jinghua
;
Li, Xuebing
;
Liu, Yingxia
;
Lei, Fumin
;
Liu, Wenjun
;
Gao, George F.
  |  
收藏
  |  
浏览/下载:100/0
  |  
提交时间:2019/07/05