中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共155条,第1-10条 帮助

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Heterocycle-fused phenylcyclohexylamines as novel multi-target antagonists of N-methyl-D-aspartate (NMDA) receptor and monoamine transporter for treating depression 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 20
作者:  
Zheng, Fuqiang;  Hu, Zhengtao;  Chen, Hai;  Cheng, Jiaxin;  Hou, Qiongqiong
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Design, Synthesis, and Biological Evaluation of Peptidomimetic Tetrahydropyrrole Spirodihydroindolones as SARS-CoV-2 3CL Protease Inhibitors 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 5, 页码: 790-796
作者:  
Hu, Liuyan;  Zhao, Zhi;  Zhang, Shujing;  Yang, Lei;  Cui, Wenjie
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/06/23
Development of RelB-targeting small-molecule inhibitors of non-canonical NF-kB signaling with antitumor efficacy 期刊论文  OAI收割
MOLECULAR THERAPY, 2025, 卷号: 33, 期号: 4, 页码: 1519-1534
作者:  
Li, Cuifeng;  Wei, Shuqi;  Sun, Donglin;  Yang, Zhuo;  Wang, Qi
  |  收藏  |  浏览/下载:0/0  |  提交时间:2025/05/27
Discovery of peptidomimetic spiropyrrolidine derivatives as novel 3CLpro inhibitors against SARS-CoV-2 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 281, 页码: 22
作者:  
Guma, Samuel Desta;  Zhou, Zhaoyin;  Song, Kang;  Yang, Feipu;  Suo, Jin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/12/11
Identification of USP2 as a novel target to induce degradation of KRAS in myeloma cells 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 12, 页码: 5235-5248
作者:  
Wang, Yingying;  Zhang, Youping;  Luo, Hao;  Wei, Wei;  Liu, Wanting
  |  收藏  |  浏览/下载:18/0  |  提交时间:2025/04/01
Synthesis of Natural Product-like Indeno[2,1-b]indole/Shikimic Acid Hybrid Analogues with Anti-osteoclastogenic Activity via Photo-Nazarov Reaction 期刊论文  OAI收割
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2024, 页码: 8
作者:  
Shao, Zhengguang;  Wang, Tianqi;  Zhang, Xiaofei;  Jiang, Min;  Zhu, Weiliang
  |  收藏  |  浏览/下载:4/0  |  提交时间:2024/12/11
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads 期刊论文  OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:  
Dong, Sanfeng;  Huang, Hui;  Li, Jintian;  Li, Xiaomei;  Bunu, Samuel Jacob
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/10/21
Synthesis and biological evaluation of multimodal monoaminergic arylpiperazine derivatives with potential antidepressant profile 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 275, 页码: 16
作者:  
Zheng, Jiefang;  Zhou, Liping;  Gong, Xudong;  Yang, Feipu;  Cheng, Jiaxin
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/08/22
Design, synthesis and structure-activity relationship of 1,8-naphthalimide derivatives as highly potent hCYP1B1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107, 页码: 8
作者:  
Wei, Yueyue;  Xiong, Yuan;  Liao, Qingyi;  Yang, Ya;  Tian, Tian
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/07/12
New Secondary Metabolites from Marine-Derived Fungus Talaromyces minnesotensis BTBU20220184 期刊论文  OAI收割
MARINE DRUGS, 2024, 卷号: 22, 期号: 6, 页码: 10
作者:  
Wang, Weiliang;  Wang, Jingjing;  Song, Fuhang;  Jia, Renming;  Wang, Long
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/09/02