机构

• 上海药物研究所 [77]

采集方式

• OAI收割 [77]

内容类型

• 期刊论文 [77]

发表日期

• 2024 [4]
• 2023 [2]
• 2022 [3]
• 2021 [4]
• 2019 [5]
• 2018 [4]
• 更多

学科主题

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浏览/检索结果: 共77条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Discovery of Thiochroman Derivatives as Potent, Oral Selective Estrogen Receptor Degraders and Antagonists for the Treatment of Endocrine-Resistant Breast Cancer 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 23, 页码: 21545-21567 作者:  Zhang, Dan;  Lu, Zhengyu;  He, Yongqi;  Leng, Xin-Yu;  Meng, Xin   |  收藏  |  浏览/下载：12/0  |  提交时间：2025/01/06 Discovery of YFJ-36: Design, Synthesis, and Antibacterial Activities of Catechol-Conjugated β-Lactams against Gram-Negative Bacteria 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21 作者:  Liu, Fangjun;  Kou, Qunhuan;  Li, Hongyuan;  Cao, Yangzhi;  Chen, Meng   |  收藏  |  浏览/下载：13/0  |  提交时间：2024/05/22 Design, Synthesis, and Biological Evaluation of Novel Arylomycins against Multidrug-Resistant Gram-Negative Bacteria 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 25 作者:  Zhang, Yinyong;  Zhang, Dan;  Zhao, Wenhao;  Li, Hongyuan;  Lu, Zhengyu   |  收藏  |  浏览/下载：20/0  |  提交时间：2024/05/22 Design, Synthesis, and Anti-tuberculosis Activity of Streptomycin Derivatives 期刊论文  OAI收割 LETTERS IN DRUG DESIGN & DISCOVERY, 2024, 卷号: 21, 期号: 4, 页码: 738-748 作者:  Zhang, Yinyong;  Zhao, Wenhao;  Yang, Yushe;  Zhou, Xianli;  Guo, Bin   |  收藏  |  浏览/下载：20/0  |  提交时间：2024/03/06 Multidrug-resistant  hydrazine  hydrazide  sulfonyl hydrazide  siderophore  synthesis  anti-tuberculosis activity   Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 14, 页码: 9972-9991 作者:  Wang, Ao;  Luo, Xianggang;  Meng, Xin;  Lu, Zhengyu;  Chen, Kaixian   |  收藏  |  浏览/下载：15/0  |  提交时间：2023/10/17 Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP 期刊论文  OAI收割 ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 12 作者:  Zhang, Yinyong;  Yang, Yushe;  Meng, Xin;  Zhou, Xianli;  Guo, Bin   |  收藏  |  浏览/下载：23/0  |  提交时间：2023/04/10 oxazolidinone  asymmetric reduction  fused ring  process development  crystal transformation   Design, Synthesis, and Biological Evaluation of Androgen Receptor Degrading and Antagonizing Bifunctional Steroidal Analogs for the Treatment of Advanced Prostate Cancer 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 22 作者:  Wang, Ao;  Luo, Xianggang;  Wang, Yawan;  Meng, Xin;  Lu, Zhengyu   |  收藏  |  浏览/下载：39/0  |  提交时间：2022/11/11 Design, Synthesis, and Structure-Activity Relationship Studies of Bisamide Derivatives of Amphotericin B with Potent Efficacy and Low Toxicity 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 17 作者:  Ma, Huijun;  Qian, Anran;  Zheng, Yazhou;  Meng, Xin;  Wang, Ting   |  收藏  |  浏览/下载：25/0  |  提交时间：2023/04/10 Discovery of Thieno[2,3-e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability br 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 7, 页码: 5724-5750 作者:  Lu, Zhengyu;  Cao, Yangzhi;  Zhang, Dan;  Meng, Xin;  Guo, Bin   |  收藏  |  浏览/下载：23/0  |  提交时间：2022/08/16 Design, Synthesis, and Biological Evaluation of Novel Pyrimido[4,5-b]indole Derivatives Against Gram-Negative Multidrug-Resistant Pathogens 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8644-8665 作者:  Kong, Qidi;  Pan, Wei;  Xu, Heng;  Xue, Yaru;  Guo, Bin   |  收藏  |  浏览/下载：46/0  |  提交时间：2021/08/17