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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
地理科学与资源研究所 [2]
大连化学物理研究所 [2]
上海光学精密机械研究... [1]
烟台海岸带研究所 [1]
采集方式
OAI收割 [13]
内容类型
期刊论文 [13]
发表日期
2024 [2]
2023 [2]
2022 [1]
2021 [3]
2016 [1]
2015 [2]
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学科主题
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浏览/检索结果:
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Synthesis and Biological Activity of Tetracyclic Dispiro Core Derivatives of Natural Products Dispirocochlearoids A-C
期刊论文
OAI收割
ORGANIC LETTERS, 2024, 卷号: 26, 期号: 45, 页码: 9654-9658
作者:
Pei, Junping
;
Wang, Ying
;
Shi, Shengjie
;
Chen, Linhai
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/12/11
Discovery of betulinic acid derivatives as gut-restricted TGR5 agonists: Balancing the potency and physicochemical properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 144, 页码: 18
作者:
Zhuo, Ning
;
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Yin, Jianpeng
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2024/03/25
Type 2 Diabetes
TGR5 agonist
Betulinic acid
Gut-restricted
Gallbladder-filling effects
Kinetophores
Development of the novel ACLY inhibitor 326E as a promising treatment for hypercholesterolemia
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 2, 页码: 739-753
作者:
Xie, Zhifu
;
Zhang, Mei
;
Song, Qian
;
Cheng, Long
;
Zhang, Xinwen
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2024/03/27
Hypercholesterolemia
Atherosclerosis
Liver
ATP-Citrate lyase (ACLY)
Lipogenesis
Cholesterol efflux
ACLY inhibitor
Temperature-related mortality in China from specific injury
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1
作者:
Hu, Jianxiong
;
He, Guanhao
;
Meng, Ruilin
;
Gong, Weiwei
;
Ren, Zhoupeng
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2024/01/04
Discovery of Betulinic Acid Derivatives as Potent Intestinal Farnesoid X Receptor Antagonists to Ameliorate Nonalcoholic Steatohepatitis
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 21
作者:
Zhang, Chenlu
;
Liu, Yameng
;
Wang, Ying
;
Ge, Xie
;
Jiao, Tingying
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/11/11
Optimization and Development of a Scalable Palladium-Catalyzed C-H Activation Process for the Geometry-Selective Preparation of Kilograms of YLF466D, a Potent AMP-Activated Protein Kinase Activator
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 10, 页码: 2260-2269
作者:
Yin, Jianpeng
;
Zhan, Desheng
;
Ma, Hui
;
Liu, Huanan
;
Yu, Lifang
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/12/16
YLF466D
AMPK activator
glucose metabolism
lipid metabolism
MIRI
domino reaction
C-H activation
Identification of Betulinic Acid Derivatives as Potent TGR5 Agonists with Antidiabetic Effects via Humanized TGR5(H88Y) Mutant Mice
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12181-12199
作者:
Yun, Ying
;
Zhang, Chenlu
;
Guo, Shimeng
;
Liang, Xiaoying
;
Lan, Yuan
  |  
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2021/11/04
The assessment of current mortality burden and future mortality risk attributable to compound hot extremes in China
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2021, 卷号: 777, 页码: 8
作者:
He, Guanhao
;
Xu, Yanjun
;
Hou, Zhulin
;
Ren, Zhoupeng
;
Zhou, Maigeng
  |  
收藏
  |  
浏览/下载:128/0
  |  
提交时间:2021/08/19
Compound hot extremes
Mortality risk
Global warming
China
Design and Synthesis of Diacylglycerol Acyltransferase 1 Inhibitors Based on Aphadilactone C
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 36, 期号: 6, 页码: 1359-1367
作者:
Li Dan
;
Yin Jianpeng
;
Li Jingya
;
Nan Fajun
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
aphadilactone C
DGAT1
selective inhibitor
PF-04620110
AZD-7687
ψ-Bufarenogin, a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling
期刊论文
OAI收割
Oncotarget, 2015, 卷号: 6, 期号: 13, 页码: 11627
作者:
Jin Ding
;
Wen Wen
;
Daimin Xiang
;
Peipei Yin
;
Liu YF(刘艳芳)
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2016/11/24