中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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期刊论文 [440]
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Discovery of Potent STING Inhibitors Bearing a Difluorobenzodioxol Structural Motif as Potent Anti-Inflammatory Agents
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 68, 期号: 8, 页码: 8907-8932
作者:
Shen, Ancheng
;
Wang, Xiyuan
;
Chen, Qingxuan
;
Zhang, Yan
;
Wang, Fang
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/05/27
Unity of terrestrial and extraterrestrial soils in granular configuration
期刊论文
OAI收割
EARTH AND PLANETARY SCIENCE LETTERS, 2025, 卷号: 654, 页码: 11
作者:
Zhang, Jun
;
Li, Yong
;
Cui, Yifei
;
Wu, Zi
;
Xue, Yuan
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2025/03/24
Soil genesis
Lunar regolith
Numerical simulant
Random simulation
Granular field
Discovery of a potential hematologic malignancies therapy: Selective and potent HDAC7 PROTAC degrader targeting non-enzymatic function
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 3, 页码: 1659-1679
作者:
Jin, Yuheng
;
Qi, Xuxin
;
Yu, Xiaoli
;
Cheng, Xirui
;
Chen, Boya
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/06/23
HDAC7
PROTAC
Selectivity
Hematologic malignancies
Non-enzymatic function
Design, synthesis and pharmacological evaluation of 1,2,3,4-tetrahydrobenzofuro[2,3-c] pyridine derivatives as p21-activated kinase 4 inhibitors for treatment of pancreatic cancer
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 438-466
作者:
Li, Yang
;
Fang, Yan
;
Chen, Xiaoyu
;
Tong, Linjiang
;
Feng, Fang
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2025/04/01
P21-activated kinase 4
Tetrahydrobenzofuro[2
3-c]pyridine
Structure-activity relationship
Allosteric inhibitor
Pharmacokinetics properties
Kinase selectivity
Pancreatic cancer
Immune infiltration
Attentional network deficits in patients with migraine: behavioral and electrophysiological evidence
期刊论文
OAI收割
JOURNAL OF HEADACHE AND PAIN, 2024, 卷号: 25, 期号: 1, 页码: 16
作者:
Chen, Yuxin
;
Xie, Siyuan
;
Zhang, Libo
;
Li, Desheng
;
Su, Hui
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/12/09
Migraine
Attention
Electroencephalography (EEG)
Vigilance
Hypersensitivity
Machine learning
GeneCompass: deciphering universal gene regulatory mechanisms with a knowledge-informed cross-species foundation model
期刊论文
OAI收割
CELL RESEARCH, 2024, 页码: 16
作者:
Yang, Xiaodong
;
Liu, Guole
;
Feng, Guihai
;
Bu, Dechao
;
Wang, Pengfei
  |  
收藏
  |  
浏览/下载:107/0
  |  
提交时间:2024/12/06
Molecular Dynamics Insights into Mechanical Stability, Elastic Properties, and Fracture Behavior of PHOTH-Graphene
期刊论文
OAI收割
MATERIALS, 2024, 卷号: 17, 期号: 19, 页码: 20
作者:
Peng, Qing
;
Chen, Gen
;
Huang, Zeyu
;
Chen, Xue
;
Li, Ao
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/11/14
PHOTH-graphene
mechanical property
MD
defects
hydrogen functionalization
Mid-Pleistocene climate transition triggered by Antarctic Ice Sheet growth
期刊论文
OAI收割
SCIENCE, 2024, 卷号: 385, 期号: 6708, 页码: 560-565
作者:
An, Zhisheng
;
Zhou, Weijian
;
Zhang, Zeke
;
Zhang, Xu
;
Liu, Zhonghui
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2025/03/28
Characterization and noncovalent inhibition of the K63-deubiquitinase activity of SARS-cov-2 PLpro
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2024, 卷号: 228, 页码: 12
作者:
Liu, Xin
;
Zheng, Miao
;
Zhang, Hongqing
;
Feng, Bo
;
Li, Jiaqi
  |  
收藏
  |  
浏览/下载:82/0
  |  
提交时间:2024/10/21
Discovery of a Highly Potent and Selective BRD9 PROTAC Degrader Based on E3 Binder Investigation for the Treatment of Hematological Tumors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 28
作者:
Duan, Haiting
;
Zhang, Jingyu
;
Gui, Renzhao
;
Lu, Yang
;
Pang, Ao
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/08/20