中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
首页
机构
成果
学者
登录
注册
登陆
×
验证码:
换一张
忘记密码?
记住我
×
校外用户登录
CAS IR Grid
机构
化学研究所 [3]
金属研究所 [2]
上海药物研究所 [1]
采集方式
OAI收割 [6]
内容类型
期刊论文 [6]
发表日期
2021 [1]
2009 [2]
2008 [1]
2006 [1]
2005 [1]
学科主题
筛选
浏览/检索结果:
共6条,第1-6条
帮助
条数/页:
5
10
15
20
25
30
35
40
45
50
55
60
65
70
75
80
85
90
95
100
排序方式:
请选择
题名升序
题名降序
发表日期升序
发表日期降序
提交时间升序
提交时间降序
作者升序
作者降序
Discovery and structure - activity relationship exploration of pyrazolo [1,5-a]pyrimidine derivatives as potent FLT3-ITD inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 48, 页码: 13
作者:
Chen, Yun
;
Bai, Gang
;
Li, Yan
;
Ning, Yi
;
Cao, Sufen
  |  
收藏
  |  
浏览/下载:73/0
  |  
提交时间:2021/12/01
FLT3
FLT3-ITD
Acute myeloid leukemia
Structure-activity relationships
Pyrazolo[1, 5-a]pyrimidine
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:
Zhi Hui
;
Chen Lanmei
;
Zhang Linlin
;
Liu Sijie
;
Wan David Chi Cheong
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/02/02
Acetylcholinesterase inhibitor
Docking screening
Heterocycle
Biological activity
5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors
期刊论文
OAI收割
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:
Zhi Hui
;
Chen Lanmei
;
Zhang Linlin
;
Liu Sijie
;
Wan David Chi Cheong
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/02/02
Acetylcholinesterase inhibitor
Docking screening
Heterocycle
Biological activity
5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative
Efficient construction of pyrazolo[1,5-a]pyrimidine scaffold and its exploration as a new heterocyclic fluorescent platform
期刊论文
OAI收割
JOURNAL OF FLUORESCENCE, 2008, 卷号: 18, 期号: 2, 页码: 357-363
作者:
Wu, Yan-Chao
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/04/09
Fluorophore
Heterocycle
Fluorescence
Pyrazolo[1
5-a]Pyrimidine
Synthesis of trifluoromethyl-promoted functional pyrazolo [1,5-a]pyrimidine and pyrazolo [5,1-d] [1,2,3,5]tetrazine-4(3H)-ones
期刊论文
OAI收割
JOURNAL OF FLUORINE CHEMISTRY, 2006, 卷号: 127, 期号: 3, 页码: 409-416
作者:
Wu, YC
;
Chen, YJ
;
Li, HJ
;
Zou, XM
;
Hu, FZ
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/04/09
Fluorine
Pyrazole
Inhibitor
Pyrazolo[1
Pyrazolo[5
5-a]Pyrimidine
1-d][1
2
3
5]Tetrazine-4(3h)-one
Synthesis of novel dipyrazolopyrimidine fused heterotricyclic compounds
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2005, 卷号: 23, 期号: 2, 页码: 182-184
作者:
Liu, Y
;
Zhang, XH
;
Jin, GY
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/04/09
1h-pyrazole-4-carboxamide
Synthesis
1h-dipyrazolo[1
1h-dipyrazolo[1
5-a : 3 '
5-a : 4 '
4 '-d]Pydmidine-4(9h)-one
3 '-e]Pyrimidine-4(5h)-one