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中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [3]
长春应用化学研究所 [3]
化学研究所 [1]
成都生物研究所 [1]
大连化学物理研究所 [1]
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OAI收割 [11]
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期刊论文 [11]
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2013 [2]
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Chemistry [1]
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Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrido[4,3-c]azepin-5-one-based novel chemotype CCR2 antagonists via scaffold hopping strategy
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12, 页码: 3559-3572
作者:
Qin, Li-Huai
;
Wang, Zhi-Long
;
Xie, Xin
;
Long, Ya-Qiu
|
收藏
|
浏览/下载:42/0
|
提交时间:2019/01/08
6,7,8,9-Tetrahydro-5H-pyrido[43-c]azepin-5-one
3,4-Dihydro-2,6-naphthyridin-1(2H)-one
CCR2 antagonist
Scaffold hopping
Structure-activity relationship
Selectivity of CCR2 over CCR5
Synthesis and Activity Evaluation of Novel 3,4-Dihydro-benzo[b]-oxazepin-5(2H)-one Derivatives as Protein Kinases Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 6, 页码: 1463-1472
作者:
Hou Guige
;
Jiang Chengshi
;
Liu Hongchun
;
Tong Linjiang
;
Peng Xia
|
收藏
|
浏览/下载:38/0
|
提交时间:2019/01/08
3,4-dihydro-benzo[b]oxazepin-5(2H)-one derivatives
synthesis
protein-tyrosine kinases inhibitors
ErbB1
ErbB2
POCl3-Mediated Reaction of 1-Acyl-1-carbamoyl Oximes: A New Entry to Cyanoformamides
期刊论文
OAI收割
organic letters, 2015, 卷号: 17, 期号: 4, 页码: 809-811
作者:
Yang,Jiming
;
Xiang,Dexuan
;
Zhang,Rui
;
Zhang,Ning
;
Liang,Yongjiu
收藏
|
浏览/下载:22/0
|
提交时间:2016/05/04
HIGHLY SUBSTITUTED PYRIDIN-2(1H)-ONES
SPONGE PSEUDOCERATINA-PURPUREA
EFFICIENT SYNTHESIS
INTRAMOLECULAR CYANOAMIDATION
DIVERGENT SYNTHESIS
CYCLOPROPANES
POCL3
2-ARYLAMINO-3-ACETYL-5
CERATINAMINE
PALLADIUM
6-DIHYDRO-4H-PYRANS
Antioxidants in volatile Mail lard reaction products: Identification and interaction
期刊论文
OAI收割
lwt-food science and technology, 2013, 卷号: 53, 期号: 1, 页码: 22-28
作者:
Yu, Xiangying
;
Zhao, Mingyue
;
Liu, Fei
;
Zeng, Shitong
;
Hu, Jun
收藏
|
浏览/下载:35/0
|
提交时间:2015/11/09
Antioxidant
Volatile Maillard reaction products (MRPs)
2
2
2-Hydroxy-3-methyl-2-cyclopenten-1-one (CP)
5-Dimethyl-4-hydroxy-3(2H)furanone (DMHF)
3-Dihydro-3
5-dihydroxy-6-methyl-4H-pyran-4-one (DDMP)
Design, Synthesis, and Structure-Activity Relationships of 3,4,5-Trisubstituted 4,5-Dihydro-1,2,4-oxadiazoles as TGR5 Agonists
期刊论文
OAI收割
CHEMMEDCHEM, 2013, 卷号: 8, 期号: 7, 页码: 1210-1223
作者:
Zhu, Junjie
;
Ye, Yangliang
;
Ning, Mengmeng
;
Mandi, Attila
;
Feng, Ying
|
收藏
|
浏览/下载:25/0
|
提交时间:2019/01/08
4
5-dihydro-1
2
4-oxadiazoles
cycloaddition
metabolic disorders
structure-activity relationships
TGR5
Regioselective Synthesis of 3-Arylamino- and 5-Arylaminoisoxazoles from Enaminones
期刊论文
OAI收割
organic letters, 2012, 卷号: 14, 期号: 2, 页码: 644-647
Xiang DX
;
Xin XQ
;
Liu X
;
Zhang R
;
Yang JM
;
Dong DW
收藏
|
浏览/下载:32/0
|
提交时间:2013/06/08
ONE-POT SYNTHESIS
2-ARYLAMINO-3-ACETYL-5
S
REGIOSPECIFIC SYNTHESIS
6-DIHYDRO-4H-PYRANS
N-ACETALS
HALOGENATED PYRIDIN-2(1H)-ONES
EFFICIENT SYNTHESIS
ISOXAZOLES
HYDROXYLAMINE
HETEROCYCLES
CYCLOPROPANES
Discovery of 5,6-Dihydro-indolo[1,2-a]quinoxaline Derivatives as New HIV-1 Inhibitors In Vitro
期刊论文
OAI收割
LETTERS IN DRUG DESIGN & DISCOVERY, 2012, 卷号: 9, 期号: 1, 页码: 44-47
作者:
Fan LL
;
Huang N
;
Yang RG
;
He SZ
;
Yang LM
收藏
|
浏览/下载:28/0
|
提交时间:2012/04/05
5
6-Dihydro-indolo[1
2-a]quinoxaline
Acquired immunodeficiency syndrome
Human immunodeficiency virus-1
Inhibitor
Ring-Opening/Recyclization Reactions of (Dimethylamino)propenoyl-Substituted Cyclopropanes: Facile Synthesis of Halogenated Pyridin-2(1H)-ones
期刊论文
OAI收割
synthesis-stuttgart, 2009, 期号: 15, 页码: 2497-2500
Zhang R
;
Zhou Y
;
Liang YJ
;
Jiang ZJ
;
Dong DW
收藏
|
浏览/下载:164/64
|
提交时间:2010/06/18
HIGHLY SUBSTITUTED PYRIDIN-2(1H)-ONES
EFFICIENT SYNTHESIS
DIVERGENT SYNTHESIS
PYRIDINE RINGS
CYCLOADDITION
HETEROCYCLES
ROUTE
ACID
2-ARYLAMINO-3-ACETYL-5
2(1H)-PYRIDONES
6-DIHYDRO-4H-PYRANS
Synthesis of 5,6-dihydro-OSW-1 and its antitumor activities
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2004, 卷号: 22, 期号: 9, 页码: 994-998
作者:
Deng, LH
;
Wu, H
;
Yu, B
;
Jiang, MR
;
Wu, JR
收藏
|
浏览/下载:19/0
|
提交时间:2015/07/22
5
analog
synthesis
anti-tumor
6-dihydro-OSW-1
Spectral study of a new dihydroisocoumarin
期刊论文
OAI收割
MAGNETIC RESONANCE IN CHEMISTRY, 2003, 卷号: 41, 期号: 9, 页码: 718-720
作者:
Wang, HM
;
Shi, W
;
Xu, YK
;
Liu, Y
;
Lu, MJ
|
收藏
|
浏览/下载:17/0
|
提交时间:2019/04/09
Nmr
H-1 Nmr
C-13 Nmr
2d Nmr
X-ray Crystallography
3
4-dihydro-6
8-dihydroxy-3-(2 '-acetyl-3 '-hydroxy-5 '-methoxy)Methyl-1h-[2]Benzopyran-1-one
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