中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [6]
化学研究所 [3]
大连化学物理研究所 [2]
海洋研究所 [2]
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OAI收割 [17]
iSwitch采集 [2]
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期刊论文 [18]
CNKI期刊论文 [1]
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2023 [1]
2019 [2]
2018 [2]
2017 [4]
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Biochemist... [1]
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Structural insights into the interaction of three Y- shaped ligands with PI3Kα
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2023, 卷号: 120, 期号: 34, 页码: 9
作者:
Zhou, Qingtong
;
Liu, Xiao
;
Neri, Dario
;
Li, Wenxin
;
Favalli, Nicholas
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/12/08
phosphoinositide 3-kinase
drug target
ligand
binding pocket
chemical scaffold
Structural Insights into Phosphite Dehydrogenase Variants Favoring a Non-natural Redox Cofactor
期刊论文
OAI收割
ACS CATALYSIS, 2019, 卷号: 9, 期号: 3, 页码: 1883-1887
作者:
Xue, Song
;
Liu, Yuxue
;
Feng, Yanbin
;
Wang, Lei
;
Guo, Xiaojia
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2019/06/20
phosphite dehydrogenase
non-natural redox cofactor
NAD-binding pocket
nicotinamide cytosine dinucleotide
cofactor preference
Structural insights into phosphite dehydrogenase variants favoring a non-natural redox cofactor
期刊论文
iSwitch采集
Acs catalysis, 2019, 卷号: 9, 期号: 3, 页码: 1883-1887
作者:
Liu, Yuxue
;
Feng, Yanbin
;
Wang, Lei
;
Guo, Xiaojia
;
Liu, Wujun
收藏
  |  
浏览/下载:101/0
  |  
提交时间:2019/05/08
Phosphite dehydrogenase
Non-natural redox cofactor
Nad-binding pocket
Nicotinamide cytosine dinucleotide
Cofactor preference
Design, synthesis and biological evaluation of benzo[cd]indo1-2(1H)-ones derivatives as BRD4 inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 264-273
作者:
Feng, Yuxin
;
Xiao, Senhao
;
Chen, Yantao
;
Jiang, Hao
;
Liu, Na
  |  
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2019/01/08
Benzo[cd]indol-2(1H)-one
Sulfonamide
BRD4 inhibitor
Bromodomain and extra-terminal domain
Acetyl-lysine binding pocket
A novel series of 4-methyl substituted pyrazole derivatives as potent glucagon receptor antagonists: Design, synthesis and evaluation of biological activities
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1896-1908
作者:
Shu, Shuangjie
;
Dai, Antao
;
Wang, Jiang
;
Wang, Bin
;
Feng, Yang
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2019/01/08
Pyrazole derivatives
Glucagon receptor antagonist
Docking study
Binding pocket
Structure-based function prediction of the expanding mollusk tyrosinase family
CNKI期刊论文
OAI收割
2017
作者:
Huang RL(黄荣莲)
;
Li L(李莉)
;
Zhang GF(张国范)
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/12/18
tyrosinase
mollusk
ligand binding pocket
substrate diversity
evolution
Structure-based function prediction of the expanding mollusk tyrosinase family
期刊论文
OAI收割
CHINESE JOURNAL OF OCEANOLOGY AND LIMNOLOGY, 2017, 卷号: 35, 期号: 6, 页码: 1454-1464
作者:
Huang Ronglian
;
Li Li
;
Zhang Guofan
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2018/01/16
Tyrosinase
Mollusk
Ligand Binding Pocket
Substrate Diversity
Evolution
Structure alignment-based classification of RNA-binding pockets reveals regional RNA recognition motifs on protein surfaces
期刊论文
OAI收割
BMC BIOINFORMATICS, 2017, 卷号: 18, 页码: 13
作者:
Liu, Zhi-Ping
;
Liu, Shutang
;
Chen, Ruitang
;
Huang, Xiaopeng
;
Wu, Ling-Yun
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2018/07/30
RNA-binding pocket
Local structure classification
Structural alignment
Network clustering
Structure motif
Anchor Effect of Interactions Between Kinesin's Nucleotide-Binding Pocket and Microtubule
期刊论文
OAI收割
CELLULAR AND MOLECULAR BIOENGINEERING, 2017, 卷号: 10, 期号: 2, 页码: 162-173
作者:
Geng, YZ
;
Jin, YM
;
Lu, LN
;
Ma, YL
;
Lu, G
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2017/12/21
Kinesin
Microtubule
Nucleotide-binding Pocket
Anchor Effect
Bavachinin, as a novel natural pan-PPAR agonist, exhibits unique synergistic effects with synthetic PPAR-gamma and PPAR-alpha agonists on carbohydrate and lipid metabolism in db/db and diet-induced obese mice
期刊论文
OAI收割
DIABETOLOGIA, 2016, 卷号: 59, 期号: 6, 页码: 1276-1286
作者:
Feng, Li
;
Luo, Huan
;
Xu, Zhijian
;
Yang, Zhuo
;
Du, Guoxin
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2016/08/22
Alternative binding site
Bavachinin
Canonical ligand-binding pocket
Carbohydrate metabolism
Lipid metabolism
Pan-PPAR agonist
Synergistic effects