中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [29]
上海营养与健康研究所 [6]
生态环境研究中心 [5]
心理研究所 [4]
上海生物化学与细胞生... [4]
水生生物研究所 [3]
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OAI收割 [69]
iSwitch采集 [3]
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期刊论文 [72]
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2024 [2]
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2020 [4]
2019 [8]
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浏览/检索结果:
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Discovery of a potent PROTAC degrader for RNA demethylase FTO as antileukemic therapy
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2024, 卷号: 14, 期号: 12, 页码: 5382-5392
作者:
Liu, Lu
;
Qiu, Yuanlai
;
Suo, Yuying
;
Tong, Siyao
;
Wang, Yiqing
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/04/01
N 6-Methyladenosine
FTO
PROTAC
RNA epigenetics
Antileukemia
Promoter methylation as a potential cause for the decrease in pyruvate metabolism during environmentally induced aestivation in Apostichopus japonicus
期刊论文
OAI收割
AQUACULTURE, 2024, 卷号: 579, 页码: 10
作者:
Jiang, Chunxi
;
Sun, Lina
;
Yang, Hongsheng
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/11/30
Environmentally induced aestivation
Epigenetics
Promoter methylation
Pyruvate metabolism
Identification of Histone Lysine Acetoacetylation as a Dynamic Post-Translational Modification Regulated by HBO1
期刊论文
OAI收割
ADVANCED SCIENCE, 2023, 页码: 11
作者:
Gao, Yan
;
Sheng, Xinlei
;
Tan, Doudou
;
Kim, SunJoo
;
Choi, Soyoung
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/10/17
acetoacetate
acetoacetylation
epigenetics
HBO1
histone marks
novel histone modification
Design, synthesis and biological evaluation of (R)-5-methylpyrrolidin-2-ones as p300 bromodomain inhibitors with Anti-Tumor activities in multiple tumor lines
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 124, 页码: 15
作者:
Liu, Ruiqi
;
Yang, Hong
;
Chen, Zonglong
;
Zhou, Kaixin
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2022/08/16
Epigenetics
p300
CBP
Bromodomain inhibitors
CCS1477
Complementary genomic and epigenomic adaptation to environmental heterogeneity
期刊论文
OAI收割
MOLECULAR ECOLOGY, 2022, 卷号: 31, 期号: 13, 页码: 3598-3612
作者:
Gao, Yangchun
;
Chen, Yiyong
;
Li, Shiguo
;
Huang, Xuena
;
Hu, Juntao
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/11/09
POPULATION-GENETICS
DNA METHYLATION
BOTRYLLID ASCIDIANS
EPIGENETICS
ASSOCIATION
PATTERNS
MARINE
MODEL
TOOL
BIOGEOGRAPHY
Design, synthesis and biological evaluation of a novel spiro oxazolidinedione as potent p300/CBP HAT inhibitor for the treatment of ovarian cancer
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 52, 页码: 12
作者:
Ding, Hong
  |  
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2022/06/15
Epigenetics
Histone acetyltransferase
P300/CBP
Ovarian cancer
Histone deacetylase inhibitor givinostat attenuates nonalcoholic steatohepatitis and liver fibrosis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Huang, He-ming
;
Fan, Shi-jie
;
Zhou, Xiao-ru
;
Liu, Yan-jun
;
Li, Xiao
  |  
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2021/11/04
nonalcoholic steatohepatitis
inflammation
histone deacetylase inhibitor
givinostat
epigenetics
Histone deacetylase inhibitor givinostat alleviates liver fibrosis by regulating hepatic stellate cell activation
期刊论文
OAI收割
MOLECULAR MEDICINE REPORTS, 2021, 卷号: 23, 期号: 5, 页码: 12
作者:
Huang, He-Ming
;
Zhou, Xiao-Ru
;
Liu, Yan-Jun
;
Fan, Shi-Jie
;
Liao, Li-Ping
  |  
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2021/05/24
liver fibrosis
hepatic stellate cell
histone deacetylase inhibitor
epigenetics
givinostat
P300/CBP inhibition sensitizes mantle cell lymphoma to PI3K delta inhibitor idelalisib
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhou, Xiao-ru
;
Li, Xiao
;
Liao, Li-ping
;
Han, Jie
;
Huang, Jing
  |  
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2021/06/11
mantle cell lymphoma
idelalisib
drug resistance
P300
CBP
synergistic drug action
PI3Kδ
epigenetics
P300/CBP inhibition sensitizes mantle cell lymphoma to PI3K delta inhibitor idelalisib
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhou, Xiao-ru
;
Li, Xiao
;
Liao, Li-ping
;
Han, Jie
;
Huang, Jing
  |  
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2021/06/11
mantle cell lymphoma
idelalisib
drug resistance
P300
CBP
synergistic drug action
PI3Kδ
epigenetics