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Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [7]
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Design, synthesis and biological evaluation of novel pyrrolo[1,2-b]pyridazin-2(1
H
)-ones as selective PARP1 inhibitors for cancer therapy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2026, 卷号: 307, 页码: 16
作者:
He, Qiaolin
;
He, Jing
;
Huan, Xiajuan
;
Song, Shanshan
;
Zhang, Xiaofei
  |  
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Structure-Based Discovery of a Series of Novel MAT2a Inhibitors
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 页码: 5
作者:
Zhou, Yushan
;
Wang, Li
;
Ren, Ruyue
;
Zhang, Junjie
;
Huan, Xiajuan
  |  
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  |  
Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:
Wang, Pingyuan
;
Zhu, Wen-Ting
;
Wang, Yajing
;
Song, Shan-Shan
;
Xi, Yong
  |  
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BCL-2 inhibitor synergizes with PI3K delta inhibitor and overcomes FLT3 inhibitor resistance in acute myeloid leukaemia
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2022, 卷号: 12, 期号: 8, 页码: 3829-3842
作者:
Yao, Ming-Yue
;
Wang, Ya-Fang
;
Zhao, Yu
;
Ling, Li-Jun
;
He, Ye
  |  
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  |  
CRISPR-cas9: a powerful tool towards precision medicine in cancer treatment
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 5, 页码: 583-587
作者:
Xing, Hui
;
Meng, Ling-hua
  |  
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Enhancement of DNA damage repair potential in germ cells of Caenorhabditis elegans by a volatile signal from their irradiated partners
期刊论文
OAI收割
DNA REPAIR, 2020, 卷号: 86, 期号: 1, 页码: 9
作者:
Tang, Huangqi
;
Chen, Liangwen
;
Dai, Zhangyu
;
Zhang, Wenjing
;
Wang, Ting
  |  
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Development of novel chromeno[4,3-c]pyrazol-4(2H)-one derivates containing piperazine as inhibitors of PI3K alpha
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2019, 卷号: 92
作者:
Yin, Yong
;
Zhou, Yang
;
Sha, Shao
;
Wu, Xun
;
Wang, She-Feng
  |  
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  |  
Development of novel chromeno[4,3-c]pyrazol-4(2H)-one derivates containing piperazine as inhibitors of PI3K alpha
会议论文
OAI收割
作者:
Yin, Yong
;
Zhou, Yang
;
Sha, Shao
;
Wu, Xun
  |  
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  |  
Lipid-Based Liquid Crystalline Nanoparticles Facilitate Cytosolic Delivery of siRNA via Structural Transformation
期刊论文
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NANO LETTERS, 2018, 卷号: 18, 期号: 4, 页码: 2411-2419
作者:
He, Shufang
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Novel PARP1/2 inhibitor mefuparib hydrochloride elicits potent in vitro and in vivo anticancer activity, characteristic of high tissue distribution
期刊论文
OAI收割
ONCOTARGET, 2017, 卷号: 8, 期号: 3, 页码: 4156-4168
作者:
He, Jin-Xue
;
Wang, Meng
;
Huan, Xia-Juan
;
Chen, Chuan-Huizi
;
Song, Shan-Shan
  |  
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