中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
长春应用化学研究所 [3]
化学研究所 [2]
上海药物研究所 [2]
福建物质结构研究所 [1]
采集方式
OAI收割 [8]
内容类型
期刊论文 [8]
发表日期
2024 [1]
2022 [1]
2015 [3]
2012 [1]
2011 [1]
2007 [1]
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学科主题
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Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 112, 页码: 5
作者:
Shen, Wen
;
Chen, Xinyao
;
Zhou, Liping
;
Cheng, Yan
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/10/21
COVID-19
SARS-CoV-2 3CL pro inhibitor
Drug design
Antiviral activities
Synthesis and Biochemical Evaluation of 8H-Indeno[1,2-d]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors
期刊论文
OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 10, 页码: 11
作者:
Wu, Jing
;
Feng, Bo
;
Gao, Li-Xin
;
Zhang, Chun
;
Li, Jia
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2022/08/16
COVID-19
M-pro inhibitors
drug design and synthesis
structure-activity relationships (SAR)
Inorganic nanocarriers for platinum drug delivery
期刊论文
OAI收割
materials today, 2015, 卷号: 18, 期号: 10, 页码: 554-564
作者:
Ma,Ping'an
;
Xiao,Haihua
;
Li,Chunxia
;
Dai,Yunlu
;
Cheng,Ziyong
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2016/04/29
NANOSCALE COORDINATION POLYMERS
GOLD NANOPARTICLES
ANTICANCER DRUGS
PRODRUG DELIVERY
PRO-DRUG
IN-VIVO
UPCONVERTING NANOPARTICLES
CELLULAR ACCUMULATION
SILICA NANOPARTICLES
ANTITUMOR-ACTIVITY
A polymer-(multifunctional single-drug) conjugate for combination therapy
期刊论文
OAI收割
journal of materials chemistry b, 2015, 卷号: 3, 期号: 24, 页码: 4913-4921
作者:
Zhou,Dongfang
;
He,Shasha
;
Cong,Yuwei
;
Xie,Zhigang
;
Chen,Xuesi
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2016/05/12
PLATINUM ANTICANCER COMPLEX
OVARIAN-CARCINOMA CELLS
POLYMER THERAPEUTICS
CANCER-CHEMOTHERAPY
DRUG-RESISTANCE
DNA-DAMAGE
ENHANCED PERMEABILITY
CO-DELIVERY
PRO-DRUG
IN-VIVO
A dextran-platinum(IV) conjugate as a reduction-responsive carrier for triggered drug release
期刊论文
OAI收割
journal of materials chemistry b, 2015, 卷号: 3, 期号: 41, 页码: 8203-8211
作者:
He,Shasha
;
Cong,Yuwei
;
Zhou,Dongfang
;
Li,Jizhen
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2016/05/12
COPOLYMER MICELLES
ANTICANCER DRUGS
CANCER-THERAPY
PRO-DRUG
DELIVERY
NANOPARTICLES
DOXORUBICIN
ENCAPSULATION
CISPLATIN
POLYMERS
A complex of cyclohexane-1,2-diaminoplatinum with an amphiphilic biodegradable polymer with pendant carboxyl groups
期刊论文
OAI收割
ACTA BIOMATERIALIA, 2012, 卷号: 8, 期号: 5, 页码: 1859-1868
作者:
Xiao, Haihua
;
Zhou, Dongfang
;
Liu, Shi
;
Zheng, Yonghui
;
Huang, Yubin
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/04/09
Cancers
Micelles
Oxaliplatin
Polymer-drug Conjugate
Pro-drug
Experimental study on biodegradable polymer-paclitaxel conjugate micelles for chemotherapy of C6 glioma
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2011, 卷号: 152, 页码: E41-E42
作者:
Wang, Zhanfeng
;
Hu, Xiuli
;
Yue, Jun
;
Jing, Xiabin
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/04/09
C6 Glioma
Wistar Rats
Paclitaxel
Pro-drug
Epr Effect
Bbb
Structural basis of specificity of a peptidyl urokinase inhibitor, upain-1
期刊论文
OAI收割
Journal of Structural Biology, 2007, 卷号: 160, 期号: 1, 页码: 1-10
G. X. Zhao
;
C. Yuan
;
T. Wind
;
Z. X. Huang
;
P. A.
;
reasen
;
M. D. Huang
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2013/04/01
urokinase-type plasminogen activator
peptidyl inhibitor
crystal
structure
pharmacophore
activator pro-upa
plasminogen-activator
crystal-structure
single-chain
selective inhibitors
drug design
complex
receptor
system
domain