机构

• 上海药物研究所 [7]
• 福建物质结构研究所 [2]
• 昆明植物研究所 [1]

采集方式

• OAI收割 [10]

内容类型

• 期刊论文 [10]

发表日期

• 2019 [1]
• 2018 [1]
• 2016 [3]
• 2012 [1]
• 2011 [2]
• 2010 [2]
• 更多

学科主题

• Chemistry,... [1]

筛选

浏览/检索结果: 共10条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85 作者:  Zhan, Wenhu;  Che, Jinxin;  Xu, Lei;  Wu, Yizhe;  Hu, Xiaobei   |  收藏  |  浏览/下载：24/0  |  提交时间：2020/07/01 Pyrazole-thiophene derivatives  Akt inhibitor  Antitumor   A novel series of 4-methyl substituted pyrazole derivatives as potent glucagon receptor antagonists: Design, synthesis and evaluation of biological activities 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 8, 页码: 1896-1908 作者:  Shu, Shuangjie;  Dai, Antao;  Wang, Jiang;  Wang, Bin;  Feng, Yang   |  收藏  |  浏览/下载：23/0  |  提交时间：2019/01/08 Pyrazole derivatives  Glucagon receptor antagonist  Docking study  Binding pocket   Structural optimization and biological evaluation of 1,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase 期刊论文  OAI收割 ACTA PHARMACEUTICA SINICA B, 2016, 卷号: 6, 期号: 1, 页码: 32-45 作者:  Zhou, Yu;  Liu, Jun;  Zheng, Mingyue;  Zheng, Shuli;  Jiang, Chunyi   |  收藏  |  浏览/下载：29/0  |  提交时间：2019/01/08 5-Lipoxygenase  5-LOX inhibitors  Pyrazole derivatives  Leukotrienes-related diseases  In vivo  Benzo-fuse heterocyle  Ischemic incults  Brain inflammation   structuraloptimizationandbiologicalevaluationofl5disubstitutedpyrazole3carboxaminesaspotentinhibitorsofhuman5lipoxygenase 期刊论文  OAI收割 actapharmaceuticasinicab, 2016, 卷号: 6, 期号: 1, 页码: 32 作者:  Zhou Yu;  Liu Jun;  Zheng Mingyue;  Zheng Shuli;  Jiang Chunyi   |  收藏  |  浏览/下载：16/0  |  提交时间：2020/07/01 5-Lipoxygenase  5-LOX inhibitors  Pyrazole derivatives  Leukotrienes-related diseases  In vivo  Benzo-fused heterocycle  Ischemic incults  Brain inflammation   Structural optimization and biological evaluation of l,5-disubstituted pyrazole-3-carboxamines as potent inhibitors of human 5-lipoxygenase 期刊论文  OAI收割 Acta Pharmaceutica Sinica B, 2016, 卷号: 6, 期号: 1, 页码: 32 作者:  Zhou Yu;  Liu Jun;  Zheng Mingyue;  Zheng Shuli;  Jiang Chunyi   |  收藏  |  浏览/下载：9/0  |  提交时间：2020/12/24 5-Lipoxygenase  5-LOX inhibitors  Pyrazole derivatives  Leukotrienes-related diseases  In vivo  Benzo-fused heterocycle  Ischemic incults  Brain inflammation   Synthesis and Antioxidant Activities of Novel 4,4 '-Arylmethylene-bis(1H-pyrazole-5-ol)s from Lignin 期刊论文  OAI收割 CHINESE JOURNAL OF CHEMISTRY, 2012, 卷号: 30, 期号: 3, 页码: 670 作者:  Yang Xiaohui;  Zhang Pinghu;  Zhou Yonghong;  Wang Junsong;  Liu Hongjun   |  收藏  |  浏览/下载：17/0  |  提交时间：2020/12/24 PYRAZOLE DERIVATIVES  SEPARATION  VANILLIN  OIL  pyrazole  microwave chemistry  aromatic aldehyde  4  4'-arylmethylene-bis(1H-pyrazole-5-ol)  lignin  antioxidants   Towards rational design of zinc(II) and cadmium(II) sulfonate-arsonates with low dimensional aggregations 期刊论文  OAI收割 Crystengcomm, 2011, 卷号: 13, 期号: 5, 页码: 1480-1489 F. Y. Yi; H. B. Xu; T. H. Zhou; J. G. Mao 收藏  |  浏览/下载：45/0  |  提交时间：2012/06/06 state coordination chemistry  phosphonate cage complexes  structural-characterization  polyoxometalate clusters  pyrazole ligands  solid-state  hydrothermal synthesis  organic derivatives  magnetic-properties  metal phosphonates   Molecular docking-based 3D-QSAR studies of pyrrolo[3,4-c]pyrazole derivatives as Aurora-A inhibitors 期刊论文  OAI收割 MOLECULAR SIMULATION, 2011, 卷号: 37, 期号: 1, 页码: 31-42 He, G.; Qiu, M. H.; Li, R.; Song, X. R.; Zheng, X.; Shi, J. Y.; Xu, G. B.; Han, J.; Yu, L. T.; Yang, S. Y.; Chen, L. J.; Wei, Y. Q. 收藏  |  浏览/下载：23/0  |  提交时间：2012/10/12 pyrrolo[3  4-c]pyrazole derivatives  3D-QSAR  molecular docking  CoMFA  CoMSIA  KINASE INHIBITORS  PROTEIN-KINASE  PHARMACOPHORE MODEL  SIMILARITY INDEXES  ANALYSIS COMSIA  POTENT  IDENTIFICATION  BINDING  PROFILE  COMFA   Discovery and structural optimization of pyrazole derivatives as novel inhibitors of Cdc25B 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 卷号: 20, 期号: 9, 页码: 2876-2879 作者:  Chen, Hai-Jun;  Liu, Yong   |  收藏  |  浏览/下载：25/0  |  提交时间：2019/01/08 Structural optimization  Cdc25B inhibitor  Pyrazole derivatives   A Series of New Manganese(II) Sulfonate-Arsonates with 2D Layer, 1D Chain, and 0D Clusters Structures 期刊论文  OAI收割 Inorganic Chemistry, 2010, 卷号: 49, 期号: 7, 页码: 3489-3500 F. Y. Yi, Q. P. Lin, T. H. Zhou and J. G. Mao 收藏  |  浏览/下载：58/0  |  提交时间：2012/11/02 phosphonate cage complexes  magnetic-properties  polyoxometalate  clusters  crystal-structures  hydrothermal synthesis  luminescent  properties  organic derivatives  metal phosphonates  pyrazole ligands  solid-state