中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [2]
过程工程研究所 [2]
昆明植物研究所 [1]
海洋研究所 [1]
上海营养与健康研究所 [1]
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OAI收割 [7]
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期刊论文 [7]
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2021 [1]
2019 [1]
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2009 [1]
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Biochemist... [2]
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Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Design, synthesis, and cytotoxic activities of novel hybrids of parthenolide and thiazolidinedione via click chemistry
期刊论文
OAI收割
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2019, 页码: 9
作者:
Qiu, Jie
;
Yuan, Chun-Mao
;
Wen, Min
;
Li, Ya-Nan
;
Chen, Juan
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2019/07/29
Parthenolide-thiazolidinedione hybrids
click chemistry
cytotoxic activities
Peroxisome Proliferator-Activated Receptor gamma and Its Role in Adipocyte Homeostasis and Thiazolidinedione-Mediated Insulin Sensitization
期刊论文
OAI收割
MOLECULAR AND CELLULAR BIOLOGY, 2018, 卷号: 38, 期号: 10, 页码: UNSP e00677
作者:
Wang, Qiong A.
;
Zhang, Fang
;
Ye, Risheng
;
An, Yu
;
Shao, Mengle
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/12/09
C/EBP alpha
insulin sensitization
PPAR gamma
thiazolidinedione
adipocyte
adipose tissue
inducible knockout
mouse model
obesity
3D QSAR studies on peroxisome proliferator-activated receptor gamma agonists using CoMFA and CoMSIA
期刊论文
OAI收割
JOURNAL OF MOLECULAR MODELING, 2004, 卷号: 10, 期号: 3, 页码: 165-177
作者:
Liao, CZ
;
Xie, AH
;
Zhou, JJ
;
Shi, LM
;
Li, ZB
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2013/11/05
3D QSAR
CoMFA
CoMSIA
PPAR
thiazolidinedione
insulin sensitizer
drug design
Eigenvalue analysis of peroxisome proliferator-activated receptor gamma agonists
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND COMPUTER SCIENCES, 2004, 卷号: 44, 期号: 1, 页码: 230-238
作者:
Liao, CZ
;
Xie, AH
;
Shi, LM
;
Zhou, JJ
;
Lu, XP
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2013/11/05
molecular similarity indexes
thiazolidinedione antihyperglycemic
agents
beta-phenylpropanoic acids
ppar-gamma
ligand-binding
biological-activity
crystal-structure
eva descriptor
field analysis
qsar