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Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [101]
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SLL-023ACP, a KOR/MOR dual agonist, produces potent antinociception with fewer side effects
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2026, 卷号: 806, 页码: 10
作者:
Shen, Yi-Quan
;
Liu, Pan-Wen
;
Zhang, Deng-Gao
;
Liu, Min
;
Luo, Jia-Wen
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Radiosynthesis and Biological Evaluation of a Small-Molecule Probe for Thyroid-Stimulating Hormone Receptor
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 16, 期号: 9, 页码: 1740-1746
作者:
Zhou, Yuanyuan
;
Tao, Ji
;
Jiang, Yuanpeng
;
Ji, Aiyan
;
Luo, Xiangning
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Structural and mechanistic insights into dual activation of cagrilintide in amylin and calcitonin receptors
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2025, 页码: 11
作者:
Gu, Yi-min
;
Yuan, Qing-ning
;
Li, Xin
;
He, Qian
;
Xu, H. Eric
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Relief of loperamide-induced constipation by peptidic and small molecule RXFP4 agonists in mice
期刊论文
OAI收割
BIOCHEMICAL PHARMACOLOGY, 2025, 卷号: 237, 页码: 12
作者:
Yan, Shiyu
;
Chen, Yan
;
Wang, Jiang
;
Wang, Qiuying
;
Zhou, Qingtong
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Structure-activity relationship analysis of meta-substituted N-cyclopropylmethyl-nornepenthones with mixed KOR/MOR activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 289, 页码: 15
作者:
Tang, Siyuan
;
Hu, Shuyang
;
Feng, Lijing
;
Kong, Linghui
;
Gui, Jiangwen
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Drug discovery targeting thyroid hormone receptor f3 (THRf3) for the treatment of liver diseases and other medical indications
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2025, 卷号: 15, 期号: 1, 页码: 35-51
作者:
Wang, Kean
;
Chen, Feiyang
;
Wang, Jiang
;
Liu, Hong
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Discovery of a non-nucleotide stimulator of interferon genes (STING) agonist with systemic antitumor effect
期刊论文
OAI收割
MEDCOMM, 2025, 卷号: 6, 期号: 1, 页码: e70001
作者:
Wang, Xiyuan
;
Zhan, Zhengsheng
;
Wang, Zhen
;
Zhang, Yan
;
Zhao, Kaiyan
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Synergistic immune augmentation enabled by covalently conjugating TLR4 and NOD2 agonists
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 278, 页码: 15
作者:
Ding, Dong
;
Gao, Runing
;
Lei, Yujuan
;
Liu, Jianing
;
Zhou, Chengkai
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The antidepressant-like effect and proposed mechanism of action of TPN672MA, a novel serotonin-dopamine receptor modulator for the treatment of schizophrenia
期刊论文
OAI收割
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 2024, 卷号: 242, 页码: 13
作者:
Cheng, Jiaxin
;
Wu, Chunhui
;
Wang, Yu
;
Wang, Zhen
;
He, Yang
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FXR activation remodels hepatic and intestinal transcriptional landscapes in metabolic dysfunction-associated steatohepatitis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 15
作者:
Wen, Ying-quan
;
Zou, Zi-yuan
;
Zhao, Guan-guan
;
Zhang, Meng-jiao
;
Zhang, Yong-xin
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