中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [13]
上海生物化学与细胞生... [7]
金属研究所 [5]
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期刊论文 [62]
SCI/SSCI论文 [4]
学位论文 [1]
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2025 [2]
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2021 [8]
2020 [2]
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Discovery of 2,4-quinazolinedione derivatives as LC3B recruiters in the facilitation of protein complex degradations
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 287, 页码: 10
作者:
Zeng, Yanping
;
Xiao, Jian
;
Shi, Li
;
Li, Yangsha
;
Xu, Yuanxin
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2025/04/01
LC3B
CDK9
Degradation
Protein complex
Discovery of SET domain-binding primary alkylamine-tethered degraders for the simultaneous degradation of NSD2-long and RE-IIBP isoforms
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 283, 页码: 17
作者:
Hu, Linghao
;
Xu, Hesong
;
Xu, Ye
;
Chen, Haowen
;
Jiang, Hanrui
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2025/04/01
NSD2
RE-IIBP
Targeted protein degradation
Multiple myeloma
Efficient biodegradation of poly(butylene adipate-co-terephthalate) in mild temperature by cutinases derived from a marine fungus
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2024, 卷号: 480, 页码: 12
作者:
Fei, Fan
;
Su, Zhenjie
;
Liu, Rui
;
Gao, Rongrong
;
Sun, Chaomin
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/12/20
PBAT degradation
Marine fungus
Cutinase
Mild temperature
Protein engineering
An overview of PROTACs targeting MDM2 as a novel approach for cancer therapy
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 272, 页码: 8
作者:
Li, Huiwen
;
Cai, Xinhui
;
Yang, Xiaoyu
;
Zhang, Xuan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/09/26
MDM2
PROTAC
p53
MDMX
Targeted protein degradation
Accelerating PROTACs Discovery Through a Direct-to-Biology Platform Enabled by Modular Photoclick Chemistry
期刊论文
OAI收割
ADVANCED SCIENCE, 2024, 页码: 12
作者:
Yan, Ke-Nian
;
Nie, Yong-Qiang
;
Wang, Jia-Yu
;
Yin, Guang-Liang
;
Liu, Qia
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2024/05/31
High-throughput chemical synthesis
modular synthesis
photoclick chemistry
PROTACs library
targeted protein degradation
Tumor-targeted PROTAC prodrug nanoplatform enables precise protein degradation and combination cancer therapy
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2024, 页码: 12
作者:
Zou, Zhi-feng
;
Yang, Lei
;
Nie, Hui-jun
;
Gao, Jing
;
Lei, Shu-min
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/05/22
proteolysis-targeting chimeras
tumor-targeted delivery
precise protein degradation
combination therapy
triple-negative breast cancer
Discovery of HyT-Based Degraders of CDK9-Cyclin T1 Complex
期刊论文
OAI收割
CHEMISTRY & BIODIVERSITY, 2023, 页码: 10
作者:
Lin, Rongkun
;
Yang, Jie
;
Liu, Ting
;
Wang, Mingyu
;
Ke, Chongrong
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2023/10/17
CDK9
cyclin T1
degrader
hydrophobic tag
protein degradation
Stimuli-activatable PROTACs for precise protein degradation and cancer therapy
期刊论文
OAI收割
SCIENCE BULLETIN, 2023, 卷号: 68, 期号: 10, 页码: 1069-1085
作者:
Gao, Jing
;
Yang, Lei
;
Lei, Shumin
;
Zhou, Feng
;
Nie, Huijun
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/10/17
PROTAC
Stimuli-activatable prodrug
Precise protein degradation
Nanomedicine
Combinatory therapy
Parallel evolution of two AIM24 protein subfamilies and their conserved functions in ER stress tolerance in land plants
期刊论文
OAI收割
PLANT COMMUNICATIONS, 2023, 卷号: 4, 期号: 3, 页码: 100513
作者:
Guan,Yanlong
;
Chang,Guanxiao
;
Zhao,Jinjie
;
Wang,Qia
;
Qin,Jiali
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/07/17
Physcomitrium
Marchantia
unfolded protein response
lncRNA
AGROBACTERIUM-MEDIATED TRANSFORMATION
RETICULUM-ASSOCIATED DEGRADATION
ENDOPLASMIC-RETICULUM
TRANSCRIPTION FACTOR
VEGETATIVE GROWTH
ARABIDOPSIS
MUTAGENESIS
EXPRESSION
RESPONSES
GENES
Insights into the mechanisms involved in the fungal degradation of plastics
期刊论文
OAI收割
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2023, 卷号: 262, 页码: 115202
作者:
Okal,Eyalira Jacob
;
Heng,Gui
;
Magige,Ephie A.
;
Khan,Sehroon
;
Wu,Shixi
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/07/22
Plastic biodegradation
Pre-treatment
Enzyme hydrolysis
Prooxidants
Molecular mechanisms
SURFACE BINDING-PROTEIN
WHITE-ROT FUNGI
MICROBIAL-DEGRADATION
MANGANESE PEROXIDASE
LIGNIN PEROXIDASE
GENE-EXPRESSION
POLYETHYLENE TEREPHTHALATE
TRANSCRIPTIONAL REGULATION
BIOLOGICAL DEGRADATION
ENZYMATIC DEGRADATION