机构

• 上海药物研究所 [8]

采集方式

• OAI收割 [8]

内容类型

• 期刊论文 [8]

发表日期

• 2024 [1]
• 2023 [1]
• 2022 [1]
• 2021 [1]
• 2020 [1]
• 2017 [1]
• 更多

学科主题

筛选

浏览/检索结果: 共8条，第1-8条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择题名升序题名降序提交时间升序提交时间降序作者升序作者降序发表日期升序发表日期降序 Design, synthesis and structure-activity relationship of 1,8-naphthalimide derivatives as highly potent hCYP1B1 inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107, 页码: 8 作者:  Wei, Yueyue;  Xiong, Yuan;  Liao, Qingyi;  Yang, Ya;  Tian, Tian   |  收藏  |  浏览/下载：8/0  |  提交时间：2024/07/12 8-naphthalimide  Structure -activity relationships (SAR)  Paclitaxel (PTX) resistance  Molecular docking   Discovery of seven-membered ring berberine analogues as highly potent and specific hCES2A inhibitors 期刊论文  OAI收割 CHEMICO-BIOLOGICAL INTERACTIONS, 2023, 卷号: 378, 页码: 11 作者:     |  收藏  |  浏览/下载：34/0  |  提交时间：2023/10/17 Human carboxylesterase 2 (hCES2A)  Berberine analogues  Structure -activity relationships (SAR)  Inhibition kinetics  Selectivity   Synthesis and Biochemical Evaluation of 8H-Indeno[1,2-d]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors 期刊论文  OAI收割 MOLECULES, 2022, 卷号: 27, 期号: 10, 页码: 11 作者:  Wu, Jing;  Feng, Bo;  Gao, Li-Xin;  Zhang, Chun;  Li, Jia   |  收藏  |  浏览/下载：41/0  |  提交时间：2022/08/16 COVID-19  M-pro inhibitors  drug design and synthesis  structure-activity relationships (SAR)   Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13 作者:  Meng, Xiang-Dong;  Gao, Li-Xin;  Wang, Zhi-Jia;  Feng, Bo;  Zhang, Chun   |  收藏  |  浏览/下载：74/0  |  提交时间：2021/12/01 2,5-diphenyl-1,3,4-oxadiazole derivatives  SHP2  Inhibitors  Structure-activity relationships (SAR)   Synthesis and biological evaluation of heterocyclic bis-aryl amides as novel Src homology 2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 11, 页码: 5 作者:  Satheeshkumar, Rajendran;  Zhu, Rui;  Feng, Bo;  Huang, Chao;  Gao, Ya   |  收藏  |  浏览/下载：48/0  |  提交时间：2020/07/01 Heterocyclic bis-aryl amides  PTP1B  SHP2  Inhibitors  Structure-activity relationships (SAR)   Benzo[c][1,2,5] thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 23, 页码: 5154-5157 作者:  Wang, Wen-Long;  Chen, Xiao-Yu;  Gao, Ya;  Gao, Li-Xin;  Sheng, Li   |  收藏  |  浏览/下载：35/0  |  提交时间：2019/01/08 Benzo[c][1,2,5] thiadiazole derivatives  PTP1B  SHP2  Inhibitors  Structure-activity relationships (SAR)   1H-2,3-Dihydroperimidine Derivatives: A New Class of Potent Protein Tyrosine Phosphatase 1B Inhibitors 期刊论文  OAI收割 MOLECULES, 2014, 卷号: 19, 期号: 1, 页码: 102-121 作者:  Wang, Wen-Long;  Yang, Dong-Lin;  Gao, Li-Xin;  Tang, Chun-Lan;  Ma, Wei-Ping   |  收藏  |  浏览/下载：29/0  |  提交时间：2019/01/08 1H-2,3-dihydroperimidine derivatives  PTP1B  inhibitors  selectivity  structure-activity relationships (SAR)   Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 卷号: 18, 期号: 5, 页码: 1773-1782 作者:  Ye, Deju;  Zhang, Yu;  Wang, Fei;  Zheng, Mingfang;  Zhang, Xu   |  收藏  |  浏览/下载：14/0  |  提交时间：2019/01/08 Protein tyrosine phosphatase 1B (PTP1B)  Inhibitors  Thiophene  Structure-activity relationships (SAR)