机构

• 上海药物研究所 [33]
• 昆明植物研究所 [8]
• 昆明动物研究所 [6]
• 南海海洋研究所 [2]
• 金属研究所 [2]
• 大连化学物理研究所 [2]
• 更多

采集方式

• OAI收割 [60]
• iSwitch采集 [1]

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浏览/检索结果: 共61条，第1-10条 帮助 条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择作者升序作者降序题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序 Design, synthesis and structure-activity relationship of 1,8-naphthalimide derivatives as highly potent hCYP1B1 inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 107, 页码: 8 作者:  Wei, Yueyue;  Xiong, Yuan;  Liao, Qingyi;  Yang, Ya;  Tian, Tian   |  收藏  |  浏览/下载：10/0  |  提交时间：2024/07/12 8-naphthalimide  Structure -activity relationships (SAR)  Paclitaxel (PTX) resistance  Molecular docking   Ecto-nucleotide pyrophosphatase/phosphodiesterase 1 inhibitors: Research progress and prospects 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 267, 页码: 13 作者:  Guan, Dezhong;  Fang, Lincheng;  Feng, Mingshun;  Guo, Shi;  Xie, Lingfeng   |  收藏  |  浏览/下载：16/0  |  提交时间：2024/05/07 ENPP1 inhibitors  cGAS-STING pathway  2 ', 3 '-cGAMP  Tumor immunotherapy   Discovery of GPX4 inhibitors through FP-based high-throughput screening 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14 作者:  Cao, Yu;  Wu, Bin;  Xu, Ying;  Wang, Mingchen;  Wu, Xinyu   |  收藏  |  浏览/下载：53/0  |  提交时间：2024/02/27 GPX4 inhibitor  HTS assay  Ferroptosis  Fluorescence polarization   Discovery of seven-membered ring berberine analogues as highly potent and specific hCES2A inhibitors 期刊论文  OAI收割 CHEMICO-BIOLOGICAL INTERACTIONS, 2023, 卷号: 378, 页码: 11 作者:  Yang, Yun   |  收藏  |  浏览/下载：35/0  |  提交时间：2023/10/17 Human carboxylesterase 2 (hCES2A)  Berberine analogues  Structure -activity relationships (SAR)  Inhibition kinetics  Selectivity   Synthesis and Biochemical Evaluation of 8H-Indeno[1,2-d]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors 期刊论文  OAI收割 MOLECULES, 2022, 卷号: 27, 期号: 10, 页码: 11 作者:  Wu, Jing;  Feng, Bo;  Gao, Li-Xin;  Zhang, Chun;  Li, Jia   |  收藏  |  浏览/下载：44/0  |  提交时间：2022/08/16 COVID-19  M-pro inhibitors  drug design and synthesis  structure-activity relationships (SAR)   Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors 期刊论文  OAI收割 BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13 作者:  Meng, Xiang-Dong;  Gao, Li-Xin;  Wang, Zhi-Jia;  Feng, Bo;  Zhang, Chun   |  收藏  |  浏览/下载：78/0  |  提交时间：2021/12/01 2,5-diphenyl-1,3,4-oxadiazole derivatives  SHP2  Inhibitors  Structure-activity relationships (SAR)   分子模拟应用于岩藻糖化糖胺聚糖 3D 结构确定及其与内源 性因子 X 酶的相互作用模式考察 学位论文  OAI收割 2021 作者:  陈鼎元   |  收藏  |  浏览/下载：9/0  |  提交时间：2023/11/02 Exploration of the SAR Connection between Morphinan- and Arylacetamide-Based kappa Opioid Receptor (kappa OR) Agonists Using the Strategy of Bridging 期刊论文  OAI收割 ACS CHEMICAL NEUROSCIENCE, 2021, 卷号: 12, 期号: 6, 页码: 1018-1030 作者:  Liu, Xiao;  Jiang, Shuang;  Kong, Linghui;  Ye, Rongrong;  Xiao, Li   |  收藏  |  浏览/下载：100/0  |  提交时间：2021/05/24 Morphinans  arylacetamidyl substituent  kappa opioid receptor modulators  structure-activity relationships   Synthesis and Structure-Activity Relationships of Ring-Opened Bengamide Analogues against Methicillin-Resistant Staphylococcus aureus(dagger) 期刊论文  OAI收割 CHINESE JOURNAL OF CHEMISTRY, 2021, 卷号: 39, 期号: 3, 页码: 671-676 作者:  Yu, Chen-Xi;  Wei, Bing-Yan;  Kong, Xue-Qing;  Yang, Cai-Guang;  Nan, Fa-Jun   |  收藏  |  浏览/下载：33/0  |  提交时间：2021/05/24 Bengamides  Staphylococcus aureus  Antibiotics  Structure‐  activity relationships  Pharmacokinetic   Chemical Synthesis of the Nucleoside Antibiotic Capuramycin 期刊论文  OAI收割 EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 2021, 期号: 26, 页码: 3681-3689 作者:  Xiao,Guozhi;  He,Haiqing   |  收藏  |  浏览/下载：26/0  |  提交时间：2022/04/02 Capuramycin  Chemical synthesis  Glycosyl ortho-(1-phenylvinyl)benzoates  One-pot glycosylation  Tuberculosis  DRUG-RESISTANT TUBERCULOSIS  GLUTAMIC-ACID-DERIVATIVES  MULTIDRUG-RESISTANT  PROTECTING GROUPS  IN-VITRO  GLYCOSYLATION  INHIBITORS  ALCOHOLS  ANALOGS  OXIDATION