中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2021 [14]
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Discovery of a Novel Androgen Receptor Antagonist Manifesting Evidence to Disrupt the Dimerization of the Ligand-Binding Domain via Attenuating the Hydrogen-Bonding Network Between the Two Monomers 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64
作者:  
Fu, Weitao;  Zhang, Minkui;  Liao, Jianing;  Tang, Qing;  Lei, Yixuan
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/03/21
Structures of the human cholecystokinin receptors bound to agonists and antagonists 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 卷号: 17, 期号: 12, 页码: 1230-1237
作者:  
Zhang, Xuefeng;  He, Chenglin;  Wang, Mu;  Zhou, Qingtong;  Yang, Dehua
  |  收藏  |  浏览/下载:16/0  |  提交时间:2024/03/21
Structure-Based Design of Dual-Acting Compounds Targeting Adenosine A(2A) Receptor and Histone Deacetylase as Novel Tumor Immunotherapeutic Agents 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16573-16597
作者:  
Yan, Wenzhong;  Ling, Lijun;  Wu, Yiran;  Yang, Kexin;  Liu, Ruiquan
  |  收藏  |  浏览/下载:16/0  |  提交时间:2022/06/15
Glycan Epitopes and Potential Glycoside Antagonists of DC-SIGN Involved in COVID-19: In Silico Study 期刊论文  OAI收割
BIOMOLECULES, 2021, 卷号: 11, 期号: 11, 页码: 16
作者:  
Gao, Meina;  Li, Hui;  Ye, Chenghao;  Chen, Kaixian;  Jiang, Hualiang
  |  收藏  |  浏览/下载:53/0  |  提交时间:2022/01/04
Constitutive signal bias mediated by the human GHRHR splice variant 1 期刊论文  OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:  
Cong, Zhaotong;  Zhou, Fulai;  Zhang, Chao;  Zou, Xinyu;  Zhang, Huibing
  |  收藏  |  浏览/下载:57/0  |  提交时间:2021/12/01
Supramolecular Antagonists Promote Mitochondrial Dysfunction 期刊论文  OAI收割
NANO LETTERS, 2021, 卷号: 21, 期号: 13, 页码: 5730-5737
作者:  
Li, Mingming;  Song, Yanqiu;  Song, Na;  Wu, Guangyao;  Zhou, Hao
  |  收藏  |  浏览/下载:31/0  |  提交时间:2021/08/17
Affinity Mass Spectrometry-Based Fragment Screening Identified a New Negative Allosteric Modulator of the Adenosine A(2A) Receptor Targeting the Sodium Ion Pocket 期刊论文  OAI收割
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 6, 页码: 991-1002
作者:  
Lu, Yan;  Liu, Hongyue;  Yang, Dehua;  Zhong, Li;  Xin, Ye
  |  收藏  |  浏览/下载:52/0  |  提交时间:2021/08/17
Amygdala dynorphin/kappa opioid receptor system modulates depressive-like behavior in mice following chronic social defeat stress 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  
Zan, Gui-ying;  Sun, Xiang;  Wang, Yu-jun;  Liu, Rui;  Wang, Chen-yao
  |  收藏  |  浏览/下载:42/0  |  提交时间:2021/08/17
Discovery of 1,5-Dihydro-4H-imidazol-4-one Derivatives as Potent, Selective Antagonists of CXC Chemokine Receptor 2 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 5, 页码: 836-845
作者:  
Che, Jinxin;  Wang, Zhilong;  Shen, Zheyuan;  Zhuang, Weihao;  Ying, Huazhou
  |  收藏  |  浏览/下载:18/0  |  提交时间:2021/08/17
Structural basis for ligand recognition of the neuropeptide Y Y-2 receptor 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 9
作者:  
Tang, Tingting;  Hartig, Christin;  Chen, Qiuru;  Zhao, Wenli;  Kaiser, Anette
  |  收藏  |  浏览/下载:23/0  |  提交时间:2021/05/24