机构

• 上海药物研究所 [179]

采集方式

• OAI收割 [179]

内容类型

• 期刊论文 [175]
• 会议论文 [2]
• 学位论文 [2]

发表日期

• 2024 [4]
• 2023 [7]
• 2022 [15]
• 2021 [13]
• 2020 [11]
• 2019 [3]
• 更多

学科主题

• Pharmacolo... [4]
• Chemistry [3]
• Biochemist... [2]

筛选

浏览/检索结果: 共179条，第1-10条 帮助 限定条件 专题：上海药物研究所    第一署名单位    第一作者单位    通讯作者单位     条数/页： 5101520253035404550556065707580859095100 排序方式： 请选择提交时间升序提交时间降序题名升序题名降序作者升序作者降序发表日期升序发表日期降序 Discovery of YFJ-36: Design, Synthesis, and Antibacterial Activities of Catechol-Conjugated β-Lactams against Gram-Negative Bacteria 期刊论文  OAI收割 JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21 作者:  Liu, Fangjun;  Kou, Qunhuan;  Li, Hongyuan   |  收藏  |  浏览/下载：0/0  |  提交时间：2024/05/22 Ecto-nucleotide pyrophosphatase/phosphodiesterase 1 inhibitors: Research progress and prospects 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 267, 页码: 13 作者:  Guan, Dezhong;  Fang, Lincheng;  Feng, Mingshun;  Guo, Shi;  Xie, Lingfeng   |  收藏  |  浏览/下载：1/0  |  提交时间：2024/05/07 ENPP1 inhibitors  cGAS-STING pathway  2 ', 3 '-cGAMP  Tumor immunotherapy   Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors 期刊论文  OAI收割 ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13 作者:  Yan, Chao;  Zhang, Qian;  Xiao, Pan;  Xie, Xinyun;  Li, Ming   |  收藏  |  浏览/下载：38/0  |  提交时间：2024/03/25 RNA modification  m(6)A  FTO  anticancer   Discovery of GPX4 inhibitors through FP-based high-throughput screening 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14 作者:  Cao, Yu;  Wu, Bin;  Xu, Ying;  Wang, Mingchen;  Wu, Xinyu   |  收藏  |  浏览/下载：26/0  |  提交时间：2024/02/27 GPX4 inhibitor  HTS assay  Ferroptosis  Fluorescence polarization   Assessment of the structure-activity relationship and antileukemic activity of diacylpyramide compounds as human ClpP agonists 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 258, 页码: 17 作者:  Zhang, Ranran;  Wang, Pengyu;  Wei, Bingyan;  Chen, Liang;  Song, Xiaomin   |  收藏  |  浏览/下载：22/0  |  提交时间：2023/10/17 ClpP agonists  Structure-activity relationship  Mitochondrial respiratory chain  Antileukemic therapy   Design, synthesis and biological evaluation of salicylanilides as novel allosteric inhibitors of human pancreatic lipase 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 91, 页码: 11 作者:  Zhao, Yitian;  Zhang, Min;  Hou, Xudong;  Han, Jiaxin;  Qin, Xiaoya   |  收藏  |  浏览/下载：12/0  |  提交时间：2023/10/17 Salicylanilide  hPL inhibitor  Structure -activity relationship  Anti -obesity   Discovery of novel triazine derivatives as potent retinoic acid receptor-related orphan receptor gamma t (ROR gamma t) inverse agonists 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 256, 页码: 18 作者:  Lu, Lixue;  Chen, Song;  Yu, Mingcheng;  Zhou, Ronghui;  Guo, Siqi   |  收藏  |  浏览/下载：16/0  |  提交时间：2023/10/17 ROR gamma t  Triazines  Inverse agonist  Psoriasis  Autoimmune diseases   Structure-based discovery of potent USP28 inhibitors derived from Vismodegib 期刊论文  OAI收割 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 254, 页码: 15 作者:  Zhou, Di;  Xu, Zhuo;  Huang, Yaodong;  Wang, Hui;  Zhu, Xiaoli   |  收藏  |  浏览/下载：25/0  |  提交时间：2023/10/17 USP28  Structure-based  Vismodegib derivatives  Structure-activity relationships  c-Myc   Discovery of seven-membered ring berberine analogues as highly potent and specific hCES2A inhibitors 期刊论文  OAI收割 CHEMICO-BIOLOGICAL INTERACTIONS, 2023, 卷号: 378, 页码: 11 作者:  Yang, Yun;  Xiong, Yuan;  Zhu, Guanghao;  Sun, Mengru;  Zou, Kun   |  收藏  |  浏览/下载：24/0  |  提交时间：2023/10/17 Human carboxylesterase 2 (hCES2A)  Berberine analogues  Structure -activity relationships (SAR)  Inhibition kinetics  Selectivity   Design, synthesis, and evaluation of pyrido.[3,4-b]pyrazin-2(1H)-one derivatives as potent FLT3 inhibitors 期刊论文  OAI收割 BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 79, 页码: 117155 作者:  Sun, Mei;  Wang, Chang;  Wang, Peipei;  Ye, Qingqing;  Zhou, Yubo   |  收藏  |  浏览/下载：2/0  |  提交时间：2024/04/09 FLT3  FLT3-D835Y  Acute myeloid leukemia  Structure -activity relationships