中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
机构
  • 上海药物研究所 [20]
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内容类型
发表日期
  • 2021 [20]
学科主题
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浏览/检索结果: 共20条,第1-10条 帮助

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Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 22, 页码: 16650-16674
作者:  
Zhang, Zhuqing;  Guo, Zuhao;  Xu, Xiaowei;  Cao, Danyan;  Yang, Hong
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 11
作者:  
Fan, Shijie;  Yue, Liyan;  Wan, Wei;  Zhang, Yuanyuan;  Zhang, Bidong
  |  收藏  |  浏览/下载:98/0  |  提交时间:2021/12/16
DRAK2 aggravates nonalcoholic fatty liver disease progression through SRSF6-associated RNA alternative splicing 期刊论文  OAI收割
CELL METABOLISM, 2021, 卷号: 33, 期号: 10, 页码: 2004-+
作者:  
Li, Yufeng;  Xu, Junyu;  Lu, Yuting;  Bian, Hua;  Yang, Lin
  |  收藏  |  浏览/下载:49/0  |  提交时间:2022/01/18
Recombinant cancer nanovaccine for targeting tumor-associated macrophage and remodeling tumor microenvironment 期刊论文  OAI收割
NANO TODAY, 2021, 卷号: 40, 页码: 14
作者:  
Tang, Yisi;  Fan, Wufa;  Chen, Guihua;  Zhang, Meng;  Tang, Xueping
  |  收藏  |  浏览/下载:41/0  |  提交时间:2021/12/01
Kynurenine derivative 3-HAA is an agonist ligand for transcription factor YY1 期刊论文  OAI收割
Journal of Hematology & Oncology, 2021, 卷号: 14, 期号: 1
作者:  
Shi,Zhaopeng;  Gan,Guifang;  Xu,Xiang;  Zhang,Jieying
  |  收藏  |  浏览/下载:36/0  |  提交时间:2021/11/04
Nuclear UHRF1 is a gate-keeper of cellular AMPK activity and function 期刊论文  OAI收割
CELL RESEARCH, 2021, 页码: 18
作者:  
Xu, Xiang;  Ding, Guangjin;  Liu, Caizhi;  Ding, Yuhan;  Chen, Xiaoxin
  |  收藏  |  浏览/下载:53/0  |  提交时间:2021/11/04
Discovery of potential small molecular SARS-CoV-2 entry blockers targeting the spike protein 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  
Wang, Lin;  Wu, Yan;  Yao, Sheng;  Ge, Huan;  Zhu, Ya
  |  收藏  |  浏览/下载:94/0  |  提交时间:2021/11/04
Facing small and biased data dilemma in drug discovery with enhanced federated learning approaches 期刊论文  OAI收割
SCIENCE CHINA-LIFE SCIENCES, 2021, 页码: 11
作者:  
Xiong, Zhaoping;  Cheng, Ziqiang;  Lin, Xinyuan;  Xu, Chi;  Liu, Xiaohong
  |  收藏  |  浏览/下载:23/0  |  提交时间:2021/11/04
Polyoxypregnanes as safe, potent, and specific ABCB1-inhibitory pro-drugs to overcome multidrug resistance in cancer chemotherapy in vitro and in vivo 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 7, 页码: 1885-1902
作者:  
Wu, Xu;  Yin, Chun;  Ma, Jiang;  Chai, Stella;  Zhang, Chunyuan
  |  收藏  |  浏览/下载:43/0  |  提交时间:2021/11/04
Structures of human mGlu2 and mGlu7 homo- and heterodimers 期刊论文  OAI收割
NATURE, 2021, 卷号: 594, 期号: 7864, 页码: 589-+
作者:  
Du, Juan;  Wang, Dejian;  Fan, Hongcheng;  Xu, Chanjuan;  Tai, Linhua
  |  收藏  |  浏览/下载:33/0  |  提交时间:2021/08/17