中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [187]
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Modular Biomimetic Strategy Enabled Discovery of Simplified Pseudo-Natural Macrocyclic P-Glycoprotein Inhibitors Capable of Overcoming Multidrug Resistance
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 4, 页码: 2550-2565
作者:
Liu, Bo
;
Yu, Xueni
;
Liu, Liping
;
Wang, Lei
;
Wang, Jie
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 12
作者:
Zhang, Yinyong
;
Yang, Yushe
;
Meng, Xin
;
Zhou, Xianli
;
Guo, Bin
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
oxazolidinone
asymmetric reduction
fused ring
process development
crystal transformation
Time- and dose-dependent detoxification and reproductive endocrine disruption induced by tetrabromobisphenol A (TBBPA) in mussel Mytilus galloprovincialis
期刊论文
OAI收割
MARINE ENVIRONMENTAL RESEARCH, 2023, 卷号: 183, 页码: 10
作者:
Wang, Shuang
;
Sun, Zuodeng
;
Ren, Chuanbo
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/08/17
Tetrabromobisphenol A
Detoxification
Reproductive endocrine disruption
Sulfation
Mytilus galloprovincialis
Anti-infective therapy using species-specific activators of Staphylococcus aureus ClpP
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 16
作者:
Wei, Bingyan
;
Zhang, Tao
;
Wang, Pengyu
;
Pan, Yihui
;
Li, Jiahui
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2023/04/10
Drug Degradation Caused by mce3R Mutations Confers Contezolid (MRX-I) Resistance in Mycobacterium tuberculosis
期刊论文
OAI收割
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2022, 卷号: 66, 期号: 10, 页码: 11
作者:
Pi, Rui
;
Chen, Xiaomin
;
Meng, Jian
;
Liu, Qingyun
;
Chen, Yiwang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/11/11
Mycobacterium tuberculosis
drug resistance
contezolid
Mce3R
Rv1936
degradation
drug resistance mechanisms
Targeted delivery and enhanced uptake of chemo-photodynamic nanomedicine for melanoma treatment
期刊论文
OAI收割
ACTA BIOMATERIALIA, 2022, 卷号: 147, 页码: 356-365
作者:
Huang, Xiaobei
;
Mu, Ning
;
Ding, Yuanfu
;
Lam, Hou Wang
;
Yue, Ludan
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/08/22
Photodynamic-chemotherapeutic therapy
Pt(IV) prodrug
Charge -reversal
Targeted drug delivery
Controlled drug release
Zinc oxide/graphene oxide nanocomposites efficiently inhibited cadmium-induced hepatotoxicity via releasing Zn ions and up-regulating MRP1 expression
期刊论文
OAI收割
ENVIRONMENT INTERNATIONAL, 2022, 卷号: 165
作者:
Liu, Yun
;
Wang, Xue
;
Si, Bo
;
Wang, Tong
;
Wu, Yun
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/12/23
Cadmium
Zinc oxide
Graphene oxide
Detoxification
Bioaccumulation
Magnetic resonance imaging
Concise Total Synthesis of Dysoxylactam A and a Simplified Analog
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2022, 页码: 8
作者:
Yang, Guan-Zhou
;
Wang, Lei
;
Fan, Yao-Yue
;
Lai, Zeng-Wei
;
Yu, Xue-Ni
  |  
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2022/08/16
Total synthesis
Dysoxylactam A
Macrocyclolipopeptide
Reversing multidrug resistance
Structure-activity relationship
Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:
Lei, E.
;
Tao, Huanyu
;
Jiao, Shang
;
Yang, Anming
;
Zhou, Yu
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/08/16
Antimicrobial peptide antibiotics inhibit aerobic denitrification via affecting electron transportation and remolding carbon metabolism
期刊论文
OAI收割
JOURNAL OF HAZARDOUS MATERIALS, 2022, 卷号: 431, 期号: 0, 页码: 128616
作者:
Wang, Na
;
Gao, Jie
;
Wang, Qiuying
;
Xiao, Shujie
;
Zhuang, Guoqiang
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2022/11/09
MICROBIAL DENITRIFICATION
PARACOCCUS-DENITRIFICANS
COMMUNITY STRUCTURE
NITRATE
TREHALOSE
NITROGEN
WATER
REMOVAL
NITRIFICATION
PERFORMANCE