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上海药物研究所 [109]
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OAI收割 [158]
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期刊论文 [154]
学位论文 [4]
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2022 [158]
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Biochemist... [2]
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发表日期:2022
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Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:
Li, Ennian
;
Wang, Kai
;
Zhang, Bei
;
Guo, Siqi
;
Xiao, Senhao
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/08/16
DNMT1 inhibitor
A549 cell lines
HCT116 cell lines
antitumor activity
pharmacokinetic
Identification of 1H-pyrazolo[3,4-b]pyridine derivatives as novel and potent TBK1 inhibitors: design, synthesis, biological evaluation, and molecular docking study
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1411-1425
作者:
Sun, Yin
;
Tang, Haotian
;
Wang, Xiaoyan
;
Feng, Fang
;
Fan, Tiantian
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2022/08/16
TBK1 inhibitors
1H-pyrazolo[3
4-b]pyridine
structure-activity relationships (SARs)
immune response
cancer therapy
PD-L1 Aptamer-Functionalized Metal-Organic Framework Nanoparticles for Robust Photo-Immunotherapy against Cancer with Enhanced Safety
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 页码: 9
作者:
Zhang, Jingfang
;
Li, Wenzhe
;
Qi, Yafei
;
Wang, Guorong
;
Li, Lele
  |  
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2023/02/22
DNA Nanotechnology
Immunotherapy
Metal-Organic Frameworks
PD-L1 Aptamer
Spherical Nucleic Acids (SNAs)
Learning with uncertainty to accelerate the discovery of histone lysine-specific demethylase 1A (KDM1A/LSD1) inhibitors
期刊论文
OAI收割
BRIEFINGS IN BIOINFORMATICS, 2022, 页码: 14
作者:
Wang, Dong
;
Wu, Zhenxing
;
Shen, Chao
;
Bao, Lingjie
;
Luo, Hao
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/04/10
uncertainty estimation
graph neural network
KDM1A
LSD1 inhibitors
upper confidence bound method
virtual screening
Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:
Bi, Kaijian
;
Cheng, Junfei
;
He, Shipeng
;
Fang, Yuxin
;
Huang, Min
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
A novel coating with SiO2 anchored on MXene loading tannic acid for self-healing anticorrosive performance
期刊论文
OAI收割
JOURNAL OF ALLOYS AND COMPOUNDS, 2022, 卷号: 928, 页码: 10
作者:
Sun, Xiaoguang
;
Ma, Chengcheng
;
Ma, Fubin
;
Wang, Tong
;
Feng, Chao
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2023/01/06
TA@MXene-SiO2
Self-healing
Anticorrosion
Discovery of 10H-Benzo[b]pyrido[2,3-e][1,4]oxazine AXL Inhibitors via Structure-Based Drug Design Targeting c-Met Kinase
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:
Zhan, Zhengsheng
;
Ji, Yinchun
;
Su, Haixia
;
Fang, Chen
;
Peng, Xia
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2023/04/10
Dual inhibition of CHK1/FLT3 enhances cytotoxicity and overcomes adaptive and acquired resistance in FLT3-ITD acute myeloid leukemia
期刊论文
OAI收割
LEUKEMIA, 2022, 页码: 11
作者:
Jiang, Kailong
;
Li, Xuemei
;
Wang, Chang
;
Hu, Xiaobei
;
Wang, Peipei
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2023/04/10
Targeting the PI3K/AKT/mTOR Signaling Pathway in the Treatment of Human Diseases: Current Status, Trends, and Solutions
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 29
作者:
Huang, Jindi
;
Chen, Liye
;
Wu, Jiangxia
;
Ai, Daiqiao
;
Zhang, Ji-Quan
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10
Identification of a class of potent USP25/28 inhibitors with broad-spectrum anti-cancer activity
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 3
作者:
Peng, Jin
;
Jiang, Kun
;
Sun, Xiao
;
Wu, Lingzhi
;
Wang, Jiewei
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2023/04/10