中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [22]
大连化学物理研究所 [6]
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OAI收割 [53]
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期刊论文 [51]
会议论文 [1]
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Cryo-EM structures of cancer-specific helical and kinase domain mutations of PI3K alpha
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 46, 页码: 11
作者:
Liu, Xiao
;
Zhou, Qingtong
;
Hart, Jonathan R.
;
Xu, Yingna
;
Yang, Su
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/10/17
phosphoinositide 3-kinase (PI3K)
mass spectrometry
mutants
S3I-201 derivative incorporating naphthoquinone unit as effective STAT3 inhibitors: Design, synthesis and anti-gastric cancer evaluation
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 71
作者:
Li, Haobin
;
Cai, Maohua
;
Cao, Fei
;
Yu, Dehua
;
Yang, Jing
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/12/22
STAT3 inhibitor
Quinone derivative
S3I-201
Anti -gastric cancer drug
Nanobodies and chemical cross-links advance the structural and functional analysis of PI3K alpha
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2022, 卷号: 119, 期号: 38, 页码: 9
作者:
Hart, Jonathan R.
;
Liu, Xiao
;
Pan, Chen
;
Liang, Anyi
;
Ueno, Lynn
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
phosphoinositide 3-kinase (PI3K)
nanobody
conformational changes
chemical cross-linking
mass spectrometry
Vav2 is a novel APP-interacting protein that regulates APP protein level
期刊论文
OAI收割
SCIENTIFIC REPORTS, 2022, 卷号: 12
作者:
Zhang, Youjia
;
Yang, Xiaxin
;
Liu, Yongrui
;
Ge, Liang
;
Wang, Jiarong
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/12/23
SH2 Domain-Containing Phosphatase 2 Inhibition Attenuates Osteoarthritis by Maintaining Homeostasis of Cartilage Metabolism via the Docking Protein 1/Uridine Phosphorylase 1/Uridine Cascade
期刊论文
OAI收割
ARTHRITIS & RHEUMATOLOGY, 2022, 页码: 12
作者:
Liu, Qianqian
;
Zhai, Linhui
;
Han, Mingrui
;
Shi, Dongquan
;
Sun, Ziying
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
Cryo-EM structures of PI3K alpha reveal conformational changes during inhibition and activation
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 45, 页码: 9
作者:
Liu, Xiao
;
Yang, Su
;
Hart, Jonathan R.
;
Xu, Yingna
;
Zou, Xinyu
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2022/01/04
phosphoinositide 3-kinase (PI3K)
activation
inhibition
activity-dependent conformational changes
Rational drug design of benzothiazole-based derivatives as potent signal transducer and activator of transcription 3 (STAT3) signaling pathway inhibitors
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 216, 页码: 20
作者:
Gao, Dingding
;
Jin, Nan
;
Fu, Yixian
;
Zhu, Yueyue
;
Wang, Yujie
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2021/06/11
STAT3 signaling pathway
Benzothiazole
Rational design
Antitumor activity
Molecular docking
Biotoxic effects and gene expression regulation of urban PM2.5 in southwestern China
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2021, 卷号: 753, 页码: 11
作者:
Zhang, Shumin
;
Zhang, Jingping
;
Guo, Dongmei
;
Peng, Chao
;
Tian, Mi
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2020/12/30
PM2.5
Biotoxic
Transcriptome
Chengdu
Chongqing
Southwestern China
Biotoxic effects and gene expression regulation of urban PM2.5 in southwestern China
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2021, 卷号: 753, 页码: 11
作者:
Zhang, Shumin
;
Zhang, Jingping
;
Guo, Dongmei
;
Peng, Chao
;
Tian, Mi
  |  
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/02/24
PM2.5
Biotoxic
Transcriptome
Chengdu
Chongqing
Southwestern China
Biochemical and NMR characterization of the interactions of Vav2-SH2 domain with lipids and the EphA2 juxtamembrane region on membrane
期刊论文
OAI收割
BIOCHEMICAL JOURNAL, 2020, 卷号: 477
作者:
Ge, Liang
;
Wu, Bo
;
Zhang, Youjia
;
Wang, Jiarong
;
Zhao, Hongxin
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/12/07