中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [16]
采集方式
OAI收割 [16]
内容类型
期刊论文 [16]
发表日期
2022 [16]
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共16条,第1-10条
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发表日期:2022
内容类型:期刊论文
专题:上海药物研究所
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In vitro and in vivo evaluation of the main protease inhibitor FB2001 against SARS-CoV-2
期刊论文
OAI收割
ANTIVIRAL RESEARCH, 2022, 卷号: 208, 页码: 10
作者:
Shang, Weijuan
;
Dai, Wenhao
;
Yao, Cheng
;
Xu, Ling
;
Tao, Xiangming
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
SARS-CoV-2
SARS-CoV-2 variants
FB2001
Main protease
PBPK
Anti-SARS-CoV-2 in vivo
Discovery of Novel N-(5-(Pyridin-3-yl)-1H-indazol-3-yl)benzamide Derivatives as Potent Cyclin-Dependent Kinase 7 Inhibitors for the Treatment of Autosomal Dominant Polycystic Kidney Disease
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 19
作者:
Yang, Bowen
;
Zhang, Haoran
;
Li, Na
;
Gao, Lixin
;
Jiang, Hong
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2023/04/10
Absorption, distribution, metabolism, and excretion of [C-14]Mefuparib (CVL218), a novel PARP1/2 inhibitor, in rats
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2022, 页码: 12
作者:
Li, Xin-mei
;
Zheng, Yuan-dong
;
Zhang, Yi-fan
;
Huan, Xia-juan
;
Yang, Chen
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/12/13
[C-14]Mefuparib
Mefuparib (CVL218)
Blood-brain barrier
Mass balance
Tissue distribution
GastroPlus simulation
First clinical applications for the NIR-II imaging with ICG in microsurgery
期刊论文
OAI收割
FRONTIERS IN BIOENGINEERING AND BIOTECHNOLOGY, 2022, 卷号: 10, 页码: 1042546
作者:
Wu, Yifan
;
Suo, Yongkuan
;
Wang, Zheng
;
Yu, Yifeng
;
Duan, Shuang
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/03/21
indocyanine green (ICG)
near-infrared II (NIR-II) imaging
fluorescenceguided surgery
vascular anastomosis
flap reconstruction
Arylnaphthalide lignans from Saussurea medusa and their anti-inflammatory activities
期刊论文
OAI收割
ARABIAN JOURNAL OF CHEMISTRY, 2022, 卷号: 15, 期号: 10, 页码: 11
作者:
Cao, Jing-Ya
;
Dong, Qi
;
Wang, Zhi-Yao
;
Zhao, Ye
;
Ren, Yu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/12/13
Saussurea medusa
Arylnaphthalide lignan
Anti-inflammatory activity
ECD calculation
Molecular docking
Development of a variant of dinutuximab with enhanced antitumor efficacy and reduced induction of neuropathic pain
期刊论文
OAI收割
FEBS OPEN BIO, 2022, 卷号: 12, 期号: 9, 页码: 1644-1656
作者:
Liu, Xin-Yuan
;
Chen, Yi-Li
;
Liu, Guo-Jian
;
Deng, Xiang-Nan
;
Cui, Yue
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/09/30
ADCC
affinity maturation
antibody engineering
anti-GD2 antibodies
engineered Fc domain
humanized
Novel assays for quality evaluation of XueBiJing: Quality variability of a Chinese herbal injection for sepsis management
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL ANALYSIS, 2022, 卷号: 12, 期号: 4, 页码: 664-682
作者:
Yu, Xuan
;
Niu, Wei
;
Wang, Ya-Ya
;
Olaleye, Olajide E.
;
Wang, Jia-Nan
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/11/11
XueBiJing
Chinese herbal medicine
Quality variability
Quality marker
One -point calibration
A Traceless Site-Specific Conjugation on Native Antibodies Enables Efficient One-Step Payload Assembly
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 页码: 11
作者:
Zeng, Yue
;
Shi, Wei
;
Dong, Qian
;
Li, Wanzhen
;
Zhang, Jianxin
  |  
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2022/08/30
Acyl Transfer
Anti-Tumor
One-Step Synthesis
Site-Specific ADCs
Thioester
Antinociceptive activities and mechanism of action of Cepharanthine
期刊论文
OAI收割
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2022, 卷号: 614, 页码: 219-224
作者:
Wei, Xiang-Yan
;
Long, Jian-Dong
;
Chai, Jing-Rui
;
Chen, Jing
;
Gao, Jian-Ping
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/08/16
Cepharanthine
Antinociception
mu opioid receptors
Constipation
Structure-Activity Relationships and Antileukemia Effects of the Tricyclic Benzoic Acid FTO Inhibitors
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 17
作者:
Liu, Zeyu
;
Duan, Zongliang
;
Zhang, Deyan
;
Xiao, Pan
;
Zhang, Tao
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2022/08/30