中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [37]
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广州生物医药与健康... [12]
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期刊论文 [157]
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浏览/检索结果:
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The aminosteroid U73122 promotes oligodendrocytes generation and myelin formation
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 12
作者:
Cui, Shi-hao
;
Suo, Na
;
Yang, Ying
;
Wu, Xuan
;
Guo, Shi-meng
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/11
oligodendrocyte
oligodendrocyte progenitor cell
differentiation
remyelination
U73122
Development of a Novel 18F-Labeled Probe for PET Imaging of Estrogen Receptor beta
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 11
作者:
Zhou, Yujing
;
Lei, Peng
;
Han, Jiaxin
;
Wang, Zhiming
;
Ji, Aiyan
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2023/04/10
Advances in Medicinal Chemistry of Estrogen-related Receptor Alpha (ERRa) Inverse Agonists
期刊论文
OAI收割
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2023, 卷号: 23, 期号: 20, 页码: 1952-1963
作者:
Zhang, Haibin
;
Du, Yongli
;
Zheng, Yong
;
Lv, Huiting
;
Yan, Zhijia
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/10/17
ERRalpha
ERRalpha inverse agonists
Breast cancer
TNBC
Signaling pathways
Inverse agonistic activity
Binding and Activation of Estrogen-Related Receptor ?: A Novel Molecular Mechanism for the Estrogenic Disruption Effects of DDT and Its Metabolites
期刊论文
OAI收割
ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2022, 卷号: 56, 期号: 17, 页码: 12358-12367
作者:
Wang, Li
;
Qie, Yu
;
Yang, Yu
;
Zhao, Qiang
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2022/11/08
ERR-GAMMA
ALPHA
PESTICIDES
CANCER
Perfluorinated Iodine Alkanes Promoted Neural Differentiation of mESCs by Targeting miRNA-34a-5p in Notch-Hes Signaling
期刊论文
OAI收割
ENVIRONMENTAL SCIENCE & TECHNOLOGY, 2022, 卷号: 56, 期号: 12, 页码: 8496-8506
作者:
Ren, Zhihua
;
Ku, Tingting
;
Gao, Yurou
;
Yang, Xiaoxi
;
Meng, Lingyi
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2022/11/08
ENDOCRINE-DISRUPTING CHEMICALS
EMBRYONIC STEM-CELLS
ESTROGEN-RECEPTOR-ALPHA
IN-VITRO
BISPHENOL-A
GENERATION
EXPOSURE
BINDING
Discovery of Thieno[2,3-e]indazole Derivatives as Novel Oral Selective Estrogen Receptor Degraders with Highly Improved Antitumor Effect and Favorable Druggability br
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 7, 页码: 5724-5750
作者:
Lu, Zhengyu
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2022/08/16
Evaluation of the binding performance of flavonoids to estrogen receptor alpha by Autodock, Autodock Vina and Surflex-Dock
期刊论文
OAI收割
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2022, 卷号: 233, 期号: 0, 页码: 113323
作者:
Xue, Qiao
;
Liu, Xian
;
Russell, Paul
;
Li, Jin
;
Pan, Wenxiao
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2022/11/08
PROTEIN-LIGAND DOCKING
MOLECULAR DOCKING
DISCOVERY
FRAMEWORK
DYNAMICS
AFFINITY
The discovery of a novel series of potential ERR alpha inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo
期刊论文
OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 125-134
作者:
Gao, Zhipei
;
Wang, Tianxiao
;
Li, Rui
;
Du, Yongli
;
Lv, Han
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2022/01/18
ERR alpha
TNBC
p-Nitrobenzenesulfonamide
inverse agonist
Toxicity pathways of lipid metabolic disorders induced by typical replacement flame retardants via data-driven analysis, in silico and in vitro approaches
期刊论文
OAI收割
CHEMOSPHERE, 2022, 卷号: 287, 页码: 9
作者:
Wang, Xiaoqing
;
Wang, Li
;
Li, Fei
;
Teng, Yuefa
;
Ji, Chenglong
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/06/16
Toxicity pathways
Lipid metabolism disorder
Bibliometric analysis
Computational toxicology
Data-driven analysis
Ionizing radiation downregulates estradiol synthesis via endoplasmic reticulum stress and inhibits the proliferation of estrogen receptor-positive breast cancer cells
期刊论文
OAI收割
CELL DEATH & DISEASE, 2021, 卷号: 12, 期号: 11, 页码: 10
作者:
Yang, Pengfei
;
Feng, Xiu
;
Li, Jin
;
Zhang, Tianyi
;
Sheng, Chengyan
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/12/13