中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Discovery of GPX4 inhibitors through FP-based high-throughput screening
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 14
作者:
Cao, Yu
;
Wu, Bin
;
Xu, Ying
;
Wang, Mingchen
;
Wu, Xinyu
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/02/27
GPX4 inhibitor
HTS assay
Ferroptosis
Fluorescence polarization
Targeting ST8SIA6-AS1 counteracts KRAS
G12C
inhibitor resistance through abolishing the reciprocal activation of PLK1/c-Myc signaling
期刊论文
OAI收割
EXPERIMENTAL HEMATOLOGY & ONCOLOGY, 2023, 卷号: 12, 期号: 1, 页码: 22
作者:
Wang, Yafang
;
Yao, Mingyue
;
Li, Cheng
;
Yang, Kexin
;
Qin, Xiaolong
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/26
KRAS(G12C)
c-Myc
PLK1
LncRNA
ST8SIA6-AS1
Drug resistance
Recent advances in point-of-care testing of COVID-19
期刊论文
OAI收割
CHEMICAL SOCIETY REVIEWS, 2023, 卷号: 52, 期号: 24, 页码: 8500-8530
作者:
Lee, Sungwoon
;
Bi, Liyan
;
Chen, Hao
;
Lin, Dong
;
Mei, Rongchao
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/01/26
Discovery of JN122, a Spiroindoline-Containing Molecule that Inhibits MDM2/p53 Protein-Protein Interaction and Exerts Robust In Vivo Antitumor Efficacy
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 24, 页码: 16991-17025
作者:
Cheng, Jing
;
Yan, Ziqin
;
Jiang, Kailong
;
Liu, Chen
;
Xu, Dehua
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/02/19
Development, methodological evaluation and application of a cell-based TRF assay for analysis of ADCC activity
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2023, 卷号: 235, 页码: 7
作者:
Zhu, Xiao
;
Gong, Likun
;
Qin, Qiuping
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Antibody-dependent cell-mediated cytotoxicity
Time-resolved fluorescence
Monoclonal antibody
Antibody-Drug Conjugate
Eu
NK-92 cells
Molecular imprinting-based indirect fluorescence detection strategy implemented on paper chip for non-fluorescent microcystin
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 12
作者:
Li, Bowei
;
Qi, Ji
;
Liu, Feng
;
Zhao, Rongfang
;
Arabi, Maryam
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/01/26
Molecular imprinting-based indirect fluorescence detection strategy implemented on paper chip for non-fluorescent microcystin
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 12
作者:
Li, Bowei
;
Qi, Ji
;
Liu, Feng
;
Zhao, Rongfang
;
Arabi, Maryam
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2024/04/07
Discovery of a novel OGT inhibitor through high-throughput screening based on Homogeneous Time-Resolved Fluorescence (HTRF)
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 139, 页码: 12
作者:
Wu, Xinyu
;
Wang, Mingchen
;
Cao, Yu
;
Xu, Ying
;
Yang, Ziqun
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/02/27
O-GlcNAcylation
O-GlcNAc transferase
High-throughput screening
Inhibitor
Dual-Mode Undistorted Visual Fluorescent Sensing Strategy through Manipulating the Coffee-Ring Effect on Microfluidic Paper-Based Chip
期刊论文
OAI收割
ANALYTICAL CHEMISTRY, 2023, 卷号: 95, 期号: 28, 页码: 10486-10491
作者:
Qi, Ji
;
Li, Bowei
;
Lin, Dong
;
Du, Zhiqiang
;
Fu, Longwen
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2024/01/26
Discovery of new small molecule inhibitors of the BPTF bromodomain
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 134, 页码: 106453
作者:
Liang, Xiaochen
;
Cao, Yu
;
Duan, Zhe
;
Wang, Mingchen
;
Zhang, Naixia
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
BPTF bromodomain
BPTF inhibitors
HTRF
c-Myc