中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [121]
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Development of a potent benzonitrile-based inhibitor of glutaminyl-peptide cyclotransferase-like protein (QPCTL) with antitumor efficacy
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2023, 卷号: 8, 期号: 1, 页码: 3
作者:
Yu, Lei
;
Zhao, Pengcheng
;
Sun, Yaoliang
;
Zheng, Zening
;
Du, Wenhao
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/01/26
Self-Adaptive Nanoregulator to Mitigate Dynamic Immune Evasion of Pancreatic Cancer
期刊论文
OAI收割
ADVANCED MATERIALS, 2023, 页码: 16
作者:
Pan, Jiaxing
;
Lai, Yi
;
Zhang, Shunan
;
Zhang, Huijuan
;
Shan, Yiming
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2023/12/08
cancer-associated fibroblasts
immune evasion
nanoregulator
pancreatic ductal adenocarcinoma
peptide-drug conjugate
Targeting lactate metabolism and immune interaction in breast tumor via protease-triggered delivery
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2023, 卷号: 358, 页码: 706-717
作者:
Zhao, Pengfei
;
Wang, Shuang
;
Jiang, Jizong
;
Gao, Yanrong
;
Wang, Yuewei
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Legumain
Lactate
Tumor immune microenvironment (TIME)
Quercetin
Immunometabolism
Substitution of D-Arginine at Position 11 of & alpha;-RgIA Potently Inhibits & alpha;7 Nicotinic Acetylcholine Receptor
期刊论文
OAI收割
MARINE DRUGS, 2023, 卷号: 21, 期号: 6, 页码: 13
作者:
Wu, Yong
;
Zhang, Junjie
;
Ren, Jie
;
Zhu, Xiaopeng
;
Li, Rui
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
conotoxin
peptide synthesis
CD structure
electrophysiology
nicotinic acetylcholine receptors
Identification and characterization of the key lethal toxin from jellyfish Cyanea nozakii
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2023, 卷号: 230, 页码: 8
作者:
Li, Rongfeng
;
Yu, Huahua
;
Li, Aoyu
;
Yu, Chunlin
;
Li, Pengcheng
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2023/12/13
Jellyfish
Venom
Toxin
Letoxcn
Cyanea nozakii
Nongenomic effects and mechanistic study of butyl benzyl phthalate-induced thyroid disruption: Based on integrated in vitro, in silico assays and proteome analysis
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2022, 卷号: 836, 期号: 0, 页码: 155715
作者:
Li, Jian
;
Xu, Ying
;
Jiang, Yuhao
;
Li, Na
;
Li, Zhanjie
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2022/11/09
HORMONE
CELLS
RECEPTOR
ALPHA(V)BETA(3)
PROLIFERATION
ACTIVATION
TOXICITY
EXPOSURE
GROWTH
ESTERS
Brain-targeting biomimetic nanoparticles for codelivery of celastrol and LY2157299 for reversing glioma immunosuppression
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF PHARMACEUTICS, 2022, 卷号: 619, 页码: 11
作者:
Zhu, Siqi
;
Sun, Feifei
;
Zhao, Pengfei
;
Liang, Gang
;
Sun, Xiaoyi
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/08/16
Glioblastoma
Tumor-associated macrophages
Brain-targeted delivery
Celastrol
Albumin nanoparticles
Structure-Based Discovery of MDM2/4 Dual Inhibitors that Exert Antitumor Activities against MDM4-Overexpressing Cancer Cells
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 65, 期号: 8, 页码: 6207-6230
作者:
Zhang, Shiyan
;
Yan, Ziqin
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/08/16
Characterization of a small-molecule inhibitor targeting NEMO/IKK beta to suppress colorectal cancer growth
期刊论文
OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 13
作者:
Yu, Zhenlong
;
Gao, Jian
;
Zhang, Xiaolei
;
Peng, Yulin
;
Wei, Wenlong
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/06/15
Transcytosis mechanisms of cell-penetrating peptides: Cation-independent CC12 and cationic penetratin
期刊论文
OAI收割
JOURNAL OF PEPTIDE SCIENCE, 2022, 页码: 9
作者:
Zhu, Minjiao
;
Liu, Haiyang
;
Cao, Wenjiao
;
Fang, Yuefei
;
Chen, Zheng
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2022/06/15
cell-penetrating peptides
direct translocation pathway
drug delivery
endocytic pathway
penetration
transcytosis
cell internalization mechanism