中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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上海药物研究所 [25]
上海生物化学与细胞生... [6]
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期刊论文 [43]
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DRAK2 suppresses autophagy by phosphorylating ULK1 at Ser
56
to diminish pancreatic β cell function upon overnutrition
期刊论文
OAI收割
SCIENCE TRANSLATIONAL MEDICINE, 2024, 卷号: 16, 期号: 733, 页码: 16
作者:
Lu, Yuting
;
Xu, Junyu
;
Li, Yufeng
;
Wang, Ruoran
;
Dai, Chengqiu
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/03/13
Luteolin Protects Pancreatic beta Cells against Apoptosis through Regulation of Autophagy and ROS Clearance
期刊论文
OAI收割
PHARMACEUTICALS, 2023, 卷号: 16, 期号: 7, 页码: 17
作者:
Han, Ming
;
Lu, Yuting
;
Tao, Yunhua
;
Zhang, Xinwen
;
Dai, Chengqiu
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/10/17
luteolin
type 2 diabetes
beta cell
autophagy
reactive oxygen species
Enantiomeric pairs of macrocyclic acylphloroglucinols from Syzygium szemaoense
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 132, 页码: 6
作者:
Huang, Jin-Chang
;
Hong Xu, Hong-
;
Shi, Qing
;
Lei, Chun
;
Li, Jing-Ya
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2023/04/10
Syzygium szemaoense
Acylphloroglucinol enantiomers
Death -associated protein kinase-related
apoptosis inducing protein kinase 2
ATP citrate lyase
Combined inhibition of PARP and ATR synergistically potentiates the antitumor activity of HER2-targeting antibody-drug conjugate in HER2-positive cancers
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2023, 卷号: 13, 期号: 1, 页码: 161-+
作者:
Li, Yongpeng
;
Li, Lin
;
Fu, Haoyu
;
Yao, Qing
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Antibody-drug conjugate
DS-8201
PARP
ATR
synergy
DNA damage
N-degron-mediated degradation of the proteolytically activated form of PKC-theta kinase attenuates its pro-apoptotic function
期刊论文
OAI收割
CELLULAR SIGNALLING, 2023, 卷号: 110
作者:
Eldeeb, Mohamed A.
;
Zhou, Wenbin
;
Esmaili, Mansoore
;
Elgohary, Alaa M.
;
Wei, Hai
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2023/12/01
ASK120067 potently suppresses B-cell or T-cell malignancies in vitro and in vivo by inhibiting BTK and ITK
期刊论文
OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13, 页码: 9
作者:
Song, Peiran
;
Bai, Gang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2023/04/10
Bruton's tyrosine kinase
interleukin-2-inducible T cell kinase
ASK120067
B-cell lymphoma
T-cell leukemia
Design, synthesis, and biological evaluation of Wee1 kinase degraders
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 21
作者:
Zhu, Shulei
;
Liu, Jieyu
;
Xiao, Donghuai
;
Wang, Peipei
;
Ma, Jingkun
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2022/11/11
CRBN
Wee1
PROTAC
Degradation
DRAK2 aggravates nonalcoholic fatty liver disease progression through SRSF6-associated RNA alternative splicing
期刊论文
OAI收割
CELL METABOLISM, 2021, 卷号: 33, 期号: 10, 页码: 2004-+
作者:
Li, Yufeng
;
Xu, Junyu
;
Lu, Yuting
;
Bian, Hua
;
Yang, Lin
  |  
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2022/01/18
SYNTHESIS, CHARACTERIZATION, AND DRAK2 INHIBITORY ACTIVITIES OF HYDROXYAURONEDERIVATIVESURONE DERIVATIVES
期刊论文
OAI收割
HETEROCYCLES, 2021, 卷号: 102, 期号: 8, 页码: 1536-1551
作者:
Zhao, Mingsheng
;
Dai, Chengqiu
;
Li, Yi
;
Liu, Yinan
;
Li, Jing-Ya
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/01/04
SYNTHESIS, CHARACTERIZATION, AND DRAK2 INHIBITORY ACTIVITIES OF HYDROXYAURONEDERIVATIVESURONE DERIVATIVES
期刊论文
OAI收割
HETEROCYCLES, 2021, 卷号: 102, 期号: 8, 页码: 1536-1551
作者:
Zhao, MS (Zhao, Mingsheng) 1 , 2
;
Dai, CQ (Dai, Chengqiu) 3 , 4
;
Li, Y (Li, Yi) 1 , 2
;
Liu, YN (Liu, Yinan) 3
;
Li, JY (Li, Jing-Ya) 3
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/12/06