中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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Gold-catalyzed
endo
-selective Ring-opening of Epoxides and its Application in Construction of Poly-ethers
期刊论文
OAI收割
CHEMISTRY-A EUROPEAN JOURNAL, 2024, 页码: 10
作者:
Wu, Kehuan
;
Kang, Kaiwen
;
Liu, Dan
;
Zhang, Chiyue
;
Wang, Xinyu
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/25
6-endo ring-opening of epoxide
Baldwin's rules
gold-catalyzed reactions
marine ladder-like poly-ethers
Nakanishi hypothesis
Meta-MolNet: A Cross-Domain Benchmark for Few Examples Drug Discovery
期刊论文
OAI收割
IEEE TRANSACTIONS ON NEURAL NETWORKS AND LEARNING SYSTEMS, 2024, 页码: 15
作者:
Lv, Qiujie
;
Chen, Guanxing
;
Yang, Ziduo
;
Zhong, Weihe
;
Chen, Calvin Yu-Chian
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2024/04/09
Benchmark platform
cross-domain meta-learning
drug discovery
few examples
Meta-MolNet
molecular property
Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:
Yan, Xue
;
Zhang, Chun
;
Gao, Li-Xin
;
Liu, Min -Min
;
Yang, Yu-Ting
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/02/27
Imidazo[124] triazole derivatives
Fluorescence property
SHP1
Bioactivity
Cellular imaging
Enzymatic Synthesis of Noncanonical α-Amino Acids Containing γ-Tertiary Alcohols
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2024, 页码: 9
作者:
Zhang, Rui
;
Zhang, Chenghua
;
Tan, Jiamu
;
He, Yifan
;
Zhuo, Dan
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/02/27
Asymmetric Synthesis
Biocatalysis
Noncanonical Amino Acids
Quantum Chemical Calculations
Tertiary Alcohols
D3Rings: A Fast and Accurate Method for Ring System Identification and Deep Generation of Drug-Like Cyclic Compounds
期刊论文
OAI收割
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2024, 卷号: 64, 期号: 3, 页码: 724-736
作者:
Ma, Minfei
;
Zhang, Xinben
;
Zhou, Liping
;
Han, Zijian
;
Shi, Yulong
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/03/13
Discovery of hematopoietic progenitor kinase 1 inhibitors using machine learning-based screening and free energy perturbation
期刊论文
OAI收割
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS, 2024, 页码: 13
作者:
Feng, Dazhi
;
Liu, Bo
;
Chen, Zhiwei
;
Xu, Jinyi
;
Geng, Meiyu
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/02/27
HPK1 inhibitor
machine learning
virtual screening
free energy perturbation
structural modification
Substrate- and Catalyst-Controlled C-H Bond Activation/Annulation for Construction of Pyrido[2,3,4-
de
]quinazolinones and Indolo[1,2-
c
]quinazolinones
期刊论文
OAI收割
ADVANCED SYNTHESIS & CATALYSIS, 2023, 页码: 8
作者:
Hou, Xinjiao
;
Wang, Run
;
Zhou, Jianhui
;
Li, Yuan
;
Li, Jiyuan
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2024/01/16
C-H bond activation
Fused heterocycles
Rh(III) catalysis
Ru(II) catalysis
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study
期刊论文
OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:
Zhao, Tian-Tian
;
Hu, Hao-Jie
;
Gao, Li-Xin
;
Zhou, Yu-Bo
;
Zhu, Yun-Long
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Protein tyrosine phosphatases inhibitors
PTP1B inhibitors
Mechanism study
Molecular dynamics
Selective activator of human ClpP triggers cell cycle arrest to inhibit lung squamous cell carcinoma
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 7069
作者:
Zhou, Lin-Lin
;
Zhang, Tao
;
Xue, Yun
;
Yue, Chuan
;
Pan, Yihui
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/03/27
Isolation and characterization of glutathione S-transferase genes and their transcripts in
Saccharina japonica
(Laminariales, Phaeophyceae) during development and under abiotic stress
期刊论文
OAI收割
BMC PLANT BIOLOGY, 2023, 卷号: 23, 期号: 1, 页码: 19
作者:
Lu, Chang
;
Zhang, Pengyan
;
Li, Shuang
;
Cheng, Mengzhen
;
Duan, Delin
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/11/30
Saccharina japonica
Glutathione S-transferase
Transcriptome
Gene expression
Abiotic stresses
Enzyme activity assay