中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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浏览/检索结果: 共173条,第1-10条 帮助

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New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 9
作者:  
Zheng, Yingying;  Lu, Li;  Li, Mengyue;  Xu, Dehua;  Zhang, Laishun
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/01/26
Exploring the mechanism of the PTP1B inhibitors by molecular dynamics and experimental study 期刊论文  OAI收割
JOURNAL OF MOLECULAR GRAPHICS & MODELLING, 2023, 卷号: 125, 页码: 12
作者:  
  |  收藏  |  浏览/下载:11/0  |  提交时间:2023/10/17
Novel thieno[2,3-b]quinoline-procaine hybrid molecules: A new class of allosteric SHP-1 activators evolved from PTP1B inhibitors 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2023, 卷号: 34, 期号: 8, 页码: 6
作者:  
Xu, Lei;  Xuyan, Xuyang;  Minmi, Minmin;  Wang, Zhiji;  Shee, Chao
  |  收藏  |  浏览/下载:27/0  |  提交时间:2023/10/17
URSOLIC ACID DERIVATIVES BEARING 1,2,3-TRIAZOLE MOIETIES AS POTENTIAL PTP1B INHIBITORS 期刊论文  OAI收割
CHEMISTRY OF NATURAL COMPOUNDS, 2023, 卷号: 59, 期号: 3, 页码: 508-511
作者:  
Liu, Zhe;  Bai, Xueqian;  Sheng, Li;  Sun, Liangpeng;  Li, Jia
  |  收藏  |  浏览/下载:35/0  |  提交时间:2023/10/17
Root-Extracted lignanamides from Limonium gmelinii (Willd.) Kuntze with a potential PTP1B inhibitory activity by regulating PI3K/AKT signaling pathway 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 132, 页码: 9
作者:  
Tuohongerbieke, Amanguli;  Liu, Liu;  Li, Jun;  Xin, Xuelei;  Aisa, Haji Akber
  |  收藏  |  浏览/下载:8/0  |  提交时间:2023/10/17
Phytochemical and biological studies on rare and endangered plants endemic to China. Part XXV. Structurally diverse triterpenoids and diterpenoids from two endangered Pinaceae plants endemic to the Chinese Qinling Mountains and their bioactivities 期刊论文  OAI收割
PHYTOCHEMISTRY, 2022, 卷号: 203, 页码: 14
作者:  
Jiang, Wei;  Zhao, Ze-Yu;  Tong, Ying-Peng;  Ma, Guang-Lei;  Zang, Yi
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/09/30
Macrocephatriolides A and B: Two Guaianolide Trimers from Ainsliaea macrocephala as PTP1B Inhibitors and Insulin Sensitizers 期刊论文  OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 86, 期号: 24, 页码: 17782-17789
作者:  
Ren, Yong-Mei;  Zhang, Rui;  Feng, Zheling;  Ke, Chang-Qiang;  Yao, Sheng
  |  收藏  |  浏览/下载:25/0  |  提交时间:2022/06/15
Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13
作者:  
Meng, Xiang-Dong;  Gao, Li-Xin;  Wang, Zhi-Jia;  Feng, Bo;  Zhang, Chun
  |  收藏  |  浏览/下载:61/0  |  提交时间:2021/12/01
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel N-Acylhydrazone Derivatives Containing Carbazole and Aromatic Ring/Aromatic Fused Heterocycle 期刊论文  OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 9, 页码: 3593-3607
作者:  
Li Yingjun;  Lin Ledi;  Liu Jihong;  Gao Lixin;  Sheng Li
  |  收藏  |  浏览/下载:43/0  |  提交时间:2021/12/01
Rearranged Diels-Alder Adducts and Prenylated Flavonoids as Potential PTP1B Inhibitors from Morus nigra 期刊论文  OAI收割
JOURNAL OF NATURAL PRODUCTS, 2021, 卷号: 84, 期号: 8, 页码: 2303-2311
作者:  
Qu, Ke-Jun;  Wang, Bin;  Jiang, Chang-Sheng;  Xie, Bao-Gang;  Liu, Ai-Hong
  |  收藏  |  浏览/下载:29/0  |  提交时间:2021/11/04