中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2022 [23]
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Design and synthesis of chromone-nitrogen mustard derivatives and evaluation of anti-breast cancer activity 期刊论文  OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 431-444
作者:  
Sun, Jianan;  Mu, Jiahui;  Wang, Shenglin;  Jia, Cai;  Li, Dahong
  |  收藏  |  浏览/下载:33/0  |  提交时间:2022/06/15
Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Bi, Kaijian;  Cheng, Junfei;  He, Shipeng;  Fang, Yuxin;  Huang, Min
  |  收藏  |  浏览/下载:16/0  |  提交时间:2023/04/10
Design, synthesis, and biological evaluation of Wee1 kinase degraders 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 243, 页码: 21
作者:  
Zhu, Shulei;  Liu, Jieyu;  Xiao, Donghuai;  Wang, Peipei;  Ma, Jingkun
  |  收藏  |  浏览/下载:34/0  |  提交时间:2022/11/11
Cyclopiumolides A and B, unusual 13-membered macrolides from the deep sea-sourced fungus Penicillium cyclopium SD-413 with antiproliferative activities 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2022, 卷号: 128, 页码: 7
作者:  
Li, Yan-He;  Yang, Sui-Qun;  Li, Xiao-Ming;  Li, Xin;  Wang, Bin-Gui
  |  收藏  |  浏览/下载:22/0  |  提交时间:2023/01/06
SOMCL-19-133, a novel, selective, and orally available inhibitor of NEDD8-activating enzyme (NAE) for cancer therapy 期刊论文  OAI收割
NEOPLASIA, 2022, 卷号: 32, 页码: 12
作者:  
Zhou, Li-Na;  Xiong, Chaodong;  Cheng, Yong-Jun;  Song, Shan-Shan;  Bao, Xu-Bin
  |  收藏  |  浏览/下载:14/0  |  提交时间:2023/04/10
Design, Synthesis, and Biological Evaluation of Androgen Receptor Degrading and Antagonizing Bifunctional Steroidal Analogs for the Treatment of Advanced Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 22
作者:  
Wang, Ao;  Luo, Xianggang;  Wang, Yawan;  Meng, Xin;  Lu, Zhengyu
  |  收藏  |  浏览/下载:30/0  |  提交时间:2022/11/11
Synthesis of Hydantoin Androgen Receptor Antagonists and Study on Their Antagonistic Activity 期刊论文  OAI收割
MOLECULES, 2022, 卷号: 27, 期号: 18, 页码: 22
作者:  
Ma, Longjun;  Zhou, Yan;  Yang, Dehua;  Wang, Ming-Wei;  Lu, Wei
  |  收藏  |  浏览/下载:13/0  |  提交时间:2022/11/11
Integrating UPLC-HR-MS/MS, Network Pharmacology, and Experimental Validation to Uncover the Mechanisms of Jin?gan Capsules against Breast Cancer br 期刊论文  OAI收割
ACS OMEGA, 2022, 卷号: 7, 期号: 32, 页码: 28003-28015
作者:  
Qiu, Jianfei;  Zhang, Zhiyin;  Hu, Anling;  Zhao, Peng;  Wei, Xuenai
  |  收藏  |  浏览/下载:21/0  |  提交时间:2022/09/30
Sheep tail fat inhibits the proliferation of non-small-cell lung cancer cells in vitro and in vivo 期刊论文  OAI收割
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13
作者:  
Xu, Changzhi;  Zhang, Lanlan;  He, Huimin;  Liu, Xiaoyi;  Pei, Xinxin
  |  收藏  |  浏览/下载:26/0  |  提交时间:2022/12/23
Integrating UPLC-HR-MS/MS, Network Pharmacology, and Experimental Validation to Uncover the Mechanisms of Jin'gan Capsules against Breast Cancer 期刊论文  OAI收割
ACS OMEGA, 2022, 页码: 13
作者:  
Qiu, Jianfei;  Zhang, Zhiyin;  Hu, Anling;  Zhao, Peng;  Wei, Xuenai
  |  收藏  |  浏览/下载:23/0  |  提交时间:2022/09/30