中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2022 [154]
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Design, synthesis, and biological evaluation of novel carbazole derivatives as potent DNMT1 inhibitors with reasonable PK properties 期刊论文  OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1537-1555
作者:  
Li, Ennian;  Wang, Kai;  Zhang, Bei;  Guo, Siqi;  Xiao, Senhao
  |  收藏  |  浏览/下载:37/0  |  提交时间:2022/08/16
Identification of 1H-pyrazolo[3,4-b]pyridine derivatives as novel and potent TBK1 inhibitors: design, synthesis, biological evaluation, and molecular docking study 期刊论文  OAI收割
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 卷号: 37, 期号: 1, 页码: 1411-1425
作者:  
Sun, Yin;  Tang, Haotian;  Wang, Xiaoyan;  Feng, Fang;  Fan, Tiantian
  |  收藏  |  浏览/下载:36/0  |  提交时间:2022/08/16
PD-L1 Aptamer-Functionalized Metal-Organic Framework Nanoparticles for Robust Photo-Immunotherapy against Cancer with Enhanced Safety 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2022, 页码: 9
作者:  
Zhang, Jingfang;  Li, Wenzhe;  Qi, Yafei;  Wang, Guorong;  Li, Lele
  |  收藏  |  浏览/下载:12/0  |  提交时间:2023/02/22
Learning with uncertainty to accelerate the discovery of histone lysine-specific demethylase 1A (KDM1A/LSD1) inhibitors 期刊论文  OAI收割
BRIEFINGS IN BIOINFORMATICS, 2022, 页码: 14
作者:  
Wang, Dong;  Wu, Zhenxing;  Shen, Chao;  Bao, Lingjie;  Luo, Hao
  |  收藏  |  浏览/下载:26/0  |  提交时间:2023/04/10
Discovery of Highly Potent Nicotinamide Phosphoribosyltransferase Degraders for Efficient Treatment of Ovarian Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Bi, Kaijian;  Cheng, Junfei;  He, Shipeng;  Fang, Yuxin;  Huang, Min
  |  收藏  |  浏览/下载:16/0  |  提交时间:2023/04/10
A novel coating with SiO2 anchored on MXene loading tannic acid for self-healing anticorrosive performance 期刊论文  OAI收割
JOURNAL OF ALLOYS AND COMPOUNDS, 2022, 卷号: 928, 页码: 10
作者:  
Sun, Xiaoguang;  Ma, Chengcheng;  Ma, Fubin;  Wang, Tong;  Feng, Chao
  |  收藏  |  浏览/下载:32/0  |  提交时间:2023/01/06
Discovery of 10H-Benzo[b]pyrido[2,3-e][1,4]oxazine AXL Inhibitors via Structure-Based Drug Design Targeting c-Met Kinase 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 15
作者:  
Zhan, Zhengsheng;  Ji, Yinchun;  Su, Haixia;  Fang, Chen;  Peng, Xia
  |  收藏  |  浏览/下载:30/0  |  提交时间:2023/04/10
Dual inhibition of CHK1/FLT3 enhances cytotoxicity and overcomes adaptive and acquired resistance in FLT3-ITD acute myeloid leukemia 期刊论文  OAI收割
LEUKEMIA, 2022, 页码: 11
作者:  
Jiang, Kailong;  Li, Xuemei;  Wang, Chang;  Hu, Xiaobei;  Wang, Peipei
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/04/10
Targeting the PI3K/AKT/mTOR Signaling Pathway in the Treatment of Human Diseases: Current Status, Trends, and Solutions 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 29
作者:  
Huang, Jindi;  Chen, Liye;  Wu, Jiangxia;  Ai, Daiqiao;  Zhang, Ji-Quan
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/04/10
Identification of a class of potent USP25/28 inhibitors with broad-spectrum anti-cancer activity 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2022, 卷号: 7, 期号: 1, 页码: 3
作者:  
Peng, Jin;  Jiang, Kun;  Sun, Xiao;  Wu, Lingzhi;  Wang, Jiewei
  |  收藏  |  浏览/下载:19/0  |  提交时间:2023/04/10