中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [787]
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Rational design and discovery of novel oxalate-like derivatives as aphid-repellent candidates based on odorant-binding protein 3 期刊论文  OAI收割
JOURNAL OF MOLECULAR STRUCTURE, 2024, 卷号: 1301, 页码: 11
作者:  
Zhu, Ziwei;  Li, Jianing;  Liu, Chong;  Li, Huilin;  Lu, Xingxing
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/04/09
Probing the dynamic thermodynamic resolution and biological activity of Cu(II) and Pd(II) complexes with Schiff base ligand derived from proline 期刊论文  OAI收割
CHINESE CHEMICAL LETTERS, 2024, 卷号: 35, 期号: 4, 页码: 7
作者:  
Yu, Tao;  Soloshonok, Vadim A.;  Xiao, Zhekai;  Liu, Hong;  Wang, Jiang
  |  收藏  |  浏览/下载:11/0  |  提交时间:2024/04/09
Structure-Activity Relationships of 2-(Arylthio)benzoic Acid FTO Inhibitors 期刊论文  OAI收割
ISRAEL JOURNAL OF CHEMISTRY, 2024, 页码: 13
作者:  
Yan, Chao;  Zhang, Qian;  Xiao, Pan;  Xie, Xinyun;  Li, Ming
  |  收藏  |  浏览/下载:28/0  |  提交时间:2024/03/25
Novel imidazo[1,2,4] triazole derivatives: Synthesis, fluorescence, bioactivity for SHP1 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 265, 页码: 15
作者:  
Yan, Xue;  Zhang, Chun;  Gao, Li-Xin;  Liu, Min -Min;  Yang, Yu-Ting
  |  收藏  |  浏览/下载:9/0  |  提交时间:2024/02/27
New chromone derivatives bearing thiazolidine-2,4-dione moiety as potent PTP1B inhibitors: Synthesis and biological activity evaluation 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2024, 卷号: 143, 页码: 9
作者:  
Zheng, Yingying;  Lu, Li
  |  收藏  |  浏览/下载:8/0  |  提交时间:2024/01/26
Design, synthesis and biological evaluation of betulinic acid derivatives as potential inhibitors of 3CL-protease of SARS-CoV-2 期刊论文  OAI收割
STEROIDS, 2024, 卷号: 202, 页码: 8
作者:  
Liu, Yaowen;  Nie, Tianqing;  Hou, Jinjun;  Long, Huali;  Zhang, Zijia
  |  收藏  |  浏览/下载:14/0  |  提交时间:2024/03/13
Koilodenoids A-G, immunosuppressive spiro dimers of diterpenoids from Koilodepas hainanense: structural elucidation and biomimetic transformation 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2024, 页码: 8
作者:  
Ren, Yu;  Zheng, Cheng-Yu;  Yao, Jia-Ying;  He, Shi-Jun;  Fan, Yao-Yue
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/03/06
Synthesis and Biological Evaluation of β-Lactam Derivatives Targeting Speckle-Type POZ Protein (SPOP) 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 15, 期号: 2, 页码: 270-279
作者:  
Zhou, Chenmao;  Hao, Xinyue;  Chen, Zhengyang;  Zhang, Runze;  Zhou, Qian
  |  收藏  |  浏览/下载:19/0  |  提交时间:2024/03/13
Design, Synthesis, and Biological Evaluation of Potent and Selective PROTAC Degraders of Oncogenic KRASG12D 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 2, 页码: 1147-1167
作者:  
Zhou, Chuan;  Fan, Zisheng;  Gu, Yuejiao;  Ge, Zhiming;  Tao, Zhaofan
  |  收藏  |  浏览/下载:10/0  |  提交时间:2024/02/27
Discovery and optimization of thieno[3,2-d]pyrimidine derivatives as highly selective inhibitors of cyclin-dependent kinase 7 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 263, 页码: 21
作者:  
Zhang, Hongjin;  Lin, Guohao;  Jia, Suyun;  Zhang, Ying;  Wu, Jianbo
  |  收藏  |  浏览/下载:5/0  |  提交时间:2024/01/26