中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [10]
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Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:  
Lei, E.;  Tao, Huanyu;  Jiao, Shang;  Yang, Anming;  Zhou, Yu
  |  收藏  |  浏览/下载:26/0  |  提交时间:2022/08/16
Impurity Identification and Scale-Up of a Novel Glycopeptide Antibiotic 期刊论文  OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2390-2402
作者:  
Jiao, Shang;  Guan, Dongliang;  Xu, Lili;  Liu, Bo;  Shi, Weiwei
  |  收藏  |  浏览/下载:22/0  |  提交时间:2022/01/18
An integrative drug repositioning framework discovered a potential therapeutic agent targeting COVID-19 期刊论文  OAI收割
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 16
作者:  
Ge, Yiyue;  Tian, Tingzhong;  Huang, Suling;  Wan, Fangping;  Li, Jingxin
  |  收藏  |  浏览/下载:28/0  |  提交时间:2022/06/15
Biomimetic metal-organic nanoparticles prepared with a 3D-printed microfluidic device as a novel formulation for disulfiram-based therapy against breast cancer 期刊论文  OAI收割
APPLIED MATERIALS TODAY, 2020, 卷号: 18, 页码: 12
作者:  
Chang, Ya;  Jiang, Jizong;  Chen, Wu;  Yang, Wen;  Chen, Lili
  |  收藏  |  浏览/下载:32/0  |  提交时间:2020/07/01
DZ2002 ameliorates fibrosis, inflammation, and vasculopathy in experimental systemic sclerosis models 期刊论文  OAI收割
ARTHRITIS RESEARCH & THERAPY, 2019, 卷号: 21, 期号: 1, 页码: 15
作者:  
Zhang, Zongwang;  Wu, Yanwei;  Wu, Bing;  Qi, Qing;  Li, Heng
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Interplay between the bacterial protein deacetylase CobB and the second messenger c-di-GMP 期刊论文  OAI收割
EMBO JOURNAL, 2019, 页码: 18
作者:  
Xu, Zhaowei;  Zhang, Hainan;  Zhang, Xingrun;  Jiang, Hewei;  Liu, Chengxi
  |  收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
Discovery of Potent and Noncovalent Reversible EGFR Kinase Inhibitors of EGFR(L858R/T790M/C797S) 期刊论文  OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 10, 期号: 6, 页码: 869-873
作者:  
Li, Qiannan;  Zhang, Tao;  Li, Shiliang;  Tong, Linjiang;  Li, Junyu
  |  收藏  |  浏览/下载:58/0  |  提交时间:2020/07/01
EGFR  mutant  inhibitor  C797S  
Design, Synthesis, and Biological Evaluation of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 13, 页码: 5609-5622
作者:  
Hao, Yongjia;  Lyu, Jiankun;  Qu, Rong;  Tong, Yi;  Sun, Deheng
  |  收藏  |  浏览/下载:61/0  |  提交时间:2019/01/08
Design, Synthesis, and Interaction Study of Quinazoline-2(1H)-thione Derivatives as Novel Potential Bcl-x(L) Inhibitors 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2010, 卷号: 53, 期号: 9, 页码: 3465-3479
作者:  
Feng, Yu;  Ding, Xiao;  Chen, Tao;  Chen, Lili;  Liu, Fang
  |  收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
4-(Phenylsulfonamidomethyl) benzamides as potent and selective inhibitors of the 11 beta-hydroxysteroid dehydrogenase type 1 with efficacy in diabetic ob/ob mice 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 卷号: 19, 期号: 15, 页码: 4455-4458
作者:  
Zhang, Xu;  Zhou, Zhou;  Yang, Huaiyu;  Chen, Junhua;  Feng, Ying
  |  收藏  |  浏览/下载:9/0  |  提交时间:2019/01/08