中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [184]
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OAI收割 [184]
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期刊论文 [176]
会议论文 [8]
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2023 [14]
2022 [9]
2021 [9]
2020 [13]
2019 [12]
2018 [9]
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专题:上海药物研究所
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Total synthesis of (±)-villosin C and (±)-teuvincenone B
期刊论文
OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2023, 页码: 5
作者:
Zhou, Jin-Xin
;
Yan, Ming-Jie
;
Shi, Xiao-Yu
;
Wang, Yue-Qi
;
Shen, Hong-Yan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2024/01/16
Circuit-specific gene therapy reverses core symptoms in a primate Parkinson's disease model
期刊论文
OAI收割
CELL, 2023, 卷号: 186, 期号: 24, 页码: 5394-+
作者:
Chen, Yefei
;
Hong, Zexuan
;
Wang, Jingyi
;
Liu, Kunlin
;
Liu, Jing
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/01/26
Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 19
作者:
Wang, Pingyuan
;
Zhu, Wen-Ting
;
Wang, Yajing
;
Song, Shan-Shan
;
Xi, Yong
  |  
收藏
  |  
浏览/下载:58/0
  |  
提交时间:2023/10/17
PARP1 inhibitor
Synthetic lethality
Drug resistance
Anticancer
Structure -activity relationship
Discovery of zolinium TSG1180 as a novel agonist of transgelin-2 for treating asthma
期刊论文
OAI收割
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2023, 卷号: 167, 页码: 115556
作者:
Yuan, Hong-Kai
;
Li, Bo
;
Wu, Leyun
;
Wang, Xue-Ling
;
Lv, Zhi-Ying
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/03/26
Active learning
Consensus labelling
Eye irritation
Serious eye damage
Structural alerts
LINC00955 suppresses colorectal cancer growth by acting as a molecular scaffold of TRIM25 and Sp1 to Inhibit DNMT3B-mediated methylation of the PHIP promoter
期刊论文
OAI收割
BMC CANCER, 2023, 卷号: 23, 期号: 1, 页码: 20
作者:
Ren, Ganglin
;
Li, Hongyan
;
Hong, Dan
;
Hu, Fangyu
;
Jin, Rongjia
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2023/12/08
LINC00955
Colorectal cancer
Cell cycle
CDK2
PHIP
Sp1
Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:
Wen, Xin
;
Zhang, Minmin
;
Duan, Zhiqiang
;
Suo, Yanrui
;
Lu, Weiwei
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2023/10/17
Highly Modified Sesquiterpene Lactones with Cytotoxic Activities from Strobocalyx chunii
期刊论文
OAI收割
JOURNAL OF ORGANIC CHEMISTRY, 2023, 卷号: 88, 期号: 15, 页码: 11122-11129
作者:
Ge, Zhan-Peng
;
Gao, Yuan
;
Zhang, Yan
;
Liu, Hong-Chun
;
Zhao, Jin-Xin
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/10/17
Triterpenoids with multi-skeletons as 11 beta-HSD1 inhibitors from Euphorbia sikkimensis
期刊论文
OAI收割
PHYTOCHEMISTRY, 2023, 卷号: 211, 页码: 12
作者:
Fang, Chu-Hong
;
Li, Yu-Peng
;
Li, Ying
;
Yue, Jian-Min
;
Bao, Jie
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2023/10/17
Euphorbia sikkimensis family
Triterpenoids
11fl-HSD1 inhibitors
Molecular docking
Metabolic abnormalities
Effect of an Herbal-Based Injection on 28-Day Mortality in Patients With Sepsis The EXIT-SEP Randomized Clinical Trial
期刊论文
OAI收割
JAMA INTERNAL MEDICINE, 2023, 卷号: 183, 期号: 7, 页码: 647-655
作者:
Liu, Songqiao
;
Yao, Chen
;
Xie, Jianfeng
;
Liu, Hong
;
Wang, Hongliang
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/03/27