中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 上海药物研究所 [100]
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Pharmacological inhibition of Kir4.1 evokes rapid-onset antidepressant responses 期刊论文  OAI收割
NATURE CHEMICAL BIOLOGY, 2024, 页码: 29
作者:  
Zhou, Xiaoyu;  Zhao, Cheng;  Xu, Haiyan;  Xu, Yixiang;  Zhan, Li
  |  收藏  |  浏览/下载:13/0  |  提交时间:2024/03/25
Discovery of a novel GPR35 agonist with high and equipotent species potency for oral treatment of IBD 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2023, 卷号: 96, 页码: 12
作者:  
Song, Zhaoxiang;  Lu, Dan;  Sun, Jun;  Ye, Yangliang;  Fang, Jiahui
  |  收藏  |  浏览/下载:26/0  |  提交时间:2024/01/16
GPR35  IBD  Lodoxamide  
ABPP-CoDEL: Activity-Based Proteome Profiling-Guided Discovery of Tyrosine-Targeting Covalent Inhibitors from DNA-Encoded Libraries 期刊论文  OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2023, 卷号: 145, 期号: 46, 页码: 25283-25292
作者:  
Jiang, Lulu;  Liu, Sixiu;  Jia, Xinglong;  Gong, Qinting;  Wen, Xin
  |  收藏  |  浏览/下载:24/0  |  提交时间:2024/01/16
Discovery of ARD-1676 as a Highly Potent and Orally Efficacious AR PROTAC Degrader with a Broad Activity against AR Mutants for the Treatment of AR plus Human Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 18, 页码: 13280-13303
作者:  
Xiang, Weiguo;  Zhao, Lijie;  Han, Xin;  Xu, Tianfeng;  Kregel, Steven
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/12/08
Ligand recognition and G protein coupling of the human itch receptor MRGPRX1 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2023, 卷号: 14, 期号: 1, 页码: 12
作者:  
Guo, Lulu;  Zhang, Yumu;  Fang, Guoxing;  Tie, Lu;  Zhuang, Yuming
  |  收藏  |  浏览/下载:20/0  |  提交时间:2024/01/16
Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1H)-one Focused DNA-Encoded Library 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 页码: 15
作者:  
Wen, Xin;  Zhang, Minmin;  Duan, Zhiqiang;  Suo, Yanrui;  Lu, Weiwei
  |  收藏  |  浏览/下载:30/0  |  提交时间:2023/10/17
GPR84 regulates pulmonary inflammation by modulating neutrophil functions 期刊论文  OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 卷号: 44, 期号: 8, 页码: 1665-1675
作者:  
Wang, Si-wei;  Zhang, Qing;  Lu, Dan;  Fang, You-chen;  Yan, Xiao-ci
  |  收藏  |  浏览/下载:3/0  |  提交时间:2024/03/27
Discovery of a Novel Bifunctional Steroid Analog, YXG-158, as an Androgen Receptor Degrader and CYP17A1 Inhibitor for the Treatment of Enzalutamide-Resistant Prostate Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 66, 期号: 14, 页码: 9972-9991
作者:  
Wang, Ao;  Luo, Xianggang;  Meng, Xin;  Lu, Zhengyu;  Chen, Kaixian
  |  收藏  |  浏览/下载:9/0  |  提交时间:2023/10/17
Preparation and characterization of nanobodies targeting SARS-CoV-2 papain-like protease 期刊论文  OAI收割
PROTEIN EXPRESSION AND PURIFICATION, 2023, 卷号: 207, 页码: 106267
作者:  
Qiao, Huarui;  Li, Lingyun;  Wang, Lu;  Yu, Haijun;  Hu, Fangzheng
  |  收藏  |  浏览/下载:1/0  |  提交时间:2024/03/27
ETCM v2.0: An update with comprehensive resource and rich annotations for traditional Chinese medicine 期刊论文  OAI收割
ACTA PHARMACEUTICA SINICA B, 2023, 卷号: 13, 期号: 6, 页码: 2559-2571
作者:  
Zhang, Yanqiong;  Li, Xin;  Shi, Yulong;  Chen, Tong;  Xu, Zhijian
  |  收藏  |  浏览/下载:21/0  |  提交时间:2023/10/17