中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2019 [12]
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fDiscovery of pyrazole-thiophene derivatives as highly Potent, orally active Akt inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 180, 页码: 72-85
作者:  
Zhan, Wenhu;  Che, Jinxin;  Xu, Lei;  Wu, Yizhe;  Hu, Xiaobei
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
New linker structures applied in glycosite-specific antibody drug conjugates 期刊论文  OAI收割
ORGANIC CHEMISTRY FRONTIERS, 2019, 卷号: 6, 期号: 17, 页码: 3144-3149
作者:  
Faridoon;  Shi, Wei;  Qin, Ken;  Tang, Yubo;  Li, Mingjie
  |  收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01
Biofilm Nanofiber-Coated Separators for Dendrite-Free Lithium Metal Anode and Ultrahigh-Rate Lithium Batteries 期刊论文  OAI收割
ACS APPLIED MATERIALS & INTERFACES, 2019, 卷号: 11, 期号: 35, 页码: 32373
作者:  
Nie, Lu;  Li, Yingfeng;  Chen, Shaojie;  Li, Ke;  Huang, Yuanqi
  |  收藏  |  浏览/下载:78/0  |  提交时间:2019/12/26
Selective Late-Stage Oxygenation of Sulfides with Ground-State Oxygen by Uranyl Photocatalysis 期刊论文  OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2019, 页码: 9
作者:  
Li, Yiming;  Rizvi, S. Aal-e-Ali;  Hu, Deqing;  Sun, Danwen;  Gao, Anhui
  |  收藏  |  浏览/下载:14/0  |  提交时间:2020/07/01
Discovery of 3,4,6-Trisubstituted Piperidine Derivatives as Orally Active, Low hERG Blocking Akt Inhibitors via Conformational Restriction and Structure-Based Design 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 15, 页码: 7264-7288
作者:  
Dong, Xiaowu;  Zhan, Wenhu;  Zhao, Mengting;  Che, Jinxin;  Dai, Xiaoyang
  |  收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01
Discovery of (R)-5-((5-(1-methyl-1H-pyrazol-4-yl)-4-(methylamino) pyrimidin-2-yl)amino)-3-(piperidin-3-yloxy)picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 173, 页码: 44-62
作者:  
Tong, Lexian;  Song, Pinrao;  Jiang, Kailong;  Xu, Lei;  Jin, Tingting
  |  收藏  |  浏览/下载:24/0  |  提交时间:2020/07/01
Tranylcypromine and 6-trifluoroethyl thienopyrimidine hybrid as LSD1 inhibitor 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 844-847
作者:  
Wang, Xiaowen;  Su, Mingbo;  Li, You;  Liu, Tongchao;  Wang, Yujie
  |  收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01
Discovery of novel indoleaminopyrimidine NIK inhibitors based on molecular docking-based support vector regression (SVR) model 期刊论文  OAI收割
CHEMICAL PHYSICS LETTERS, 2019, 卷号: 718, 页码: 38-45
作者:  
Ye, Qing;  Li, Qiu;  Gao, Anhui;  Ying, Huazhou;  Cheng, Gang
  |  收藏  |  浏览/下载:10/0  |  提交时间:2020/07/01
Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors 期刊论文  OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 423-439
作者:  
Yu, Jianjun;  Liu, Jieyu;  Li, Daqiang;  Xu, Lei;  Hong, Duidui
  |  收藏  |  浏览/下载:20/0  |  提交时间:2020/07/01
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 4, 页码: 589-603
作者:  
Liu, Xiaoqi;  Hu, Yuanyuan;  Gao, Anhui;  Xu, Meng
  |  收藏  |  浏览/下载:21/0  |  提交时间:2020/07/01