中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [15]
植物研究所 [1]
采集方式
OAI收割 [16]
内容类型
期刊论文 [16]
发表日期
2020 [16]
学科主题
Agronomy [1]
Plant Scie... [1]
Soil Scien... [1]
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浏览/检索结果:
共16条,第1-10条
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发表日期:2020
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A Peptide Binder of E3 Ligase Adaptor SPOP Disrupts Oncogenic SPOP-Protein Interactions in Kidney Cancer Cells
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 274-280
作者:
Wang, Zhen
;
Zhang, Hao
;
Chen, Baoen
;
Ouyang, Sisheng
;
Zheng, Tong
  |  
收藏
  |  
浏览/下载:123/0
  |  
提交时间:2021/05/24
SPOP
Protein‐
protein interaction
Clear cell Renal Cell Carcinomas
Crystal structure
Peptide inhibitor
Structure-based drug optimization and biological evaluation of tetrahydroquinolin derivatives as selective and potent CBP bromodomain inhibitors
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 22, 页码: 7
作者:
Bi, Xiaoyang
;
Chen, Yu
;
Sun, Zhongya
;
Lu, Wenchao
;
Xu, Pan
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/05/24
Drug design
CBP
Bromodomain
Inhibitor
Acute myeloid leukemia
Structural basis for activation of the growth hormone-releasing hormone receptor
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:
Zhou, Fulai
;
Zhang, Huibing
;
Cong, Zhaotong
;
Zhao, Li-Hua
;
Zhou, Qingtong
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2020/12/21
Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 11
作者:
Chen, Yu
;
Bi, Xiaoyang
;
Zhang, Fengcai
;
Sun, Zhongya
;
Xu, Pan
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2020/12/24
In silico screening
Drug design
CBP
Bromodomain
Inhibitor
Acute Myeloblastic Leukemia
Discovery of novel USP8 inhibitors via Ubiquitin-Rho-110 fluorometric assay based high throughput screening
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 9
作者:
Han, Jie
;
Tian, Yucheng
;
Yu, Liang
;
Zhang, Qilin
;
Xu, Xi
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2020/12/24
Ubiquitination
High throughput screening
Drug discovery
USP8
Sorting Nexin 10 Mediates Metabolic Reprogramming of Macrophages in Atherosclerosis Through the Lyn-Dependent TFEB Signaling Pathway
期刊论文
OAI收割
CIRCULATION RESEARCH, 2020, 卷号: 127, 期号: 4, 页码: 534-549
作者:
You, Yan
;
Bao, Wei-Lian
;
Zhang, Su-Lin
;
Li, Hai-Dong
;
Li, Hui
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/12/24
atherosclerosis
foam cell
lipid metabolism
monocytes
sorting nexin
Structural basis for inhibition of the RNA-dependent RNA polymerase from SARS-CoV-2 by remdesivir
期刊论文
OAI收割
SCIENCE, 2020, 卷号: 368, 期号: 6498, 页码: 1499-+
作者:
Yin, Wanchao
;
Mao, Chunyou
;
Luan, Xiaodong
;
Shen, Dan-Dan
;
Shen, Qingya
  |  
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2020/12/24
Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease
期刊论文
OAI收割
SCIENCE, 2020, 卷号: 368, 期号: 6497, 页码: 1331-+
作者:
Dai, Wenhao
;
Zhang, Bing
;
Jiang, Xia-Ming
;
Su, Haixia
;
Li, Jian
  |  
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/12/24
Structure-Activity Relationship of SPOP Inhibitors against Kidney Cancer
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 9, 页码: 4849-4866
作者:
Dong, Ze
;
Wang, Zhen
;
Guo, Zhong-Qiang
;
Gong, Shouzhe
;
Zhang, Tao
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2020/07/01
Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion
期刊论文
OAI收割
ADVANCED SCIENCE, 2020, 页码: 13
作者:
Sun, Zhongya
;
Zhang, Hao
;
Zhang, Yuanyuan
;
Liao, Liping
;
Zhou, Wen
  |  
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2020/07/01
anti-metastasis activities
crystal structures
inhibitors
novel pockets
rho family proteins