中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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  • 2020 [16]
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A Peptide Binder of E3 Ligase Adaptor SPOP Disrupts Oncogenic SPOP-Protein Interactions in Kidney Cancer Cells 期刊论文  OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 274-280
作者:  
Wang, Zhen;  Zhang, Hao;  Chen, Baoen;  Ouyang, Sisheng;  Zheng, Tong
  |  收藏  |  浏览/下载:123/0  |  提交时间:2021/05/24
Structure-based drug optimization and biological evaluation of tetrahydroquinolin derivatives as selective and potent CBP bromodomain inhibitors 期刊论文  OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 22, 页码: 7
作者:  
Bi, Xiaoyang;  Chen, Yu;  Sun, Zhongya;  Lu, Wenchao;  Xu, Pan
  |  收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
Structural basis for activation of the growth hormone-releasing hormone receptor 期刊论文  OAI收割
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  
Zhou, Fulai;  Zhang, Huibing;  Cong, Zhaotong;  Zhao, Li-Hua;  Zhou, Qingtong
  |  收藏  |  浏览/下载:33/0  |  提交时间:2020/12/21
Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 11
作者:  
Chen, Yu;  Bi, Xiaoyang;  Zhang, Fengcai;  Sun, Zhongya;  Xu, Pan
  |  收藏  |  浏览/下载:28/0  |  提交时间:2020/12/24
Discovery of novel USP8 inhibitors via Ubiquitin-Rho-110 fluorometric assay based high throughput screening 期刊论文  OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 9
作者:  
Han, Jie;  Tian, Yucheng;  Yu, Liang;  Zhang, Qilin;  Xu, Xi
  |  收藏  |  浏览/下载:36/0  |  提交时间:2020/12/24
Sorting Nexin 10 Mediates Metabolic Reprogramming of Macrophages in Atherosclerosis Through the Lyn-Dependent TFEB Signaling Pathway 期刊论文  OAI收割
CIRCULATION RESEARCH, 2020, 卷号: 127, 期号: 4, 页码: 534-549
作者:  
You, Yan;  Bao, Wei-Lian;  Zhang, Su-Lin;  Li, Hai-Dong;  Li, Hui
  |  收藏  |  浏览/下载:38/0  |  提交时间:2020/12/24
Structural basis for inhibition of the RNA-dependent RNA polymerase from SARS-CoV-2 by remdesivir 期刊论文  OAI收割
SCIENCE, 2020, 卷号: 368, 期号: 6498, 页码: 1499-+
作者:  
Yin, Wanchao;  Mao, Chunyou;  Luan, Xiaodong;  Shen, Dan-Dan;  Shen, Qingya
  |  收藏  |  浏览/下载:34/0  |  提交时间:2020/12/24
Structure-based design of antiviral drug candidates targeting the SARS-CoV-2 main protease 期刊论文  OAI收割
SCIENCE, 2020, 卷号: 368, 期号: 6497, 页码: 1331-+
作者:  
Dai, Wenhao;  Zhang, Bing;  Jiang, Xia-Ming;  Su, Haixia;  Li, Jian
  |  收藏  |  浏览/下载:41/0  |  提交时间:2020/12/24
Structure-Activity Relationship of SPOP Inhibitors against Kidney Cancer 期刊论文  OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 9, 页码: 4849-4866
作者:  
Dong, Ze;  Wang, Zhen;  Guo, Zhong-Qiang;  Gong, Shouzhe;  Zhang, Tao
  |  收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion 期刊论文  OAI收割
ADVANCED SCIENCE, 2020, 页码: 13
作者:  
Sun, Zhongya;  Zhang, Hao;  Zhang, Yuanyuan;  Liao, Liping;  Zhou, Wen
  |  收藏  |  浏览/下载:78/0  |  提交时间:2020/07/01