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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [223]
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OAI收割 [223]
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期刊论文 [200]
会议论文 [17]
学位论文 [6]
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2023 [6]
2021 [6]
2020 [5]
2019 [8]
2018 [7]
2016 [10]
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Chemistry [13]
Pharmacolo... [9]
Biochemist... [8]
Physics [4]
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浏览/检索结果:
共223条,第1-10条
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专题:上海药物研究所
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Berberine derivative DCZ0358 induce oxidative damage by ROS-mediated JNK signaling in DLBCL cells
期刊论文
OAI收割
INTERNATIONAL IMMUNOPHARMACOLOGY, 2023, 卷号: 125, 页码: 15
作者:
Feng, Qilin
;
Hu, Ke
;
Hu, Huifang
;
Lu, Yumeng
;
Zhang, Hui
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2024/01/16
DLBCL
ROS
DNA damage
JNK
Mitochondrial dysfunction
TI17, a novel compound, exerts anti-MM activity by impairing Trip13 function of DSBs repair and enhancing DNA damage
期刊论文
OAI收割
CANCER MEDICINE, 2023, 页码: 14
作者:
Chang, Shuaikang
;
Xiao, Wenqin
;
Xie, Yongsheng
;
Xu, Zhijian
;
Li, Bo
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/12/11
DNA damage
DSBs repair
myeloma
TI17
Trip13
Advancements and Obstacles of PARP Inhibitors in Gastric Cancer
期刊论文
OAI收割
CANCERS, 2023, 卷号: 15, 期号: 21, 页码: 19
作者:
Chen, Hongjie
;
Hu, Yangchan
;
Zhuang, Zirui
;
Wang, Dingyi
;
Ye, Zu
  |  
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/19
gastric cancer
DNA damage repair
PARP inhibitor
cancer therapy
Design, Construction, and Screening of Diversified Pyrimidine-Focused DNA-Encoded Libraries
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 14, 期号: 8, 页码: 1073-1078
作者:
Seydimemet, Mengnisa
;
Yang, Yixuan
;
Lv, Yuhan
;
Liu, Jiaxiang
;
Yan, Ziqin
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/10/17
DNA-encoded library technology
Pyrimidine-focusedDNA-encodedlibrary
BRD4
Affinity screening
Inhibitor
Privileged heterocycles for DNA-encoded library design and hit-to-lead optimization
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 248, 页码: 26
作者:
Wen, Xin
;
Wu, Xinyuan
;
Jin, Rui
;
Lu, Xiaojie
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/04/10
DNA Encoded library
Drug discovery
Heterocycles
Hit identification
Lead generation
Combined inhibition of PARP and ATR synergistically potentiates the antitumor activity of HER2-targeting antibody-drug conjugate in HER2-positive cancers
期刊论文
OAI收割
AMERICAN JOURNAL OF CANCER RESEARCH, 2023, 卷号: 13, 期号: 1, 页码: 161-+
作者:
Li, Yongpeng
;
Li, Lin
;
Fu, Haoyu
;
Yao, Qing
;
Wang, Lei
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/10/17
Antibody-drug conjugate
DS-8201
PARP
ATR
synergy
DNA damage
Triazine-Based Covalent DNA-Encoded Libraries for Discovery of Covalent Inhibitors of Target Proteins
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 页码: 8
作者:
Li, Linjie
;
Su, Mingbo
;
Lu, Weiwei
;
Song, Hongzhi
;
Liu, Jiaxiang
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/09/30
DNA encoded library
covalent library
library design
covalent inhibitors
Phosphoproteomics Reveals the AMPK Substrate Network in Response to DNA Damage and Histone Acetylation
期刊论文
OAI收割
GENOMICS PROTEOMICS & BIOINFORMATICS, 2022, 卷号: 20, 期号: 4, 页码: 597-613
作者:
Jiang, Yuejing
;
Cong, Xiaoji
;
Jiang, Shangwen
;
Dong, Ying
;
Zhao, Lei
  |  
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2023/04/10
AMPK
Phosphoproteomics
Histone modification
DNA damage
Apoptosis
Preclinical validation and phase I trial of 4-hydroxysalicylanilide, targeting ribonucleotide reductase mediated dNTP synthesis in multiple myeloma
期刊论文
OAI收割
Journal of Biomedical Science, 2022, 卷号: 29, 期号: 1
作者:
Xie,Yongsheng
;
Wang,Yingcong
;
Xu,Zhijian
;
Lu,Yumeng
;
Song,Dongliang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/06/15
4-Hydroxysalicylanilid
Ribonucleotide reductase
Deoxyribonucleotides
DNA damage repair
Multiple myeloma
Aristolochic acids exposure was not the main cause of liver tumorigenesis in adulthood
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 5, 页码: 2252-2267
作者:
Chen, Shuzhen
;
Dong, Yaping
;
Qi, Xinming
;
Cao, Qiqi
;
Luo, Tao
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/08/16
Aristolochic acids (AAs)
Mutational signature
AA-DNA adduct
Hepatocellular carcinoma (HCC)
Liver tumorigenesis
Hepatitis B virus (HBV)
Risk factors
Tumor prevention