中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [31]
采集方式
OAI收割 [31]
内容类型
期刊论文 [31]
发表日期
2023 [31]
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发表日期:2023
专题:上海药物研究所
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A first-in-human phase 1 study of simnotrelvir, a 3CL-like protease inhibitor for treatment of COVID-19, in healthy adult subjects
期刊论文
OAI收割
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2023, 卷号: 191, 页码: 9
作者:
Yang, Xin-Mei
;
Yang, Yang
;
Yao, Bu-Fan
;
Ye, Pan-Pan
;
Xu, Yan
  |  
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2023/12/11
COVID-19
Simnotrelvir
Safety
Pharmacokinetics
Healthy subjects
Glimepiride, a novel soluble epoxide hydrolase inhibitor, protects against heart failure via increasing epoxyeicosatrienoic acids
期刊论文
OAI收割
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2023, 卷号: 185, 页码: 13-25
作者:
Zhao, Chengcheng
;
Jiang, Xiangrui
;
Peng, Liyuan
;
Zhang, Yan
;
Li, Huihui
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2024/01/16
Heart failure
Hypertrophy
Epoxyeicosatrienoic acids
Soluble epoxide hydrolase
Design and synthesis of 1H-pyrazolo[3,4-
d
]pyrimidine derivatives as hematopoietic progenitor kinase 1 (HPK1) inhibitors
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 140, 页码: 18
作者:
Zhang, Junjie
;
Li, Yan
;
Tang, Haotian
;
Zhou, Qianqian
;
Tong, Linjiang
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2023/12/08
Cancer immunotherapy
HPK1
Structure -based design
HPK1 inhibitor
The Cocrystal of Ubiquinol: Improved Stability and Bioavailability
期刊论文
OAI收割
PHARMACEUTICS, 2023, 卷号: 15, 期号: 10, 页码: 12
作者:
Zhang, Qi
;
Xia, Mengyuan
;
Zheng, Chenxuan
;
Yang, Yinghong
;
Bao, Junjie
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2023/12/11
ubiquinol
cocrystal
polymorph
stability
bioavailability
Precolumn derivatization LC-MS/MS method to simultaneous quantitation of 10 monosaccharides in rat plasma
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2023, 卷号: 234, 页码: 10
作者:
Li, Mengxue
;
Li, Ping
;
Ji, Yuting
;
Tian, Yihua
;
Zeng, Huiying
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2023/10/17
LC-MS
MS
Monosaccharides
Derivatization
1-Phenyl-3-methyl-5-pyrazolone (PMP)
Biomarker
AhR-STAT3-HO-1/COX-2 signalling pathway may restrict ferroptosis and improve hMSC accumulation and efficacy in mouse liver
期刊论文
OAI收割
BRITISH JOURNAL OF PHARMACOLOGY, 2023, 页码: 17
作者:
Han, Li
;
Ma, Chenhui
;
Wu, Zhitao
;
Xu, Huiming
;
Li, Hai
  |  
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2023/12/08
aryl hydrocarbon receptor
ferroptosis
iron
ischaemia/reperfusion liver injury
liver disease
mesenchymal stem cells
Human Aha1's N-terminal extension confers it holdase activity in vitro
期刊论文
OAI收割
PROTEIN SCIENCE, 2023, 卷号: 32, 期号: 9, 页码: 15
作者:
Tang, Junying
;
Hu, Huifang
;
Zhou, Chen
;
Zhang, Naixia
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Aha1
holdase activity
intrinsically disordered region
NMR
N-terminal extension
Smilagenin induces expression and epigenetic remodeling of BDNF in alzheimer's disease
期刊论文
OAI收割
PHYTOMEDICINE, 2023, 卷号: 118, 页码: 11
作者:
Yang, Shuangshuang
;
Fan, Lei
;
Zhang, Rui
;
Song, Chenghuan
;
Shi, Jiyun
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2023/10/17
Alzheimer's disease
Brain-derived neurotrophic factor
Histone acetylation
Smilagenin
Undescribed steroidal alkaloids from the bulbs of Fritillaria sinica
期刊论文
OAI收割
PHYTOCHEMISTRY, 2023, 卷号: 213, 页码: 11
作者:
Li, Jia-yuan
;
Wu, Shi-fei
;
An, Ya-ling
;
Yao, Chang-liang
;
Yao, Shuai
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/10/17
Fritillaria sinica
Liliaceae
Zhonghuabeimu
Steroidal alkaloid derivatives
Anti -cancer effect
Anti -oxidation
Anti -inflammation
DZ2002 alleviates corneal angiogenesis and inflammation in rodent models of dry eye disease via regulating STAT3-PI3KAkt-NF-kappa B pathway
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2023, 页码: 14
作者:
Wu, Chun-mei
;
Mao, Jia-wen
;
Zhu, Jin-zhi
;
Xie, Can-can
;
Yao, Jia-ying
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/10/17
dry eye disease
DZ2002
corneal angiogenesis
immunomodulatory function
NF-kappa B
ophthalmic therapy