中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [67]
采集方式
OAI收割 [67]
内容类型
期刊论文 [67]
发表日期
2021 [67]
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共67条,第1-10条
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存缴方式:oaiharvest
发表日期:2021
专题:上海药物研究所
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GLP-1 mimetics as a potential therapy for nonalcoholic steatohepatitis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:
Chen, Yan
;
Xu, Ying-na
;
Ye, Chen-yu
;
Feng, Wen-bo
;
Zhou, Qing-tong
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/06/15
NAFLD
NASH
GLP-1R
GLP-1 mimetics
dual agonists
triple agonists
GPCR
Potent and Selective RIPK1 Inhibitors Targeting Dual-Pockets for the Treatment of Systemic Inflammatory Response Syndrome and Sepsis
期刊论文
OAI收割
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 6
作者:
Yang, Xiangbo
;
Lu, Huimin
;
Xie, Hang
;
Zhang, Binbin
;
Nie, Tianqing
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/01/18
Binding studies
Drug discovery
Necroptosis
RIPK1 inhibitors
Sepsis
GPR84 signaling promotes intestinal mucosal inflammation via enhancing NLRP3 inflammasome activation in macrophages
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhang, Qing
;
Chen, Lin-hai
;
Yang, Hui
;
Fang, You-chen
;
Wang, Si-wei
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2022/01/18
GPR84
medium chain fatty acid receptor
GPCR
inflammatory bowel diseases
ulcerative colitis
NLRP3 inflammasome
macrophages
Advancing COVID-19 diagnosis with privacy-preserving collaboration in artificial intelligence
期刊论文
OAI收割
NATURE MACHINE INTELLIGENCE, 2021, 卷号: 3, 期号: 12, 页码: 1081-1089
作者:
Bai, Xiangd
;
Wang, Hanchen
;
Ma, Liya
;
Xu, Yongchao
;
Gan, Jiefeng
  |  
收藏
  |  
浏览/下载:65/0
  |  
提交时间:2022/01/18
High-Throughput Screening Campaign Identified a Potential Small Molecule RXFP3/4 Agonist
期刊论文
OAI收割
MOLECULES, 2021, 卷号: 26, 期号: 24, 页码: 10
作者:
Lin, Guangyao
;
Feng, Yang
;
Cai, Xiaoqing
;
Zhou, Caihong
;
Shao, Lijun
  |  
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2022/06/15
RXFP3
RXFP4
high-throughput screening
agonist
WNN0109-C011
Structures of the human cholecystokinin receptors bound to agonists and antagonists
期刊论文
OAI收割
NATURE CHEMICAL BIOLOGY, 2021, 卷号: 17, 期号: 12, 页码: 1230-1237
作者:
Zhang, Xuefeng
;
He, Chenglin
;
Wang, Mu
;
Zhou, Qingtong
;
Yang, Dehua
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/03/21
Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site
期刊论文
OAI收割
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 11, 页码: 2444-2452
作者:
Wang, Jiang
;
Yang, Dehua
;
Cheng, Xi
;
Yang, Linlin
;
Wang, Zhaohui
  |  
收藏
  |  
浏览/下载:40/0
  |  
提交时间:2022/01/04
SN38-based albumin-binding prodrug for efficient targeted cancer chemotherapy
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2021, 卷号: 339, 页码: 297-306
作者:
Huang, Ying
;
Wang, Lei
;
Cheng, Zhiyang
;
Yang, Biyu
;
Yu, Jiahui
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/12/01
Antitumour
Chemotherapy
SN38
Drug delivery systems
Albumin
Cryo-EM structures of PI3K alpha reveal conformational changes during inhibition and activation
期刊论文
OAI收割
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 45, 页码: 9
作者:
Liu, Xiao
;
Yang, Su
;
Hart, Jonathan R.
;
Xu, Yingna
;
Zou, Xinyu
  |  
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2022/01/04
phosphoinositide 3-kinase (PI3K)
activation
inhibition
activity-dependent conformational changes
Three new carabrane sesquiterpenoid derivatives from the whole plant of Carpesium abrotanoides L.
期刊论文
OAI收割
CHINESE JOURNAL OF NATURAL MEDICINES, 2021, 卷号: 19, 期号: 11, 页码: 868-873
作者:
Wu Jie-Wei
;
Tang Chun-Ping
;
Yao Sheng
;
Ke Chang-Qiang
;
Ye Yang
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2022/01/18
Sesquiterpenoid dimer
Carpesium abrotanoides L.
Carabrane sesquiterpenoid
Dicarabrol B
Dicarabrol C
11R-hydroxycarabrol