中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [26]
采集方式
OAI收割 [26]
内容类型
期刊论文 [26]
发表日期
2018 [26]
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发表日期:2018
专题:上海药物研究所
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Development and evaluation of a novel series of Nitroxoline-derived BET inhibitors with antitumor activity in renal cell carcinoma
期刊论文
OAI收割
ONCOGENESIS, 2018, 卷号: 7
作者:
Chen, Wei
;
Zhang, Hao
;
Chen, Zhifeng
;
Jiang, Hao
;
Liao, Liping
  |  
收藏
  |  
浏览/下载:108/0
  |  
提交时间:2019/01/08
Synthesis of novel tetrandrine derivatives and their inhibition against NSCLC A549 cells
期刊论文
OAI收割
JOURNAL OF ASIAN NATURAL PRODUCTS RESEARCH, 2018, 卷号: 20, 期号: 11, 页码: 1064-1074
作者:
Yang, Qian-Hao
;
Jiang, Cheng-Shi
;
Jin, Tao
;
Xu, Jin-Fang
;
Qu, Ting-Li
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2020/07/01
Tetrandrine derivatives
non-small cell lung carcinoma
NSCLC A549 cells
anticancer activities
Suzuki-Miyaura reaction
Chemical cocktails enable hepatic reprogramming of human urine-derived cells with a single transcription factor
期刊论文
OAI收割
Acta pharmacologica Sinica, 2018
作者:
Tang, Wei
;
Guo, Ren
;
Shen, Shi-Jun
;
Zheng, Yang
;
Lu, Yu-Ting
  |  
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2019/01/08
Total synthesis of lithospermic acid using Fe-catalyzed Cross-Dehydrogenative-Coupling reaction and Pd-catalyzed ester-directed C-H olefination
期刊论文
OAI收割
TETRAHEDRON, 2018, 卷号: 74, 期号: 40, 页码: 5950-5954
作者:
Zheng, Yong
;
Song, Weibin
;
Zhu, Yefu
;
Wei, Bole
;
Xuan, Lijiang
  |  
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
Total synthesis
Lithospermic acid
Cross-Dehydrogenative-Coupling
C-H olefination
Anti-inflammatory constituents from Perilla frutescens on lipopolysaccharide-stimulated RAW264.7 cells
期刊论文
OAI收割
FITOTERAPIA, 2018, 卷号: 130, 页码: 61-65
作者:
Wang, Xiao-Feng
;
Li, Heng
;
Jiang, Kun
;
Wang, Qi-Qi
;
Zheng, Yan-Hai
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
Perilla frutescens
Lamiaceae
Monoterpenoid
Anti-inflammation
RAW264.7 cell
Targeting Epigenetic Crosstalk as a Therapeutic Strategy for EZH2-Aberrant Solid Tumors
期刊论文
OAI收割
CELL, 2018, 卷号: 175, 期号: 1, 页码: 186-+
作者:
Huang, Xun
;
Yan, Juan
;
Zhang, Min
;
Wang, Yafang
;
Chen, Yi
  |  
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2019/01/08
CUDC-907 displays potent antitumor activity against human pancreatic adenocarcinoma in vitro and in vivo through inhibition of HDAC6 to downregulate c-Myc expression
期刊论文
OAI收割
Acta pharmacologica Sinica, 2018
作者:
Fu, Xu-Hong
;
Zhang, Xiong
;
Yang, Hong
;
Xu, Xiao-Wei
;
Hu, Zong-Long
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
7 beta-Methyl substituent is a structural locus associated with activity cliff for nepenthone analogues
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 14, 页码: 4254-4263
作者:
Sun, Hui-jiao
;
Wang, Yu-hua
;
Yuan, Cong-min
;
Kong, Ling-hui
;
Xu, Xue-jun
  |  
收藏
  |  
浏览/下载:80/0
  |  
提交时间:2019/01/08
7 beta-Methyl-nepenthone analogues
KOR ligands
Concept of hybridization
Opioid receptor binding and functional activities
CTC clusters induced by heparanase enhance breast cancer metastasis
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1326-1337
作者:
Wei, Rong-rui
;
Sun, Dan-ni
;
Yang, Hong
;
Yan, Juan
;
Zhang, Xiong
  |  
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2019/01/08
human breast cancer
CTC clusters
heparanase
metastasis
cell adhesion
adhesion molecules
suspension culture method
Novel Tadalafil Derivatives Ameliorates Scopolamine-Induced Cognitive Impairment in Mice via Inhibition of Acetyicholinesterase (AChE) and Phosphodiesterase 5 (PDE5)
期刊论文
OAI收割
ACS CHEMICAL NEUROSCIENCE, 2018, 卷号: 9, 期号: 7, 页码: 1625-1636
作者:
Ni, Wei
;
Wang, Huan
;
Li, Xiaokang
;
Zheng, Xinyu
;
Wang, Manjiong
  |  
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
Multifunctional agents
AChE inhibitors
PDE5 inhibitors
Alzheimer's disease