中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [30]
采集方式
OAI收割 [30]
内容类型
期刊论文 [30]
发表日期
2020 [30]
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发表日期:2020
专题:上海药物研究所
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Diphyllin Improves High-Fat Diet-Induced Obesity in Mice Through Brown and Beige Adipocytes
期刊论文
OAI收割
FRONTIERS IN ENDOCRINOLOGY, 2020, 卷号: 11, 页码: 13
作者:
Duan, Ya-Nan
;
Ge, Xiang
;
Jiang, Hao-Wen
;
Zhang, Hong-Jie
;
Zhao, Yu
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2021/05/24
diphyllin
obesity
brown adipocyte
differentiation
thermogenesis
V-ATPase
Development of Taccalonolide AJ-Hydroxypropyl-beta-Cyclodextrin Inclusion Complexes for Treatment of Clear Cell Renal-Cell Carcinoma
期刊论文
OAI收割
MOLECULES, 2020, 卷号: 25, 期号: 23, 页码: 14
作者:
Han, Jing
;
Zhang, Siwang
;
Niu, Junxin
;
Zhang, Chunli
;
Dai, Weichen
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
taccalonolide AJ
microtubule stabilizer
hydroxypropyl-β
-cyclodextrin
inclusion complex
clear-cell renal-cell carcinoma
Liquid chromatography-tandem mass spectrometric assay for TPN171 in human plasma
期刊论文
OAI收割
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2020, 卷号: 191, 页码: 8
作者:
Zhang, Mengqi
;
Liu, Haiming
;
He, Jiajin
;
Gui, Yuzhou
;
Qian, Hongjie
  |  
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2020/12/24
TPN171
LC-MS/MS
Human plasma
Protein precipitation
Pyrazolone derivative C29 protects against HFD-induced obesity in mice via activation of AMPK in adipose tissue
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Li, Bo-han
;
Zhang, Mei
;
Duan, Ya-nan
;
Shuai, Lin
;
Jiang, Hao-wen
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2020/12/21
AMP-activated protein kinase
pyrazolone derivative C29
obesity
energy expenditure
thermogenesis
inguinal white adipose tissue
white adipose browning
Design, Synthesis, and Biological Activities of Novel Triazolothiadiazole Derivatives Linked with Amino Side Chain Containing Urea Group as DOT1L Inhibitors
期刊论文
OAI收割
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 8, 页码: 2450-2459
作者:
Liu Na
;
Guo Siqi
;
Liu Junfang
;
Chen Yantao
;
Xu Xiaoming
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/12/24
DOT1L inhibitor
triazolothiadiazole
triazolothiadiazine
nucleophilic substitution
A potent pyrimidinone Axl inhibitor DW17401
期刊论文
OAI收割
CANCER RESEARCH, 2020, 卷号: 80, 期号: 16, 页码: 1
作者:
Zhang, Hefeng
;
Peng, Xia
;
Ji, Yinchun
;
Dai, Yang
;
Shen, Yanyan
  |  
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2021/05/24
Diterpenoids as potential anti-inflammatory agents from Ajuga pantantha
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 9
作者:
Liu, Wenpei
;
Song, Ziteng
;
Wang, Huimei
;
Yang, Xueyuan
;
Joubert, Elizabeth
  |  
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/12/24
Nitric oxide inhibitory effects
Ajuga pantantha
Diterpenoids
Inflammation
Molecular docking
Zebrafish model
Nitric oxide inhibitory iridoids as potential anti-inflammatory agents from Valeriana jatamansi
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 9
作者:
Wang, Huimei
;
Song, Ziteng
;
Xing, Honghong
;
Shi, Zhaoyu
;
Wu, Peng
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2020/12/24
Iridoids
NO inhibitory activities
Valeriana jatamansi
Inflammation
Molecular docking
Anti-SARS-CoV-2 activities in vitro of Shuanghuanglian preparations and bioactive ingredients
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Su, Hai-xia
;
Yao, Sheng
;
Zhao, Wen-feng
;
Li, Min-jun
;
Liu, Jia
  |  
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2020/12/24
SARS-CoV-2
3CL protease
traditional Chinese medicines
Shuanghuanglian oral liquid
baicalin
baicalein
AMPK activator C24 inhibits hepatic lipogenesis and ameliorates dyslipidemia in HFHC diet-induced animal models
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:
Sun, Shui-mei
;
Xie, Zhi-fu
;
Zhang, Yang-ming
;
Zhang, Xin-wen
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2020/12/24
adenosine 5 '-monophosphate-activated protein kinase
AMPK activator
C24
liver
triglycerides
cholesterol
VLDL
hypolipidemic drug
metabolic syndrome