中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [7]
采集方式
OAI收割 [7]
内容类型
期刊论文 [7]
发表日期
2022 [7]
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发表日期:2022
专题:上海药物研究所
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Mass spectrometry imaging: new eyes on natural products for drug research and development
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 16
作者:
Hou, Jin-jun
;
Zhang, Zi-jia
;
Wu, Wen-yong
;
He, Qing-qing
;
Zhang, Teng-qian
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/11/11
natural product
mass spectrometry imaging
MALDI
DESI
molecular imaging
ion mobility
Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 卷号: 240, 页码: 114574
作者:
Kayumov, Muzaffar
;
Jia, Li
;
Pardaev, Azizbek
;
Song, Shan-Shan
;
Mirzaakhmedov, Sharafitdin
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2024/03/21
PARP1
Olaparib
Alantolactone
Syntheticlethality
BRCA1/2mutant
SOMCL-19-133, a novel, selective, and orally available inhibitor of NEDD8-activating enzyme (NAE) for cancer therapy
期刊论文
OAI收割
NEOPLASIA, 2022, 卷号: 32, 页码: 12
作者:
Zhou, Li-Na
;
Xiong, Chaodong
;
Cheng, Yong-Jun
;
Song, Shan-Shan
;
Bao, Xu-Bin
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2023/04/10
SOMCL-19-133
NAE inhibitor
MLN4924
NEDD8
Oral administration
Therapeutic potential of traditional Chinese medicine for the treatment of NAFLD: A promising drug Potentilla discolor Bunge
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 9, 页码: 3529-3547
作者:
Ji, Longshan
;
Li, Qian
;
He, Yong
;
Zhang, Xin
;
Zhou, Zhenhua
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/12/13
Anti-inflammatory
Lipid metabolism
Insulin resistance
Endoplasmic reticulum stress
Intestinal microflora
Nonalcoholic fatty liver disease (NAFLD)
Traditional Chinese medicine
Acupuncture
Potentilla discolor Bunge (PDB)
Natural active compounds
Anti-oxidative
Chemo- and Site-Selective Lysine Modification of Peptides and Proteins under Native Conditions Using the Water-Soluble Zolinium
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2022, 页码: 14
作者:
Sun, Haiguo
;
Xi, Mengyu
;
Jin, Qiang
;
Zhu, Zhengdan
;
Zhang, Yani
  |  
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2022/09/30
Tumour-derived extracellular vesicle membrane hybrid lipid nanovesicles enhance siRNA delivery by tumour-homing and intracellular freeway transportation
期刊论文
OAI收割
JOURNAL OF EXTRACELLULAR VESICLES, 2022, 卷号: 11, 期号: 3, 页码: 16
作者:
Zhou, Xin
;
Miao, Yunqiu
;
Wang, Ying
;
He, Shufang
;
Guo, Linmiao
  |  
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2022/06/15
tumour-derived extracellular vesicles
hybrid lipid nanovesicles
tumour homing
siRNA delivery
hepatocellular carcinoma
Atractylenolide III ameliorates Non-Alcoholic Fatty Liver Disease by activating Hepatic Adiponectin Receptor 1-Mediated AMPK Pathway
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF BIOLOGICAL SCIENCES, 2022, 卷号: 18, 期号: 4, 页码: 1594-1611
作者:
Li, Qian
;
Tan, Jia-Xin
;
He, Yong
;
Bai, Fang
;
Li, Shi-Wei
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2022/06/15
ATL III
AdipoR1
oxidative stress
inflammation
AMPK
SIRT1