中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [16]
采集方式
OAI收割 [16]
内容类型
期刊论文 [16]
发表日期
2022 [16]
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共16条,第1-10条
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发表日期:2022
内容类型:期刊论文
专题:上海药物研究所
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In-situ clickable prodrug nanoplatform locally activates T lymphocytes to potentiate cancer immunotherapy
期刊论文
OAI收割
NANO TODAY, 2022, 卷号: 47, 页码: 11
作者:
Hou, Bo
;
Ye, Jiayi
;
Li, Junhao
;
Xu, Zhiai
;
Yu, Haijun
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2023/04/10
Immune-excluded tumor
Extracellular matrix
In-situ click reaction
Prodrug nanoparticles
Immune resistance
Targeting PI3K alpha overcomes resistance to KRas(G12C) inhibitors mediated by activation of EGFR and/or IGF1R
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 12
作者:
Qi, Wei-liang
;
Li, Hui-yu
;
Wang, Yi
;
Xu, Lan
;
Deng, Jie-ting
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2023/04/10
AMG510
KRas(G12C)
PI3K
drug resistance
combination therapy
Drug Degradation Caused by mce3R Mutations Confers Contezolid (MRX-I) Resistance in Mycobacterium tuberculosis
期刊论文
OAI收割
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2022, 卷号: 66, 期号: 10, 页码: 11
作者:
Pi, Rui
;
Chen, Xiaomin
;
Meng, Jian
;
Liu, Qingyun
;
Chen, Yiwang
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2022/11/11
Mycobacterium tuberculosis
drug resistance
contezolid
Mce3R
Rv1936
degradation
drug resistance mechanisms
Discovery of novel heteroaryl alkynes for highly potent KITD816V cells inhibition to treat gastrointestinal stromal tumors
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 10, 页码: 4004-4007
作者:
Xie, Zhicheng
;
Li, Lin
;
Guo, Yihao
;
Zhang, Mi
;
Chen, Taiwen
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/12/13
KITD816V cells
Mutation
Drug resistance
Gastrointestinal stromal tumors
Therapeutic potential of traditional Chinese medicine for the treatment of NAFLD: A promising drug Potentilla discolor Bunge
期刊论文
OAI收割
ACTA PHARMACEUTICA SINICA B, 2022, 卷号: 12, 期号: 9, 页码: 3529-3547
作者:
Ji, Longshan
;
Li, Qian
;
He, Yong
;
Zhang, Xin
;
Zhou, Zhenhua
  |  
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2022/12/13
Anti-inflammatory
Lipid metabolism
Insulin resistance
Endoplasmic reticulum stress
Intestinal microflora
Nonalcoholic fatty liver disease (NAFLD)
Traditional Chinese medicine
Acupuncture
Potentilla discolor Bunge (PDB)
Natural active compounds
Anti-oxidative
14-Deoxygarcinol improves insulin sensitivity in high-fat diet-induced obese mice via mitigating NF-kappa B/Sirtuin 2-NLRP3-mediated adipose tissue remodeling
期刊论文
OAI收割
ACTA PHARMACOLOGICA SINICA, 2022, 页码: 12
作者:
Chen, Jia-li
;
Feng, Zhe-ling
;
Zhou, Fei
;
Lou, Ruo-han
;
Peng, Cheng
  |  
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/09/30
14-deoxygarcinol
adipose tissue inflammation
insulin resistance
interleukin-1 beta
NLRP3 inflammasome
Sirtuin 2
Concise Total Synthesis of Dysoxylactam A and a Simplified Analog
期刊论文
OAI收割
CHINESE JOURNAL OF CHEMISTRY, 2022, 页码: 8
作者:
Yang, Guan-Zhou
;
Wang, Lei
;
Fan, Yao-Yue
;
Lai, Zeng-Wei
;
Yu, Xue-Ni
  |  
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2022/08/16
Total synthesis
Dysoxylactam A
Macrocyclolipopeptide
Reversing multidrug resistance
Structure-activity relationship
Genome-wide gain-of-function screening identifies EZH2 mediating resistance to PI3K alpha inhibitors in oesophageal squamous cell carcinoma
期刊论文
OAI收割
CLINICAL AND TRANSLATIONAL MEDICINE, 2022, 卷号: 12, 期号: 5, 页码: 17
作者:
Xing, Hui
;
Gao, Mengshi
;
Wang, Yuxiang
;
Zhang, Xu
;
Shi, Jiajie
  |  
收藏
  |  
浏览/下载:47/0
  |  
提交时间:2022/08/16
CDKNIA
cell cycle
CRISPR-SAM
CYH33
ESCC
EZH2
PI3K alpha inhibitor
resistance
Comprehensive Transcriptome Profiling of NAFLD- and NASH-Induced Skeletal Muscle Dysfunction
期刊论文
OAI收割
FRONTIERS IN ENDOCRINOLOGY, 2022, 卷号: 13, 页码: 14
作者:
Guo, Mingwei
;
Xiang, Liping
;
Yao, Jing
;
Zhang, Jun
;
Zhu, Shuangshuang
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2022/08/30
NAFLD
NASH
quadriceps muscle
lipid deposition
insulin resistance
myokines
Design, Synthesis, and Biological Evaluation of Novel EGFR PROTACs Targeting Del19/T790M/C797S Mutation
期刊论文
OAI收割
ACS MEDICINAL CHEMISTRY LETTERS, 2022, 卷号: 13, 期号: 2, 页码: 278-283
作者:
Zhang, Hualin
;
Xie, Ruliang
;
AI-furas, Hawaa
;
Li, Yupeng
;
Wu, Qingxia
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/06/15
NSCLC
acquired resistance
EGFR C797S
PROTACs
selectivity