中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [210]
大连化学物理研究所 [88]
上海营养与健康研究... [48]
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期刊论文 [642]
学位论文 [26]
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2024 [13]
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Discovery of potent PROTAC degraders of Pin1 for the treatment of acute myeloid leukemia
期刊论文
OAI收割
CHEMICAL SCIENCE, 2024, 卷号: 15, 期号: 13, 页码: 5027-5035
作者:
Shi, Yunkai
;
Liu, Minmin
;
Li, Mengna
;
Mao, Yiwen
;
Ma, Jingkun
  |  
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2024/05/07
In vitro inhibition of six active sesquiterpenoids in zedoary turmeric oil on human liver cytochrome P450 enzymes
期刊论文
OAI收割
JOURNAL OF ETHNOPHARMACOLOGY, 2024, 卷号: 322, 页码: 10
作者:
Liu, Suyan
;
Zhao, Yong
;
Tang, Xuan
;
Yang, Junling
;
Pan, Chen
  |  
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2024/02/27
Sesquiterpenoids
Inhibition
CYP450s
Drug-drug interactions
Mechanism
Excessive fatty acids activate PRMT5/MDM2/Drosha pathway to regulate miRNA biogenesis and lipid metabolism
期刊论文
OAI收割
LIVER INTERNATIONAL, 2024, 页码: 17
作者:
Hou, Aijun
;
Xu, Xiaoding
;
Zhang, Yu
;
He, Hongxiu
;
Feng, Yihan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2024/05/07
Drosha degradation
lipid metabolism
miRNA biogenesis
NAFLD
PRMT5
Pharmacokinetics, mass balance, and metabolism of [
14
C]envonalkib (TQ-B3139), a novel ALK tyrosine kinase inhibitor, in healthy Chinese subjects
期刊论文
OAI收割
CANCER CHEMOTHERAPY AND PHARMACOLOGY, 2024, 页码: 11
作者:
Ma, Sheng
;
Wang, Xin
;
Yan, Shu
;
Miao, Liyan
;
Wan, Xiaojing
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2024/05/07
Envonalkib
TQ-B3139
Pharmacokinetics
Mass balance
Excretion
Metabolism
Energy preservation for skeletal muscles: Shenqi Fuzheng injection prevents tissue wasting and restores bioenergetic profiles in a mouse model of chemotherapy-induced cachexia
期刊论文
OAI收割
PHYTOMEDICINE, 2024, 卷号: 125, 页码: 13
作者:
Li, Wei
;
Zhang, Zijia
;
Berik, Entezar
;
Liu, Yawen
;
Pei, Wenqiang
  |  
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2024/04/09
Shenqi Fuzheng injection
Chemotherapy-induce cachexia
Bioenergetic profiles
Glycolysis
TCA cycle
lipid metabolism
Pharmacokinetics and metabolite identification of 23-hydroxybetulinic acid in rats by using liquid chromatography-mass spectrometry method
期刊论文
OAI收割
JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 2024, 卷号: 1234, 页码: 10
作者:
Xue, Mingzhen
;
Yang, Cheng
;
Huang, Wensi
;
He, Yifei
;
Yang, Chen
  |  
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/05/22
23-hydroxybetulinic acid
Pharmacokinetics
Metabolism
UPLC-MS
LC-MS/MS
Turning Threat to Therapy: A Nanozyme-Patch in Surgical Bed for Convenient Tumor Vaccination by Sustained In Situ Catalysis
期刊论文
OAI收割
ADVANCED HEALTHCARE MATERIALS, 2024, 页码: 13
作者:
Wang, Zhaohui
;
Dong, Min
;
Pan, Yuhang
;
Zhang, Lu
;
Lei, Haozhuo
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2024/03/11
biocompatible nanozyme
microneedle patch
postsurgical recurrence
trans-surgical bed
tumor vaccine
Blocking tumor-platelet crosstalk to prevent tumor metastasis via reprograming glycolysis using biomimetic membrane-hybridized liposomes
期刊论文
OAI收割
JOURNAL OF CONTROLLED RELEASE, 2024, 卷号: 366, 页码: 328-341
作者:
Zhu, Jie
;
Wang, Rui
;
Yang, Chenxiao
;
Shao, Xinyue
;
Zhang, Yi
  |  
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2024/03/06
Platelet
Circulating tumor cells (CTCs)
Glycolysis
Metastasis
Hybrid-membrane liposome
Quercetin
Shikonin
Metabolic regulation of homologous recombination repair by MRE11 lactylation
期刊论文
OAI收割
CELL, 2024, 卷号: 187, 期号: 2, 页码: 40
作者:
Chen, Yuping
;
Wu, Jinhuan
;
Zhai, Linhui
;
Zhang, Tingting
;
Yin, Hui
  |  
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2024/04/09
Breathing in danger: Unveiling the link between human exposure to outdoor PM
2.5
-bound polycyclic aromatic hydrocarbons and lung cancer risk in an urban residential area of China
期刊论文
OAI收割
SCIENCE OF THE TOTAL ENVIRONMENT, 2024, 卷号: 907, 页码: 11
作者:
Famiyeh, Lord
;
Xu, Honghui
;
Chen, Ke
;
Tang, Yu-Ting
;
Ji, Dongsheng
  |  
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2024/01/02
Human exposure
Breathing
PAHs
Lung cancer
Urban
Residential area