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Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [100]
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Discovery of YFJ-36: Design, Synthesis, and Antibacterial Activities of Catechol-Conjugated β-Lactams against Gram-Negative Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 21
作者:
Liu, Fangjun
;
Kou, Qunhuan
;
Li, Hongyuan
;
Cao, Yangzhi
;
Chen, Meng
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浏览/下载:0/0
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提交时间:2024/05/22
Design, Synthesis, and Biological Evaluation of Novel Arylomycins against Multidrug-Resistant Gram-Negative Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 页码: 25
作者:
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浏览/下载:0/0
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提交时间:2024/05/22
A Vancomycin-Templated DNA-Encoded Library for Combating Drug-Resistant Bacteria
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 5, 页码: 3778-3794
作者:
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浏览/下载:3/0
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提交时间:2024/05/07
Design, Synthesis, and Anti-tuberculosis Activity of Streptomycin Derivatives
期刊论文
OAI收割
LETTERS IN DRUG DESIGN & DISCOVERY, 2024, 卷号: 21, 期号: 4, 页码: 738-748
作者:
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浏览/下载:8/0
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提交时间:2024/03/06
Multidrug-resistant
hydrazine
hydrazide
sulfonyl hydrazide
siderophore
synthesis
anti-tuberculosis activity
A facile and selective derivatization approach on kynurenine-NH2 in daptomycin, leading to the discovery of hexakynomycin to combat multidrug-resistant Gram-positive pathogens especially daptomycin-resistant bacteria
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 259, 页码: 14
作者:
Guan, Dongliang
;
Li, Jian
;
Chen, Feifei
;
Li, Jiaqi
;
Bian, Xiaolei
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浏览/下载:9/0
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提交时间:2023/10/17
Lipopeptide
Daptomycin derivatives
Multidrug-resistant bacteria
Kynurenine
Hexakynomycin
Resin glycosides from Merremia hederacea with multidrug-resistant reversal activities
期刊论文
OAI收割
PHYTOCHEMISTRY LETTERS, 2023, 卷号: 54, 页码: 14-17
作者:
Li, Chen-Yue
;
Fang, Jie
;
Li, Guang-Yao
;
Wang, Wen-Qiong
;
Xuan, Li-Jiang
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浏览/下载:7/0
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提交时间:2023/10/17
Merremia hederacea
Resin glycoside
Multidrug-resistant reversal activity
Efficient Kilogram-Scale Synthesis of a Novel Oxazolidinone Antibacterial Candidate YG-056SP
期刊论文
OAI收割
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2023, 页码: 12
作者:
Zhang, Yinyong
;
Yang, Yushe
;
Meng, Xin
;
Zhou, Xianli
;
Guo, Bin
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浏览/下载:16/0
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提交时间:2023/04/10
oxazolidinone
asymmetric reduction
fused ring
process development
crystal transformation
Anti-infective therapy using species-specific activators of Staphylococcus aureus ClpP
期刊论文
OAI收割
NATURE COMMUNICATIONS, 2022, 卷号: 13, 期号: 1, 页码: 16
作者:
Wei, Bingyan
;
Zhang, Tao
;
Wang, Pengyu
;
Pan, Yihui
;
Li, Jiahui
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浏览/下载:17/0
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提交时间:2023/04/10
Drug Degradation Caused by mce3R Mutations Confers Contezolid (MRX-I) Resistance in Mycobacterium tuberculosis
期刊论文
OAI收割
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2022, 卷号: 66, 期号: 10, 页码: 11
作者:
Pi, Rui
;
Chen, Xiaomin
;
Meng, Jian
;
Liu, Qingyun
;
Chen, Yiwang
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浏览/下载:27/0
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提交时间:2022/11/11
Mycobacterium tuberculosis
drug resistance
contezolid
Mce3R
Rv1936
degradation
drug resistance mechanisms
Potentiation of Vancomycin: Creating Cooperative Membrane Lysis through a "Derivatization-for-Sensitization" Approach
期刊论文
OAI收割
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2022, 卷号: 144, 期号: 23, 页码: 10622-10639
作者:
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浏览/下载:26/0
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提交时间:2022/08/16