中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
机构
上海药物研究所 [27]
昆明动物研究所 [8]
数学与系统科学研究院 [5]
地质与地球物理研究所 [4]
化学研究所 [4]
青岛生物能源与过程研... [3]
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期刊论文 [65]
会议论文 [1]
学位论文 [1]
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2024 [4]
2023 [5]
2022 [1]
2021 [4]
2020 [6]
2019 [2]
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物理化学 [1]
网络心理学 [1]
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Discovery of CZL-046 with an (
S
)-3-Fluoropyrrolidin-2-one Scaffold as a p300 Bromodomain Inhibitor for the Treatment of Multiple Myeloma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 20, 页码: 18606-18628
作者:
Chen, Zonglong
;
Yang, Hong
;
Zhang, Yan
;
Lyu, Xiaodong
;
Shi, Qiongyu
  |  
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2024/11/05
Development of ketalized unsaturated saccharides as multifunctional cysteine-targeting covalent warheads
期刊论文
OAI收割
COMMUNICATIONS CHEMISTRY, 2024, 卷号: 7, 期号: 1, 页码: 10
作者:
Dong, Sanfeng
;
Huang, Hui
;
Li, Jintian
;
Li, Xiaomei
;
Bunu, Samuel Jacob
  |  
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2024/10/21
Discovery of Novel PROTAC Degraders of p300/CBP as Potential Therapeutics for Hepatocellular Carcinoma
期刊论文
OAI收割
JOURNAL OF MEDICINAL CHEMISTRY, 2024, 卷号: 67, 期号: 4, 页码: 2466-2486
作者:
Chang, Qi
;
Li, Jiayi
;
Deng, Yue
;
Zhou, Ruilin
;
Wang, Bingwei
  |  
收藏
  |  
浏览/下载:36/0
  |  
提交时间:2024/03/25
Design and synthesis of cantharidin derivative DCZ5418 as a TRIP13 inhibitor with anti-multiple myeloma activity
in
vitro
and
in
vivo
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2024, 卷号: 98, 页码: 7
作者:
Dong, Sanfeng
;
Hu, Ke
;
Shi, Yulong
;
Wang, Guanli
;
Yu, Dandan
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2024/02/19
Multiple myeloma
TRIP13 inhibitor
Cantharidin
DCZ5418
DCZ0415
Synthesis, evaluation and molecular dynamics study of human toll-like receptor 2/6 specific monoacyl lipopeptides as candidate immunostimulants
期刊论文
OAI收割
BIOORGANIC CHEMISTRY, 2023, 卷号: 141, 页码: 17
作者:
Zhu, Yueyue
;
Liu, Bo
;
Chen, Zonglong
;
Wang, Xianyang
;
Wang, Yujie
  |  
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2023/12/08
Toll -like receptor 2/6 agonists
PamCS
Structure-activity relationship
Lipopeptide
Immunostimulants
Design, synthesis of auristatins-glucuronide conjugates targeting the β-glucuronidase in tumor microenvironment
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2023, 卷号: 95, 页码: 5
作者:
Wang, Yujie
;
Xu, Keshi
;
Liu, Hongchun
;
Zhang, Wei
;
Hu, Chun
  |  
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2023/12/19
Auristatin E
beta-Glucuronidase
Antiproliferation
Tumor microenvironment
The first record of Lower Cretaceous theropod tracks in Turpan-Hami Basin, Xinjiang, northwestern China
期刊论文
OAI收割
HISTORICAL BIOLOGY, 2023, 页码: 6
作者:
Li, Yang
;
Jiang, Shunxing
;
Yan, Feng
;
Ma, Yingxia
;
Wang, Xiaolin
  |  
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2023/11/02
Theropod tracks
Lower Cretaceous
Hami pterosaur fauna
Turpan-Hami Basin
Xinjiang
Optimization of potent, selective and orally bioavailable biphenyl scaffold as FABP4 inhibitors for anti-inflammation
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2023, 卷号: 253, 页码: 16
作者:
He, Yulong
;
Li, Shunyi
;
Zhu, Yueyue
;
Wang, Yujie
;
Chen, Yuqi
  |  
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2023/10/17
Structure-activity relationship
FABP4 inhibitor
Biphenyl scaffold
Selectivity
Oral bioavailability
Anti-inflammation
Inhibitory activity of a sulfated oligo-porphyran from Pyropia yezoensis against SARS-CoV-2
期刊论文
OAI收割
CARBOHYDRATE POLYMERS, 2023, 卷号: 299, 页码: 9
作者:
Geng, Lihua
;
Zhang, Quanbin
;
Suo, Qishan
;
Wang, Jing
;
Wang, Yingxia
  |  
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2023/01/04
Pyropia yezoensis
Oligo-porphyran
Oligosaccharide
SARS-CoV-2
SPR
Pseudovirus test
Application of Pt loaded graphite felt in SO2-depolarized electrolyzer
期刊论文
OAI收割
INTERNATIONAL JOURNAL OF HYDROGEN ENERGY, 2022, 卷号: 47, 期号: 74, 页码: 31575-31586
作者:
Ma, Xiaoshan
;
Ding, Xifeng
;
Sun, Xinliang
;
Zhang, Ping
;
Wang, Laijun
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2023/02/24
Hydrogen production
Hybrid sulfur (HyS) process
SO2-depolarized electrolysis (SDE)
Pt-loaded graphite felt
Three-dimensional anode