中国科学院机构知识库网格
Chinese Academy of Sciences Institutional Repositories Grid
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CAS IR Grid
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上海药物研究所 [92]
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期刊论文 [245]
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Structural optimization of phthalazine derivatives for anti-HBV activities to improve oral bioavailability
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY, 2025, 卷号: 128, 页码: 10
作者:
Yang, Yurong
;
Xiao, Fuling
;
Zuo, Jianping
;
Yang, Li
;
Hu, Youhong
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
HBV
Capsid assembly modulators
Structural optimization
Oxidative metabolism
Design and synthesis of CDK9/EZH2 dual-target inhibitors to achieve synergistic antitumor effects
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 14
作者:
Tian, Lina
;
Xiao, Jian
;
Zeng, Yanping
;
Li, Yangsha
;
Wei, Aihuan
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
CDK9
EZH2
Dual target inhibitor
DLBCL
Discovery of potent anti-idiopathic pulmonary fibrosis (IPF) agents based on an o-aminopyridinyl alkynyl scaffold
期刊论文
OAI收割
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 294, 页码: 15
作者:
Wang, Yang
;
Fan, Wenhui
;
Guo, Yihao
;
Sun, Li
;
Hu, Youhong
  |  
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2025/08/20
IPF
EMT
Key kinases
Inhibitors
Discovery of novel Ebola entry inhibitors with 1,2,3,4-tetrahydroisoquinoline-3-carboxamide based on (3S,4aS,8aS)-2-(3-amino-2-hydroxypropyl) decahydroisoquinoline-3-carboxamide scaffold
期刊论文
OAI收割
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2025, 卷号: 123, 页码: 4
作者:
Lin, Junzhen
;
Xiao, Fuling
;
Han, Sheng
;
Hu, Youhong
;
Zuo, Jianping
  |  
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2025/06/23
Ebola virus entry inhibitor
Tetrahydroisoquinoline
Spectroastrometry and Reverberation Mapping of Active Galactic Nuclei. II. Measuring Geometric Distances and Black Hole Masses of Four Nearby Quasars
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL, 2025, 卷号: 988, 期号: 1
作者:
Li, Yan-Rong
;
Shangguan, Jinyi
;
Wang, Jian-Min
;
Davies, Ric
;
Santos, Daryl J. D.
  |  
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2025/07/21
Diterpenoids and diarylheptanoids from the fruits of
Alpinia
zerumbet
and their anti-inflammatory activity
期刊论文
OAI收割
FITOTERAPIA, 2025, 卷号: 184, 页码: 10
作者:
Zhang, Zhenghan
;
Li, Guangqian
;
Luo, Xin
;
Xiao, Fang
;
Zhang, Yan
  |  
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2025/08/20
Alpinia zerumbet
Labdane-type diterpenoid
Diarylheptanoid
Anti-inflammatory
ISG pathway
TDDFT ECD calculation
Native Ligand-Inspired peptides for c-MET targeted PET probes development
期刊论文
OAI收割
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2025, 页码: 18
作者:
Luo, Renli
;
Tan, Boyu
;
Zhang, Ying
;
Hu, Jing
;
Lin, Jia
  |  
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2025/08/20
C-MET
Native ligand
HGF
PET/CT imaging
Radiopharmaceuticals
Peptide probes
Multiple flares and asymmetric broad emission lines in a recurring changing-look active galactic nucleus
期刊论文
OAI收割
ASTRONOMY & ASTROPHYSICS, 2025, 卷号: 698
作者:
Guo, Wei-Jian
;
Zhang, Zhi-Xiang
;
Moiseev, Alexei
;
Fawcett, Victoria A.
;
Chen, Yong-Jie
  |  
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2025/06/23
galaxies: active
galaxies: nuclei
quasars: supermassive black holes
Monitoring AGNs with Hβ Asymmetry. V. Long-term Variation and Evolution of the Broad Hβ Emission-line Profiles
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL SUPPLEMENT SERIES, 2025, 卷号: 278, 期号: 2
作者:
Fang, Feng-Na
;
Du, Pu
;
Brotherton, Michael S.
;
McLane, Jacob N.
;
Zastrocky, T. E.
  |  
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2025/06/10
Supermassive Black Holes with High Accretion Rates in Active Galactic Nuclei. XIV. Long-duration High-cadence Reverberation Mapping Results for 11 PG Quasars
期刊论文
OAI收割
ASTROPHYSICAL JOURNAL SUPPLEMENT SERIES, 2025, 卷号: 278, 期号: 2
作者:
Hu, Chen
;
Yao, Zhu-Heng
;
Chen, Yong-Jie
;
Songsheng, Yu-Yang
;
Wang, Yi-Lin
  |  
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2025/06/23